Search Count: 17
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Crystal Structure Of Gdp-Bound Human M-Ras Protein In Crystal Form I
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.96 Å Release Date: 2024-09-11 Classification: HYDROLASE Ligands: MG, GDP, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-09-11
Ligands: MG, GDP, GOL
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Crystal Structure Of Gdp-Bound Human M-Ras Protein In Crystal Form Ii
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.27 Å Release Date: 2024-09-11 Classification: HYDROLASE Ligands: MG, GDP, PGE, PG4, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-09-11
Ligands: MG, GDP, PGE, PG4, PEG
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Crystal Structure Of Human Ptpn2 Catalytic Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2024-09-04 Classification: HYDROLASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-09-04
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Crystal Structure Of Human Ptpn2 In Complex With Active Site Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.36 Å Release Date: 2024-09-04 Classification: HYDROLASE/INHIBITOR Ligands: 527 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-09-04
Ligands: 527
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Crystal Structure Of Human Ptpn2 In Complex With Allosteric Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.43 Å Release Date: 2024-09-04 Classification: HYDROLASE/INHIBITOR Ligands: FRJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-09-04
Ligands: FRJ
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Crystal Structure Of Mutant Cmet D1228N Kinase Domain In Complex With Inhibitor Compound 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2024-08-21 Classification: SIGNALING PROTEIN Ligands: GOL, A1ATS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-08-21
Ligands: GOL, A1ATS
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Crystal Structure Of Non-Receptor Protein Tyrosine Phosphatase Shp2 In Complex With Pf-07284892
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.06 Å Release Date: 2024-05-29 Classification: HYDROLASE/INHIBITOR Ligands: A1AQ1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-05-29
Ligands: A1AQ1
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Akt1 With Amp-Pnp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2012-05-23 Classification: TRANSFERASE Ligands: ANP, MN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-05-23
Ligands: ANP, MN
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Akt1 With Gdc0068
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2012-05-23 Classification: TRANSFERASE Ligands: 0RF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-05-23
Ligands: 0RF
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Human B-Raf Kinase Domain In Complex With An Bromopyridine Benzamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.40 Å Release Date: 2011-10-05 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: TV4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-05
Ligands: TV4
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Human B-Raf Kinase Domain In Complex With A Methoxypyrazolopyridinyl Benzamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.30 Å Release Date: 2011-10-05 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: B0R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-05
Ligands: B0R
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Spirocyclic Sulfonamides As Akt Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2011-04-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SM9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-04-06
Ligands: SM9
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Spirochromane Akt Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2011-03-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SMH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-30
Ligands: SMH
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Spirochromane Akt Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2011-03-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SMR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-30
Ligands: SMR
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Discovery Of Dihydrothieno- And Dihydrofuropyrimidines As Potent Pan Akt Inhibitors
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2010-11-10 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: SMY |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2010-11-10
Ligands: SMY
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Discovery Of Dihydrothieno- And Dihydrofuropyrimidines As Potent Pan Akt Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2010-11-10 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: SMY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-11-10
Ligands: SMY
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Crystal Structure Of Human Akt1 With An Allosteric Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2010-10-13 Classification: TRANSFERASE Ligands: IQO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-10-13
Ligands: IQO
