Search Count: 35
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Crystal Structure Of The Mycobacterium Tuberculosis Regulator Virs (N-Terminal Fragment 4-208) In Complex With The Drug Candidate Alpibectir
Organism: Mycobacterium tuberculosis h37rv
Method: X-RAY DIFFRACTION Resolution:1.49 Å Release Date: 2025-10-29 Classification: TRANSCRIPTION Ligands: YPQ |
Organism: Mycobacterium tuberculosis h37rv
Method: X-RAY DIFFRACTION
Release Date: 2025-10-29
Ligands: YPQ
 |
Crystal Structure Of Trim25 Pryspry Covalently Bound To 2-Chloro-1-[4-(3-Methyl-4-Phenyl-Phenyl)Carbonyl-1,4-Diazepan-1-Yl]Ethanone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2025-05-21 Classification: LIGASE Ligands: A1IZK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-21
Ligands: A1IZK
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Human Cdk8/Cyclin-C Complex With Inhibitor 2-9
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.57 Å Release Date: 2025-01-22 Classification: TRANSCRIPTION Ligands: EDO, GOL, A1IS8, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-22
Ligands: EDO, GOL, A1IS8, DMS
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Human Cdk8/Cyclin-C Complex With Inhibitor 3-7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.16 Å Release Date: 2025-01-22 Classification: TRANSCRIPTION Ligands: CL, EDO, GOL, A1ITF, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-22
Ligands: CL, EDO, GOL, A1ITF, DMS
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Human Dnmt1(729-1600) Bound To Zebularine-Containing 12Mer Dsdna
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2021-07-07 Classification: TRANSFERASE Ligands: SAH, ZN, EDO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: SAH, ZN, EDO, GOL
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Human Dnmt1(729-1600) Bound To Zebularine-Containing 12Mer Dsdna And Inhibitor Gsk3830052
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.79 Å Release Date: 2021-07-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR/DNA Ligands: ZN, EDO, X52 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: ZN, EDO, X52
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Human Dnmt1(729-1600) Bound To Zebularine-Containing 12Mer Dsdna And Inhibitor Gsk3685032A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2021-07-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR/DNA Ligands: ZN, EDO, UXM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: ZN, EDO, UXM
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Brd9 With 4-Chloro-2-Methyl-Methylamino-Pyridazinone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2021-04-14 Classification: TRANSCRIPTION Ligands: 82I |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-14
Ligands: 82I
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Brd9 With Biphenyl-Methylamino-Dimethylpyridazinone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.68 Å Release Date: 2021-03-24 Classification: TRANSCRIPTION Ligands: P8W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-24
Ligands: P8W
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Brd9 With Methylpiperazinyl-Benzyl-Amino-Dimethylpyridazinone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.68 Å Release Date: 2021-03-24 Classification: TRANSCRIPTION Ligands: P8Z |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-24
Ligands: P8Z
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N-Terminal Domain Of Brd4 With Biphenyl-Methyamino-Dimethylpyridazinone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.39 Å Release Date: 2021-03-24 Classification: TRANSCRIPTION Ligands: P8W, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-24
Ligands: P8W, EDO
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N-Terminal Bromodomain Of Human Brd4 With Gsk789
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.62 Å Release Date: 2020-07-29 Classification: TRANSCRIPTION Ligands: QAN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-29
Ligands: QAN
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N-Terminal Bromodomain Of Human Brd4 (3R,4R)-N-Cyclohexyl-4-((3-Methyl-2-Oxo-1,2-Dihydro-1,7-Naphthyridin-8-Yl)Amino)Piperidine-3-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.26 Å Release Date: 2020-07-29 Classification: TRANSCRIPTION Ligands: QAZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-29
Ligands: QAZ
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N-Terminal Bromodomain Of Human Brd4 With Ibet-Bd1 (Gsk778)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.28 Å Release Date: 2020-04-01 Classification: TRANSCRIPTION Ligands: GLU, LWB, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-01
Ligands: GLU, LWB, EDO
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C-Terminal Bromodomain Of Human Brd2 With Ibet-Bd1 (Gsk778)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2020-04-01 Classification: TRANSCRIPTION Ligands: LWB, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-01
Ligands: LWB, EDO
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C-Terminal Bromodomain Of Human Brd2 With Ibet-Bd2 (Gsk046)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2020-04-01 Classification: TRANSCRIPTION Ligands: EDO, LW5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-01
Ligands: EDO, LW5
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N-Terminal Bromodomain Of Human Brd4 With Ibet-Bd2 (Gsk046)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2020-04-01 Classification: TRANSCRIPTION Ligands: EDO, LW5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-01
Ligands: EDO, LW5
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Crystal Structure Of Human Atad2 Bromodomain In Complex With 3-Methyl-8-((8-Methyl-8-Azabicyclooctan-3-Yl)Amino)-1,7-Naphthyridin-2(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2018-09-26 Classification: TRANSCRIPTION Ligands: SO4, EDO, FZB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-09-26
Ligands: SO4, EDO, FZB
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Crystal Structure Of Human Atad2 Bromodomain In Complex With 8-(((1R,2R,3R,5S)-2-(2-(1,1-Dioxidotetrahydro-2H-Thiopyran-4-Yl)Ethyl)-8-Azabicyclo[3.2.1]Octan-3-Yl)Amino)-3-Methyl-5-(5-Methylpyridin-3-Yl)Quinolin-2(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.61 Å Release Date: 2018-09-26 Classification: TRANSCRIPTION Ligands: EDO, FZH, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-09-26
Ligands: EDO, FZH, SO4
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N-Terminal Bromodomain Of Human Brd4 With : 8-(((1R,2R,3R,5S)-2-(2-(4,4-Difluorocyclohexyl)Ethyl)-8-Azabicyclo[3.2.1]Octan-3-Yl)Amino)-3-Methyl-5-(5-Methylpyridin-3-Yl)-1,7-Naphthyridin-2(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2018-09-26 Classification: TRANSCRIPTION Ligands: EDO, FZE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-09-26
Ligands: EDO, FZE