Search Count: 19
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Discovery Of Mk-8353: An Orally Bioavailable Dual Mechanism Erk Inhibitor For Oncology
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2018-08-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, G67 |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2018-08-08
Ligands: SO4, G67
 |
Discovery Of 3(S)-Thiomethyl Pyrrolidine Erk Inhibitors For Oncology
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2018-05-23 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: SO4, F8V |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2018-05-23
Ligands: SO4, F8V
 |
Discovery Of Novel, Dual Mechanism Erk Inhibitors By Affinity Selection Screening Of An Inactive Kinase State
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2014-11-12 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3G7, SO4 |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2014-11-12
Ligands: 3G7, SO4
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Modulating The Interaction Between Cdk2 And Cyclin A With A Quinoline-Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2013-11-27 Classification: transferase/transferase inhibitor Ligands: 2KD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-11-27
Ligands: 2KD
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Crystal Structure Of Cyclin-Dependent Kinase 2 With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2008-01-22 Classification: TRANSFERASE Ligands: SC8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-01-22
Ligands: SC8
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Crystal Structure Of Cyclin-Dependent Kinase 2 With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2008-01-22 Classification: TRANSFERASE Ligands: SC9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-01-22
Ligands: SC9
 |
Crystal Structure Of Cyclin-Dependent Kinase 2 With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2008-01-22 Classification: TRANSFERASE Ligands: SCE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-01-22
Ligands: SCE
 |
Crystal Structure Of Cyclin-Dependent Kinase 2 With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.28 Å Release Date: 2008-01-22 Classification: TRANSFERASE Ligands: SCF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-01-22
Ligands: SCF
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Crystal Structure Of Cyclin-Dependent Kinase 2 With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2008-01-22 Classification: TRANSFERASE Ligands: SCJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-01-22
Ligands: SCJ
 |
Crystal Structure Of Cyclin-Dependent Kinase 2 With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2008-01-22 Classification: TRANSFERASE Ligands: SCQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-01-22
Ligands: SCQ
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Crystal Structure Of Cyclin-Dependent Kinase 2 With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2008-01-22 Classification: TRANSFERASE Ligands: SCW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-01-22
Ligands: SCW
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Crystal Structure Of Cyclin-Dependent Kinase 2 With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2008-01-22 Classification: TRANSFERASE Ligands: SCX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-01-22
Ligands: SCX
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Crystal Structure Of Cyclin-Dependent Kinase 2 With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2008-01-22 Classification: TRANSFERASE Ligands: SCZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-01-22
Ligands: SCZ
 |
Crystal Structure Of Cyclin-Dependent Kinase 2 With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2008-01-22 Classification: TRANSFERASE Ligands: 2SC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-01-22
Ligands: 2SC
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Crystal Structure Of Cyclin-Dependent Kinase 2 With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.66 Å Release Date: 2008-01-22 Classification: TRANSFERASE Ligands: 3SC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-01-22
Ligands: 3SC
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Crystal Structure Of Cyclin-Dependent Kinase 2 With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.35 Å Release Date: 2008-01-22 Classification: TRANSFERASE Ligands: 5SC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-01-22
Ligands: 5SC
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Crystal Structure Of Cyclin-Dependent Kinase 2 With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.47 Å Release Date: 2008-01-22 Classification: TRANSFERASE Ligands: 6SC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-01-22
Ligands: 6SC
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Structure Of Fpt Bound To The Inhibitor Sch66336
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2003-10-21 Classification: transferase/transferase inhibitor Ligands: ZN, FPP, 336 |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2003-10-21
Ligands: ZN, FPP, 336
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Structure Of Rat Farnesyl Protein Transferase Complexed With A Cvim Peptide And Alpha-Hydroxyfarnesylphosphonic Acid.
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 1999-06-18 Classification: TRANSFERASE Ligands: ACT, ZN, HFP |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 1999-06-18
Ligands: ACT, ZN, HFP