Search Count: 23
![]() |
E3 Ligase Cbl-B In Complex With A Triazolone Core Inhibitor (Compound 1)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.79 Å Release Date: 2024-07-31 Classification: LIGASE Ligands: A1IEW, ZN, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-07-31
Ligands: A1IEW, ZN, NA
![]() |
E3 Ligase Cbl-B In Complex With A Lactam Scaffold Inhibitor (Compound 7)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2024-07-31 Classification: LIGASE Ligands: A1IEV, ZN, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-07-31
Ligands: A1IEV, ZN, NA
![]() |
E3 Ligase Cbl-B In Complex With A Carbamate Scaffold Inhibitor (Compound 12)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.56 Å Release Date: 2024-07-31 Classification: LIGASE Ligands: A1IE5, ZN, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-07-31
Ligands: A1IE5, ZN, NA
![]() |
Crystal Structure Of Mgat5 (Alpha-1,6-Mannosylglycoprotein 6-Beta-N-Acetylglucosaminyltransferase V) Luminal Domain With A Lys329-Ile345 Loop Truncation, In Complex With 3D Fragment 2548
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.89 Å Release Date: 2024-02-21 Classification: CARBOHYDRATE Ligands: EDO, UE0, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-02-21
Ligands: EDO, UE0, SO4
![]() |
Crystal Structure Of Cbl-B In Complex With An Allosteric Inhibitor (Compound 31)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.87 Å Release Date: 2024-01-24 Classification: LIGASE Ligands: ZN, NA, WX9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-01-24
Ligands: ZN, NA, WX9
![]() |
Crystal Structure Of Cbl-B In Complex With An Allosteric Inhibitor (Compound 9)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.42 Å Release Date: 2024-01-10 Classification: LIGASE Ligands: WUQ, ZN, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-01-10
Ligands: WUQ, ZN, NA
![]() |
Crystal Structure Of Cbl-B In Complex With An Allosteric Inhibitor (Compound 8)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2024-01-10 Classification: LIGASE Ligands: WX0, ZN, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-01-10
Ligands: WX0, ZN, NA
![]() |
Crystal Structure Of Cbl-B In Complex With An Allosteric Inhibitor (Compound 30)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.52 Å Release Date: 2024-01-10 Classification: LIGASE Ligands: ZN, NA, WUI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-01-10
Ligands: ZN, NA, WUI
![]() |
Crystal Structure Of The E3 Ubiquitin Ligase Cbl-B With An Allosteric Inhibitor (Benzodiazepine Hts Hit Compound 1)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2023-11-22 Classification: LIGASE Ligands: W89, ZN, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-22
Ligands: W89, ZN, NA
![]() |
Crystal Structure Of The E3 Ubiquitin Ligase Cbl-B With An Allosteric Inhibitor (Wo2020264398 Ex23)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2023-11-22 Classification: LIGASE Ligands: Z3N, ZN, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-22
Ligands: Z3N, ZN, NA
![]() |
Crystal Structure Of The E3 Ubiquitin Ligase Cbl-B With An Allosteric Inhibitor (Benzodiazepine Compound 25)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.48 Å Release Date: 2023-11-22 Classification: LIGASE Ligands: W7R, ZN, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-22
Ligands: W7R, ZN, NA
![]() |
Human Gls In Complex With Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2023-01-18 Classification: HYDROLASE Ligands: SO4, 04A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-01-18
Ligands: SO4, 04A
![]() |
Human Gls In Complex With Compound 12
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.38 Å Release Date: 2023-01-18 Classification: HYDROLASE Ligands: R90 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-01-18
Ligands: R90
![]() |
Human Gls In Complex With Compound 18
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.78 Å Release Date: 2023-01-18 Classification: HYDROLASE Ligands: SO4, 5XX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-01-18
Ligands: SO4, 5XX
![]() |
Human Gls In Complex With Compound 27
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2023-01-18 Classification: HYDROLASE Ligands: SO4, R0C |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-01-18
Ligands: SO4, R0C
![]() |
Irak4 In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.44 Å Release Date: 2020-10-28 Classification: SIGNALING PROTEIN Ligands: NBK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-10-28
Ligands: NBK
![]() |
Irak4 In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2020-10-28 Classification: SIGNALING PROTEIN Ligands: N9Z |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-10-28
Ligands: N9Z
![]() |
Irak4 In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.38 Å Release Date: 2020-10-28 Classification: SIGNALING PROTEIN Ligands: NB5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-10-28
Ligands: NB5
![]() |
Irak4 In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.32 Å Release Date: 2020-10-28 Classification: SIGNALING PROTEIN Ligands: NBW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-10-28
Ligands: NBW
![]() |
Irak4 In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.52 Å Release Date: 2020-10-28 Classification: SIGNALING PROTEIN Ligands: ND2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-10-28
Ligands: ND2
