Search Count: 17
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.13 Å Release Date: 2025-12-24 Classification: HYDROLASE Ligands: A1IW3, EDO |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.73 Å Release Date: 2025-12-24 Classification: HYDROLASE Ligands: A1IWL |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2025-12-24 Classification: HYDROLASE Ligands: A1IWN |
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Crystal Structure Of Human Pyruvate Dehydrogenase Kinase Isoform 1 In Complex With Atp Competitive Inhibitor 29
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.14 Å Release Date: 2025-06-25 Classification: TRANSFERASE Ligands: SO4, TF3, EDO, GOL, A1EQH |
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Crystal Structure Of Human Pyruvate Dehydrogenase Kinase Isoform 2 In Complex With Atp Competitive Inhibitor 24
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.92 Å Release Date: 2025-06-25 Classification: TRANSFERASE Ligands: EDO, TF3, GOL, A1EQJ |
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Crystal Structure Of Human Pyruvate Dehydrogenase Kinase Isoform 2 In Complex With Atp Competitive Inhibitor 22
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.08 Å Release Date: 2025-06-11 Classification: TRANSFERASE Ligands: TF3, A1EQI, DMS |
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Crystal Structure Of Human Pyruvate Dehydrogenase Kinase Isoform 1 In Complex With Atp Competitive Inhibitor 8
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.76 Å Release Date: 2025-04-02 Classification: TRANSFERASE Ligands: K, A1EMR, GOL |
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Crystal Structure Of Human Pyruvate Dehydrogenase Kinase Isoform 1 In Complex With Atp Competitive Inhibitor 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.01 Å Release Date: 2025-04-02 Classification: TRANSFERASE Ligands: K, SZ6, GOL |
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6-Phenyl-1H-Imidazo[4,5-C]Pyridine-4-Carbonitrile As Cathepsin S Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2011-04-06 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: EF3, DMS, SO4 |
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Cathepsin K Covalently Bound To A Cyano-Pyrimidine Inhibitor With Improved Selectivity Over Herg
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2011-03-30 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: O47 |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.49 Å Release Date: 2010-12-22 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: O64, DMS |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.02 Å Release Date: 2010-12-22 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: O96, SO4 |
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Cathepsin K Covalently Bound To A 2-Cyano Pyrimidine Inhibitor With A Benzyl P3 Group.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2010-10-06 Classification: HYDROLASE Ligands: SO4, O75 |
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4-(3-Trifluoromethylphenyl)-Pyrimidine-2-Carbonitrile As Cathepsin S Inhibitors: N3, Not N1 Is Critically Important
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2010-07-14 Classification: HYDROLASE Ligands: PEG, DMS, 935, 93N, SO4, GOL |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2010-03-02 Classification: HYDROLASE Ligands: ORG, TFA |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.49 Å Release Date: 2010-03-02 Classification: HYDROLASE Ligands: SO4, KWZ |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.51 Å Release Date: 2010-03-02 Classification: HYDROLASE Ligands: KX1, SO4 |

















