Search Count: 15
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C-Abl Kinase Domain With The Activator(Cmpd6), 2-Cyano-N-(4-(3,4-Dichlorophenyl)Thiazol-2-Yl)Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2019-03-13 Classification: TRANSFERASE Ligands: SO4, STI, KWD, 2PE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-03-13
Ligands: SO4, STI, KWD, 2PE
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C-Abl Kinase Domain With The Activator(Cmpd29), N-(1-(3,4-Dichlorophenyl)-4,5-Dihydro-1H-Pyrazol-3-Yl)Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.33 Å Release Date: 2019-03-13 Classification: TRANSFERASE Ligands: STI, KWV, SO4, GOL, 2PE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-03-13
Ligands: STI, KWV, SO4, GOL, 2PE
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C-Abl Kinase Domain With The Activator(Cmpd51), N-(1-(3,4-Dichlorophenyl)-4-(2-Hydroxyethyl)-4,5-Dihydro-1H-Pyrazol-3-Yl)Isonicotinamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.86 Å Release Date: 2019-03-13 Classification: TRANSFERASE Ligands: SO4, STI, KWP, GOL, 2PE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-03-13
Ligands: SO4, STI, KWP, GOL, 2PE
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Pim1 Complexed With N-(6-(4-Hydroxyphenyl)-1H-Indazol-3-Yl)Cyclopropanecarboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2017-12-27 Classification: Transferase/Transferase Inhibitor Ligands: C2J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-27
Ligands: C2J
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Gsk3Beta Complex With N-(6-(3,4-Dihydroxyphenyl)-1H-Pyrazolo[3,4-B]Pyridin-3-Yl)Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.20 Å Release Date: 2017-11-01 Classification: TRANSFERASE Ligands: SO4, B4K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-11-01
Ligands: SO4, B4K
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Crystal Structure Of Mouse Pi3 Kinase Delta In Complex With Gsk2269557
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.42 Å Release Date: 2015-09-16 Classification: TRANSFERASE Ligands: VVX |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2015-09-16
Ligands: VVX
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Crystal Structure Of Mouse Pi3 Kinase Delta In Complex With Gsk2292767
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.44 Å Release Date: 2015-09-16 Classification: TRANSFERASE Ligands: OKO |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2015-09-16
Ligands: OKO
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X-Ray Crystal Structure At 2.20A Resolution Of Human Mitochondrial Branched Chain Aminotransferase (Bcatm) Complexed With A Pyrazolopyrimidinone Fragment And An Internal Aldimine Linked Plp.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2015-07-01 Classification: TRANSFERASE Ligands: PLP, 4VT, CL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-07-01
Ligands: PLP, 4VT, CL, EDO
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X-Ray Crystal Structure At 2.20A Resolution Of Human Mitochondrial Branched Chain Aminotransferase (Bcatm) Complexed With A Pyrazolopyrimidinone Fragment And An Internal Aldimine Linked Plp.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2015-07-01 Classification: TRANSFERASE Ligands: PLP, 4VS, CL, EDO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-07-01
Ligands: PLP, 4VS, CL, EDO, GOL
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X-Ray Crystal Structure At 2.17A Resolution Of Human Mitochondrial Branched Chain Aminotransferase (Bcatm) Complexed With A Triazolopyrimidinone Compound And An Internal Aldimine Linked Plp Cofactor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.17 Å Release Date: 2015-07-01 Classification: TRANSFERASE Ligands: PLP, 4VR, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-07-01
Ligands: PLP, 4VR, EDO
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X-Ray Crystal Structure At 1.86A Resolution Of Human Mitochondrial Branched Chain Aminotransferase (Bcatm) Complexed With A Pyrazolopyrimidinone Compound And An Internal Aldimine Linked Plp Cofactor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.86 Å Release Date: 2015-07-01 Classification: TRANSFERASE Ligands: PLP, 775, CL, EDO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-07-01
Ligands: PLP, 775, CL, EDO, GOL
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X-Ray Crystal Structure At 1.82A Resolution Of Human Mitochondrial Branched Chain Aminotransferase (Bcatm) Complexed With A Pyrrolidine Amide Compound And An Internal Aldimine Linked Plp Cofactor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2015-07-01 Classification: TRANSFERASE Ligands: PLP, 4W6, EDO, CL, GOL, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-07-01
Ligands: PLP, 4W6, EDO, CL, GOL, DMS
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X-Ray Crystal Structure At 1.70A Resolution Of Human Mitochondrial Branched Chain Aminotransferase (Bcatm) Complexed With A 4-Chloro-2-Fluoro Substituted Pyrazolopyrimidinone Compound And An Internal Aldimine Linked Plp Cofactor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2015-07-01 Classification: TRANSFERASE Ligands: PLP, 4W4, EDO, CL, GOL, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-07-01
Ligands: PLP, 4W4, EDO, CL, GOL, DMS
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Discovery And Characterization Of A Cell-Permeable, Small-Molecule C-Abl Kinase Activator That Binds To The Myristoyl Binding Site
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2011-03-09 Classification: TRANSFERASE Ligands: SO4, STI, 3YY, 2PE, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-09
Ligands: SO4, STI, 3YY, 2PE, GOL
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Crystal Structure Of Vegfr2 With A Benzimidazole-Urea Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2007-09-18 Classification: TRANSFERASE Ligands: SO4, GIG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-09-18
Ligands: SO4, GIG
