Search Count: 9
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Discovery Of (4-Pyrazolyl)-2-Aminopyrimidines As Potent And Selective Inhibitors Of Cyclin-Dependent Kinase 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2024-02-14 Classification: TRANSFERASE/INHIBITOR Ligands: XKU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-02-14
Ligands: XKU
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Structure Of Pseudomonas Nrps Protein, Ambb-Tc Bound To Ppant-L-Ala
Organism: Pseudomonas aeruginosa pao1
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2022-07-13 Classification: BIOSYNTHETIC PROTEIN Ligands: 868 |
Organism: Pseudomonas aeruginosa pao1
Method: X-RAY DIFFRACTION
Release Date: 2022-07-13
Ligands: 868
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Structure Of Pseudomonas Nrps Protein, Ambb-Tc In Apo Form
Organism: Pseudomonas aeruginosa pao1
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2022-07-06 Classification: BIOSYNTHETIC PROTEIN Ligands: 7Z8 |
Organism: Pseudomonas aeruginosa pao1
Method: X-RAY DIFFRACTION
Release Date: 2022-07-06
Ligands: 7Z8
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Structure Of Pseudomonas Nrps Protein, Ambb-Tc Bound To Ppant
Organism: Pseudomonas aeruginosa pao1
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2022-06-15 Classification: BIOSYNTHETIC PROTEIN Ligands: PNS |
Organism: Pseudomonas aeruginosa pao1
Method: X-RAY DIFFRACTION
Release Date: 2022-06-15
Ligands: PNS
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Crystal Structure Of The Human Brd2 Bd1 Bromodomain In Complex With 9-(Cyclopropylmethyl)-7-[(2R,6S)-2,6-Dimethylmorpholine-4-Carbonyl]-3-(3,5-Dimethyl-1,2-Oxazol-4-Yl)-9H-Carbazole-1-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2021-09-29 Classification: CELL CYCLE Ligands: YW1, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-29
Ligands: YW1, EDO
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Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With 9-Benzyl-2-(3,5-Dimethyl-1,2-Oxazol-4-Yl)-7-(2-Hydroxypropan-2-Yl)-9H-Carbazole-4-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2021-09-29 Classification: CELL CYCLE Ligands: YW4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-29
Ligands: YW4, EDO
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Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With 2-(3,5-Dimethyl-1,2-Oxazol-4-Yl)-7-(2-Hydroxypropan-2-Yl)-9-[(S)-(Oxan-4-Yl)(Phenyl)Methyl]-9H-Carbazole-4-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2021-09-29 Classification: CELL CYCLE Ligands: YW7, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-29
Ligands: YW7, EDO
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Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With Bms-986158, 2-{3-(1,4-Dimethyl-1H-1,2,3-Triazol-5-Yl)-5-[(S)-(Oxan-4-Yl)(Phenyl)Methyl]-5H-Pyrido[3,2-B]Indol-7-Yl}Propan-2-Ol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2021-09-29 Classification: CELL CYCLE Ligands: YWA, IOD, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-29
Ligands: YWA, IOD, EDO
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Tyrosine-Protein Kinase Lck Bound To Compound 11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.81 Å Release Date: 2019-10-09 Classification: SIGNALING PROTEIN/INHIBITOR Ligands: ODJ, CXS, SO4, NI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-10-09
Ligands: ODJ, CXS, SO4, NI
