Search Count: 16
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Crystal Structure Of Hpk1 T165E/S171E In Complex With Compound 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.64 Å Release Date: 2025-02-19 Classification: TRANSFERASE Ligands: A1ITC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-19
Ligands: A1ITC
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Crystal Structure Of Hpk1 T165E/S171E In Complex With Compound 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2025-02-19 Classification: TRANSFERASE Ligands: A1ITA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-19
Ligands: A1ITA
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Crystal Structure Of Hpk1 T165E/S171E In Complex With Pyrazine Carboxamide Inhibitor Az3246 (Compound 24)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.39 Å Release Date: 2025-02-19 Classification: TRANSFERASE Ligands: A1ITB, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-19
Ligands: A1ITB, EDO
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Crystal Structure Of Parp1 Catalytic Domain Bound To Azd5305 (Saruparib)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2024-12-04 Classification: TRANSFERASE Ligands: A1H63, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-04
Ligands: A1H63, SO4
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Crystal Structure Of Parp1 Catalytic Domain Bound To Azd9574
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2024-12-04 Classification: TRANSFERASE Ligands: A1H64, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-04
Ligands: A1H64, SO4
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Crystal Structure Of Cbl-B In Complex With An Allosteric Inhibitor (Compound 31)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.87 Å Release Date: 2024-01-24 Classification: LIGASE Ligands: ZN, NA, WX9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-01-24
Ligands: ZN, NA, WX9
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Crystal Structure Of Cbl-B In Complex With An Allosteric Inhibitor (Compound 9)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.42 Å Release Date: 2024-01-10 Classification: LIGASE Ligands: WUQ, ZN, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-01-10
Ligands: WUQ, ZN, NA
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Crystal Structure Of Cbl-B In Complex With An Allosteric Inhibitor (Compound 8)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2024-01-10 Classification: LIGASE Ligands: WX0, ZN, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-01-10
Ligands: WX0, ZN, NA
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Crystal Structure Of Cbl-B In Complex With An Allosteric Inhibitor (Compound 30)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.52 Å Release Date: 2024-01-10 Classification: LIGASE Ligands: ZN, NA, WUI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-01-10
Ligands: ZN, NA, WUI
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Parp1 Catalytic Domain In Complex With 8-Chloroquinazolinone-Based Inhibitor (Compound 9)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2021-09-15 Classification: TRANSFERASE Ligands: VKW, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-15
Ligands: VKW, SO4
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Parp1 Catalytic Domain In Complex With Isoquinolone-Based Inhibitor (Compound 16)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2021-09-15 Classification: TRANSFERASE Ligands: VKT, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-15
Ligands: VKT, SO4
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Parp1 Catalytic Domain In Complex With A Selective Pyridine Carboxamide-Based Inhibitor (Compound 22)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2021-09-15 Classification: TRANSFERASE Ligands: VKQ, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-15
Ligands: VKQ, SO4
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Human Glutamate Carboxypeptidase Ii In Complex With Antibody- Recruiting Molecule Arm-P8
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2010-09-08 Classification: HYDROLASE Ligands: AR8, ZN, CA, CL, NAG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-09-08
Ligands: AR8, ZN, CA, CL, NAG
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Human Glutamate Carboxypeptidase Ii In Complex With Antibody- Recruiting Molecule Arm-P4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2010-09-08 Classification: HYDROLASE Ligands: ZN, CA, CL, NAG, CI9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-09-08
Ligands: ZN, CA, CL, NAG, CI9
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Human Glutamate Carboxypeptidase Ii In Complex With Antibody- Recruiting Molecule Arm-P2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2010-09-08 Classification: HYDROLASE Ligands: ZN, CA, CL, NAG, ARK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-09-08
Ligands: ZN, CA, CL, NAG, ARK
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Human Glutamate Carboxypeptidase Ii In Complex With Arm-M4, Urea- Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.78 Å Release Date: 2010-09-08 Classification: HYDROLASE Ligands: ZN, CA, CL, NAG, OKD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-09-08
Ligands: ZN, CA, CL, NAG, OKD
