Search Count: 28
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Identification Of Gdc-1971 (Rly-1971), A Shp2 Inhibitor Designed For The Treatment Of Solid Tumors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2023-10-11 Classification: HYDROLASE Ligands: SO4, YR2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-10-11
Ligands: SO4, YR2
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Identification Of Gdc-1971 (Rly-1971), A Shp2 Inhibitor Designed For The Treatment Of Solid Tumors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.84 Å Release Date: 2023-10-11 Classification: HYDROLASE Ligands: SO4, YT2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-10-11
Ligands: SO4, YT2
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Identification Of Gdc-1971 (Rly-1971), A Shp2 Inhibitor Designed For The Treatment Of Solid Tumors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2023-10-11 Classification: HYDROLASE Ligands: ZH5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-10-11
Ligands: ZH5
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Identification Of Gdc-1971 (Rly-1971), A Shp2 Inhibitor Designed For The Treatment Of Solid Tumors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.27 Å Release Date: 2023-10-11 Classification: HYDROLASE/INHIBITOR Ligands: ZJX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-10-11
Ligands: ZJX
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Structure Of Full Length Human Ampk (A2B1G1) In Complex With A Small Molecule Activator Msg011
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.95 Å Release Date: 2022-06-29 Classification: SIGNALING PROTEIN Ligands: 4O7, ZQV, AMP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-06-29
Ligands: 4O7, ZQV, AMP
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Cdk2 In Complex With Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.67 Å Release Date: 2021-11-03 Classification: TRANSFERASE/INHIBITOR Ligands: 3I3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-11-03
Ligands: 3I3
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Type 1 Prmt In Complex With The Inhibitor Gsk3368715
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.48 Å Release Date: 2019-07-10 Classification: ANTITUMOR PROTEIN Ligands: SAH, KZS, GOL, DTT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-10
Ligands: SAH, KZS, GOL, DTT
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Crystal Structure Of Smyd2 With Sam And Epz033294
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.69 Å Release Date: 2018-04-25 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: SAM, ZN, 8WG, PEG, EDO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-04-25
Ligands: SAM, ZN, 8WG, PEG, EDO, GOL
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Crystal Structure Of Smyd3 With Sam And Epz028862
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.42 Å Release Date: 2018-03-07 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: ZN, SAM, 8WD, PEG, DMS, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-07
Ligands: ZN, SAM, 8WD, PEG, DMS, EDO
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Crystal Structure Of Carm1 With Epz022302 And Sah
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.92 Å Release Date: 2018-02-07 Classification: TRANSFERASE Ligands: SAH, BW4, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-02-07
Ligands: SAH, BW4, GOL, SO4
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Crystal Structure Of Carm1 With Compound 2 And Sah
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2018-02-07 Classification: TRANSFERASE Ligands: SAH, BW7, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-02-07
Ligands: SAH, BW7, GOL
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Crystal Structure Of Prmt5:Mep50 With Compound 8 And Sinefungin
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.27 Å Release Date: 2016-02-24 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SFG, 5QJ, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-24
Ligands: SFG, 5QJ, GOL
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Crystal Structure Of Prmt5:Mep50 With Compound 9 And Sinefungin
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.52 Å Release Date: 2016-02-24 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SFG, 5QH, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-24
Ligands: SFG, 5QH, GOL
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Crystal Structure Of Prmt5:Mep50 With Compound 10 And Sam
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.39 Å Release Date: 2016-02-24 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SAM, 5QK, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-24
Ligands: SAM, 5QK, GOL
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Crystal Structure Of Prmt5:Mep50 With Compound 15 And Sinefungin
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.37 Å Release Date: 2016-02-24 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SFG, 5QL, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-24
Ligands: SFG, 5QL, GOL
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Crystal Structure Of Smyd3 With Sam And Oxindole Compound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2015-09-09 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: ZN, SAM, 4ZW, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-09
Ligands: ZN, SAM, 4ZW, EDO
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Crystal Structure Of Smyd3 With Sam And Epz030456
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2015-09-09 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: ZN, SAM, 4ZX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-09
Ligands: ZN, SAM, 4ZX
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Crystal Structure Of Prmt5:Mep50 With Epz015666 And Sinefungin
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2015-04-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SFG, 3XV, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: SFG, 3XV, GOL
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Crystal Structure Of Prmt5:Mep50 With Epz015666 And Sam
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.85 Å Release Date: 2015-04-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SAM, 3XV, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: SAM, 3XV, GOL
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Crystal Structure Of Prmt5:Mep50 With Epz015666 And Sah
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.05 Å Release Date: 2015-04-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SAH, 3XV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: SAH, 3XV
