Search Count: 11
![]() |
Crystal Structure Of Glucokinase (Hexokinase 4) Complexed With Ligand Diethyl ({2-[3-(4-Methanesulfonylpheno Xy)-5-{[(2S)-1-Methoxypropan-2-Yl]Oxy}Benzamido]-1,3-Thiaz Ol-4-Yl}Methyl)Phosphonate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2022-03-02 Classification: TRANSFERASE Ligands: GLC, NA, G2T, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-03-02
Ligands: GLC, NA, G2T, EDO
![]() |
Crystal Structure Of Glucokinase (Hexokinase 4) Complexed With Ligand Aka Diethyl {[3-(3-{[5-(Azetidine-1-Carbon Yl)Pyrazin-2-Yl]Oxy}-5-(Propan-2-Yloxy)Benzamido)-1H- Pyrazol-1-Yl]Methyl}Phosphonate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2022-03-02 Classification: TRANSFERASE Ligands: G1S, GLC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-03-02
Ligands: G1S, GLC
![]() |
Crystal Structure Of Human Dipeptidyl Peptidase Iv (Dpp Iv) Complexed With Abt-341, A Cyclohexene-Constrained Phenethylamine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2007-10-09 Classification: HYDROLASE Ligands: KIQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-10-09
Ligands: KIQ
![]() |
Crystal Structure Of Human Dipeptidyl Peptidase Iv (Dppiv) With Pyrrolidine-Constrained Phenethylamine 29G
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2007-09-11 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: DLI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-09-11
Ligands: DLI
![]() |
Crystal Structure Of Rat Dipeptidyl Peptidase (Dppiv) With Thiazole-Based Peptide Mimetic #31
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2007-02-27 Classification: HYDROLASE Ligands: SO4, AIL |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2007-02-27
Ligands: SO4, AIL
![]() |
Crystal Structure Of Human Dipeptidyl Peptidase 4 (Dpp Iv) With Potent Alkynyl Cyanopyrrolidine (Abt-279)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2006-12-12 Classification: HYDROLASE Ligands: AXD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-12-12
Ligands: AXD
![]() |
Crystal Structure Of Human Dipeptidyl Peptidase Iv (Dppiv) Complexed With Cyanopyrrolidine (C5-Pro-Pro) Inhibitor 21Ac
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2006-07-04 Classification: HYDROLASE Ligands: ADF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-07-04
Ligands: ADF
![]() |
Crystal Structure Of Human Dipeptidyl Peptidase Iv (Dppiv) Complexed With Cyanopyrrolidine (C5-Pro-Pro) Inhibitor 21Ag
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2006-07-04 Classification: HYDROLASE Ligands: ACF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-07-04
Ligands: ACF
![]() |
Crystal Structure Of Human Dipeptidyl Peptidase Iv (Dppiv) Complexed With Cyanopyrrolidine (C5-Pro-Pro) Inhibitor 24B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2006-07-04 Classification: HYDROLASE Ligands: AAF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-07-04
Ligands: AAF
![]() |
Oxalyl-Aryl-Amino Benzoic Acid Inhibitors Of Ptp1B, Compound 17
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2003-05-20 Classification: HYDROLASE Ligands: 588 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2003-05-20
Ligands: 588
![]() |
Oxalyl-Aryl-Amino Benzoic Acid Inhibitors Of Ptp1B, Compound 8B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2003-05-20 Classification: HYDROLASE Ligands: 968 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2003-05-20
Ligands: 968
