Search Count: 34
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Crystal Structure Of The Human Cdkl2 Kinase Domain With Compound 9
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2025-02-26 Classification: TRANSFERASE Ligands: A1H5G, EDO, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-26
Ligands: A1H5G, EDO, CL
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Crystal Structure Of The Human Cdkl5 Kinase Domain With Compound Yl-354
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2023-06-14 Classification: TRANSFERASE Ligands: US0, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-06-14
Ligands: US0, SO4
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Crystal Structure Of Human Brachyury In Complex With A Single T Box Binding Element Dna
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2023-03-22 Classification: TRANSCRIPTION |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-03-22
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Crystal Structure Of Human Casein Kinase Ii Subunit Alpha (Ck2A1) In Complex With Compound 2 (Aa-Cs-9-003)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2022-11-23 Classification: TRANSFERASE Ligands: SO4, QIA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-23
Ligands: SO4, QIA
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Crystal Structure Of Human Brachyury G177D Variant In Complex With (S)-N-(3-Aminopropyl)-3-((1-(2-Fluorophenyl)-2-Oxopyrrolidin-3-Yl)Amino)-N-Methylbenzamide (Cf-2-125)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2022-10-05 Classification: TRANSCRIPTION Ligands: PO4, L9E |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-10-05
Ligands: PO4, L9E
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Crystal Structure Of Human Brachyury G177D Variant In Complex With Molpolrt-020-049-143
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2022-07-13 Classification: TRANSCRIPTION Ligands: A1IYK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-07-13
Ligands: A1IYK
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Crystal Structure Of Human Brachyury G177D Variant In Complex With Csc027898502
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2022-06-22 Classification: TRANSCRIPTION Ligands: PO4, IU4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-06-22
Ligands: PO4, IU4
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Crystal Structure Of Human Brachyury G177D Variant In Complex With Cf-5-86
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.49 Å Release Date: 2022-06-22 Classification: TRANSCRIPTION Ligands: A1I1T, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-06-22
Ligands: A1I1T, PO4
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Crystal Structure Of Human Brachyury G177D Variant In Complex With Molpolrt-039-246-810
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2022-06-22 Classification: TRANSCRIPTION Ligands: IXB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-06-22
Ligands: IXB
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The Mark3 Kinase Domain Bound To Aa-Cs-1-008
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2021-07-14 Classification: TRANSFERASE Ligands: V5E, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-14
Ligands: V5E, EDO
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Crystal Structure Of Stk17B With Bound Dovitinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.08 Å Release Date: 2020-12-02 Classification: TRANSFERASE Ligands: EDO, 38O |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-02
Ligands: EDO, 38O
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Ck2 Alpha Bound To Chemical Probe Sgc-Ck2-1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.17 Å Release Date: 2020-07-29 Classification: TRANSFERASE Ligands: SO4, QBE, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-29
Ligands: SO4, QBE, PEG
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Ck2 Alpha Bound To Chemical Probe Sgc-Ck2-1 Derivative
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2020-07-29 Classification: TRANSFERASE Ligands: SO4, QB8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-29
Ligands: SO4, QB8
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Crystal Structure Of Stk17B (Drak2) In Complex With Ap-229
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2020-07-29 Classification: TRANSFERASE Ligands: QM2, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-29
Ligands: QM2, EDO
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Crystal Structure Of Stk17B (Drak2) In Complex With Pkis43
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2020-03-11 Classification: TRANSFERASE Ligands: OD2, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-03-11
Ligands: OD2, EDO
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Crystal Structure Of Stk17B (Drak2) In Complex With Unc-Ap-194 Probe
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2020-03-11 Classification: TRANSFERASE Ligands: OBW, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-03-11
Ligands: OBW, EDO
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X-Ray Structure Of Nsd3-Pwwp1 In Complex With Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2019-06-26 Classification: ONCOPROTEIN Ligands: EH2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-26
Ligands: EH2
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X-Ray Structure Of Nsd3-Pwwp1 In Complex With Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.43 Å Release Date: 2019-06-26 Classification: ONCOPROTEIN Ligands: EHQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-26
Ligands: EHQ
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X-Ray Structure Of Nsd3-Pwwp1 In Complex With Compound 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2019-06-26 Classification: ONCOPROTEIN Ligands: EHE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-26
Ligands: EHE
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X-Ray Structure Of Nsd3-Pwwp1 In Complex With Compound 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2019-06-26 Classification: ONCOPROTEIN Ligands: EHK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-26
Ligands: EHK
