Search Count: 17
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Sarm1 Tir Domain In Complex With Compound 7-Adpr
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.13 Å Release Date: 2025-12-24 Classification: HYDROLASE Ligands: A1IW3, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-12-24
Ligands: A1IW3, EDO
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Sarm1 Tir Domain In Complex With Compound 7-Adpr
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.73 Å Release Date: 2025-12-24 Classification: HYDROLASE Ligands: A1IWL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-12-24
Ligands: A1IWL
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Sarm1 Tir Domain In Complex With Compound 28-Adpr
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2025-12-24 Classification: HYDROLASE Ligands: A1IWN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-12-24
Ligands: A1IWN
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Crystal Structure Of Human Pyruvate Dehydrogenase Kinase Isoform 1 In Complex With Atp Competitive Inhibitor 29
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.14 Å Release Date: 2025-06-25 Classification: TRANSFERASE Ligands: SO4, TF3, EDO, GOL, A1EQH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-06-25
Ligands: SO4, TF3, EDO, GOL, A1EQH
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Crystal Structure Of Human Pyruvate Dehydrogenase Kinase Isoform 2 In Complex With Atp Competitive Inhibitor 24
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.92 Å Release Date: 2025-06-25 Classification: TRANSFERASE Ligands: EDO, TF3, GOL, A1EQJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-06-25
Ligands: EDO, TF3, GOL, A1EQJ
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Crystal Structure Of Human Pyruvate Dehydrogenase Kinase Isoform 2 In Complex With Atp Competitive Inhibitor 22
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.08 Å Release Date: 2025-06-11 Classification: TRANSFERASE Ligands: TF3, A1EQI, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-06-11
Ligands: TF3, A1EQI, DMS
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Crystal Structure Of Human Pyruvate Dehydrogenase Kinase Isoform 1 In Complex With Atp Competitive Inhibitor 8
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.76 Å Release Date: 2025-04-02 Classification: TRANSFERASE Ligands: K, A1EMR, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-04-02
Ligands: K, A1EMR, GOL
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Crystal Structure Of Human Pyruvate Dehydrogenase Kinase Isoform 1 In Complex With Atp Competitive Inhibitor 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.01 Å Release Date: 2025-04-02 Classification: TRANSFERASE Ligands: K, SZ6, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-04-02
Ligands: K, SZ6, GOL
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6-Phenyl-1H-Imidazo[4,5-C]Pyridine-4-Carbonitrile As Cathepsin S Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2011-04-06 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: EF3, DMS, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-04-06
Ligands: EF3, DMS, SO4
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Cathepsin K Covalently Bound To A Cyano-Pyrimidine Inhibitor With Improved Selectivity Over Herg
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2011-03-30 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: O47 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-30
Ligands: O47
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Cathepsin S In Complex With A Covalent Inhibitor With An Aldehyde Warhead
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.49 Å Release Date: 2010-12-22 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: O64, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-12-22
Ligands: O64, DMS
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Cathepsin K In Complex With A Covalent Inhibitor With A Ketoamide Warhead
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.02 Å Release Date: 2010-12-22 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: O96, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-12-22
Ligands: O96, SO4
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Cathepsin K Covalently Bound To A 2-Cyano Pyrimidine Inhibitor With A Benzyl P3 Group.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2010-10-06 Classification: HYDROLASE Ligands: SO4, O75 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-10-06
Ligands: SO4, O75
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4-(3-Trifluoromethylphenyl)-Pyrimidine-2-Carbonitrile As Cathepsin S Inhibitors: N3, Not N1 Is Critically Important
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2010-07-14 Classification: HYDROLASE Ligands: PEG, DMS, 935, 93N, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-07-14
Ligands: PEG, DMS, 935, 93N, SO4, GOL
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X-Ray Structure Of Cathepsin K Covalently Bound To A Triazine Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2010-03-02 Classification: HYDROLASE Ligands: ORG, TFA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-03-02
Ligands: ORG, TFA
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Cathepsin K In Complex With A Non-Selective 2-Cyano-Pyrimidine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.49 Å Release Date: 2010-03-02 Classification: HYDROLASE Ligands: SO4, KWZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-03-02
Ligands: SO4, KWZ
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Cathepsin K In Complex With A Selective 2-Cyano-Pyrimidine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.51 Å Release Date: 2010-03-02 Classification: HYDROLASE Ligands: KX1, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-03-02
Ligands: KX1, SO4