Search Count: 75
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Highly Optimized Cns Penetrant Inhibitors Of Egfr Exon20 Insertion Mutations
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.42 Å Release Date: 2025-02-12 Classification: SIGNALING PROTEIN Ligands: A1IZ7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-12
Ligands: A1IZ7
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Highly Optimized Cns Penetrant Inhibitors Of Egfr Exon20 Insertion Mutations
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.91 Å Release Date: 2025-02-12 Classification: SIGNALING PROTEIN Ligands: A1IZ8, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-12
Ligands: A1IZ8, SO4
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Highly Optimized Cns Penetrant Inhibitors Of Egfr Exon20 Insertion Mutations
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2025-02-12 Classification: SIGNALING PROTEIN Ligands: A1IZ9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-12
Ligands: A1IZ9
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Highly Optimized Cns Penetrant Inhibitors Of Egfr Exon20 Insertion Mutations
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.22 Å Release Date: 2025-02-12 Classification: SIGNALING PROTEIN Ligands: Q6K, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-12
Ligands: Q6K, SO4
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Highly Optimized Cns Penetrant Inhibitors Of Egfr Exon20 Insertion Mutations. Compound 51 Bound To Egfrinsnpg [V948R]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2025-02-05 Classification: SIGNALING PROTEIN Ligands: A1IUK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-05
Ligands: A1IUK
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Crystal Structure Of Menin In Complex With Inhibitor Compound 15
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2025-01-15 Classification: PROTEIN BINDING/INHIBITOR Ligands: A1AVE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-15
Ligands: A1AVE
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Crystal Structure Of Menin In Complex With Inhibitor Compound 26
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2025-01-15 Classification: PROTEIN BINDING/INHIBITOR Ligands: A1AVF, K, EPE, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-15
Ligands: A1AVF, K, EPE, SO4
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Crystal Structure Of Menin In Complex With Inhibitor Compound 20
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2025-01-15 Classification: PROTEIN BINDING/INHIBITOR Ligands: A1AVG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-15
Ligands: A1AVG
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Optimisation Of Potent, Efficacious, Selective And Blood-Brain Barrier Penetrating Inhibitors Targeting Egfr Exon20 Insertion Mutations
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.44 Å Release Date: 2024-11-06 Classification: SIGNALING PROTEIN Ligands: A1H7N, IOD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-11-06
Ligands: A1H7N, IOD
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Optimisation Of Potent, Efficacious, Selective And Blood-Brain Barrier Penetrating Inhibitors Targeting Egfr Exon20 Insertion Mutations
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.02 Å Release Date: 2024-10-16 Classification: SIGNALING PROTEIN Ligands: A1H7O |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-16
Ligands: A1H7O
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Crystal Structure Of Human Ptpn2 Catalytic Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2024-09-04 Classification: HYDROLASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-09-04
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Crystal Structure Of Human Ptpn2 In Complex With Active Site Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.36 Å Release Date: 2024-09-04 Classification: HYDROLASE/INHIBITOR Ligands: 527 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-09-04
Ligands: 527
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Crystal Structure Of Human Ptpn2 In Complex With Allosteric Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.43 Å Release Date: 2024-09-04 Classification: HYDROLASE/INHIBITOR Ligands: FRJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-09-04
Ligands: FRJ
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Cryo-Em Structure Of Spike Glycoprotein From Civet Coronavirus Sz3 In Closed Conformation
Organism: Civet sars cov sz3/2003
Method: ELECTRON MICROSCOPY Release Date: 2024-05-15 Classification: VIRAL PROTEIN Ligands: NAG, EIC |
Organism: Civet sars cov sz3/2003
Method: ELECTRON MICROSCOPY
Release Date: 2024-05-15
Ligands: NAG, EIC
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Cryo-Em Structure Of Spike Glycoprotein From Bat Coronavirus Wiv1 In Closed Conformation
Organism: Bat sars-like coronavirus wiv1
Method: ELECTRON MICROSCOPY Release Date: 2024-05-01 Classification: VIRAL PROTEIN Ligands: NAG, EIC |
Organism: Bat sars-like coronavirus wiv1
Method: ELECTRON MICROSCOPY
Release Date: 2024-05-01
Ligands: NAG, EIC
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Cryo-Em Structure Of Spike Glycoprotein From Civet Coronavirus 007 In Closed Conformation
Organism: Civet sars cov 007/2004
Method: ELECTRON MICROSCOPY Release Date: 2024-05-01 Classification: VIRAL PROTEIN Ligands: NAG, EIC |
Organism: Civet sars cov 007/2004
Method: ELECTRON MICROSCOPY
Release Date: 2024-05-01
Ligands: NAG, EIC
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Crystal Structure Of Lymantria Dispar Cpv14 Polyhedra 14 Crystals
Organism: Lymantria dispar
Method: X-RAY DIFFRACTION Resolution:1.34 Å Release Date: 2023-11-08 Classification: VIRAL PROTEIN Ligands: GTP, MG |
Organism: Lymantria dispar
Method: X-RAY DIFFRACTION
Release Date: 2023-11-08
Ligands: GTP, MG
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Crystal Structure Of Lymantria Dispar Cpv14 Polyhedra Single Crystal
Organism: Lymantria dispar
Method: X-RAY DIFFRACTION Resolution:1.30 Å Release Date: 2023-11-08 Classification: VIRAL PROTEIN Ligands: GTP, MG |
Organism: Lymantria dispar
Method: X-RAY DIFFRACTION
Release Date: 2023-11-08
Ligands: GTP, MG
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Estrogen Receptor Alpha In Complex With Compound 29
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.68 Å Release Date: 2023-02-01 Classification: TRANSCRIPTION Ligands: H09 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-02-01
Ligands: H09
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Oestrogen Receptor Ligand Binding Domain In Complex With Compound 38
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2023-02-01 Classification: GENE REGULATION Ligands: GZI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-02-01
Ligands: GZI
