Search Count: 20
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Crystal Structure Of Rar-Related Orphan Receptor C (Nhis-Rorgt(244-487)-L6-Src1(678-692) In Complex With A Novel Tricyclic-Carbocylic Rorgt Inverse Agonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2021-02-24 Classification: TRANSCRIPTION/Agonist Ligands: Z8G |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-02-24
Ligands: Z8G
 |
Crystal Structure Of Rar-Related Orphan Receptor C (Nhis-Rorgt(244-487)-L6-Src1(678-692)) In Complex With {3,5-Dichloro-4-[4-Methoxy-3-(Propan-2-Yl)Phenoxy]Phenyl}Methanol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.62 Å Release Date: 2021-01-20 Classification: TRANSFERASE/Agonist Ligands: Z7G |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-20
Ligands: Z7G
 |
Crystal Structure Of Rar-Related Orphan Receptor C (Nhis-Rorgt(244-487)-L6-Src1(678-692)) In Complex With {3,5-Dichloro-4-[4-Methoxy-3-(Propan-2-Yl)Phenoxy]Phenyl}Methanol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.42 Å Release Date: 2021-01-20 Classification: TRANSFERASE/Agonist Ligands: Z7H |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-20
Ligands: Z7H
 |
Crystal Structure Of Rar-Related Orphan Receptor C (Nhis-Rorgt(244-487)-L6-Src1(678-692)) In Complex With {3,5-Dichloro-4-[4-Methoxy-3-(Propan-2-Yl)Phenoxy]Phenyl}Methanol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.14 Å Release Date: 2021-01-20 Classification: TRANSFERASE/Agonist Ligands: Z7I |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-20
Ligands: Z7I
 |
Crystal Structure Of Rar-Related Orphan Receptor C (Nhis-Rorgt(244-487)-L6-Src1(678-692)) In Complex With A Tricyclic Sulfone Inverse Agonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.05 Å Release Date: 2020-11-25 Classification: DNA BINDING PROTEIN/Agonist Ligands: Z8I |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-11-25
Ligands: Z8I
 |
Crystal Structure Of Rar-Related Orphan Receptor C (Nhis-Rorgt(244-487)-L6-Src1(6T78-692) In Complex With A Tricyclic Sulfone Rorgt Inverse Agonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.43 Å Release Date: 2020-09-16 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: VK7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-09-16
Ligands: VK7
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Crystal Structure Of Rar-Related Orphan Receptor C In Complex With A Novel Inverse Agonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2020-08-12 Classification: TRANSCRIPTION/Agonist Ligands: V27 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-08-12
Ligands: V27
 |
Crystal Structure Of Rar-Related Orphan Receptor C In Complex With A Potent, Selective And Orally Bioavailable Ror-Gamma-T Inverse Agonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.37 Å Release Date: 2020-08-12 Classification: TRANSCRIPTION/AGONIST Ligands: VBG, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-08-12
Ligands: VBG, SO4
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Substituted Benzyloxytricyclic Compounds As Retinoic Acid-Related Orphan Receptor Gamma T Agonists
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.26 Å Release Date: 2020-06-17 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: Z7F |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-06-17
Ligands: Z7F
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Substituted Benzyloxytricyclic Compounds As Retinoic Acid-Related Orphan Receptor Gamma T Agonists
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2020-04-29 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: TKJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-29
Ligands: TKJ
 |
Substituted Benzyloxytricyclic Compounds As Retinoic Acid-Related Orphan Receptor Gamma T Agonists
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.61 Å Release Date: 2020-04-29 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: Z7D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-29
Ligands: Z7D
 |
Crystal Structure Of Rar-Related Orphan Receptor C (Nhis-Rorgt(244- 487)-L6-Src1(678-692)) In Complex With An Inverse Agonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2020-04-08 Classification: TRANSCRIPTION Ligands: R7V, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-08
Ligands: R7V, GOL
 |
Structure Of Human Pregnane X Receptor Ligand Binding Domain Bound Tethered With Src Co-Activator Peptide And Compound-3 Aka 1,1,1,3,3,3-Hexafluoro-2-{4-[1-(4- Luorobenzenesulfonyl)Cyclopentyl]Phenyl}Propan-2-Ol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.27 Å Release Date: 2020-02-12 Classification: TRANSFERASE Ligands: L7D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-02-12
Ligands: L7D
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Crystal Structure Of Rar-Related Orphan Receptor C (Nhis- Rorgt(244-487)-L6-Src1(678-692)) In Complex With A Tricyclic Inverse Agonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.61 Å Release Date: 2019-11-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: O5B, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-06
Ligands: O5B, GOL
 |
Crystal Structure Of Rar-Related Orphan Receptor C (Nhis-Rorgt(244-487)-L6-Src1(678-692)) In Complex With A Phenyl (3-Phenylpyrrolidin-3-Yl)Sulfone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2019-07-17 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: O5A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-17
Ligands: O5A
 |
Crystal Structure Of Rar-Related Orphan Receptor C In Complex With A Phenyl (3-Phenylpyrrolidin-3-Yl)Sulfone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.29 Å Release Date: 2019-03-20 Classification: TRANSCRIPTION/INHIBITOR Ligands: L8A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-03-20
Ligands: L8A
 |
Identification Of Bicyclic Hexafluoroisopropyl Alcohol Sulfonamides As Rorgt/Rorc Inverse Agonists
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2017-12-20 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: XGH, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-20
Ligands: XGH, SO4
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Structure Of Human Pregnane X Receptor Ligand Binding Domain Bound Tethered With Src Co-Activator Peptide And Compound 25A Aka Bicyclic Hexafluoroisopropyl 2 Alcohol Sulfonamides
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.56 Å Release Date: 2017-12-20 Classification: NUCLEAR PROTEIN Ligands: XGH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-20
Ligands: XGH
 |
Crystal Structure Of Pi3K Delta In Complex With A Trifluoro-Ethyl-Pyrazol-Pyrolotriazine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2017-06-07 Classification: TRANSFERASE/TRANSFERASE REGULATOR Ligands: 9EM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-07
Ligands: 9EM
 |
Crystal Structure Of The Human Pxr-Lbd In Complex With N-{(2R)-1-[(4S)-4-(4-Chlorophenyl)-4-Hydroxy-3,3-Dimethylpiperidin-1-Yl]-3-Methyl-1-Oxobutan-2-Yl}-3-Hydroxy-3-Methylbutanamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2014-08-27 Classification: TRANSCRIPTION/TRANSCRIPTION inhibitor Ligands: 2Q4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-08-27
Ligands: 2Q4, GOL