Search Count: 21
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Crystal Structure Of Fms Kinase Domain With A Small Molecular Inhibitor, Plx5622
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2019-09-18 Classification: TRANSFERASE Ligands: 622 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-09-18
Ligands: 622
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N-Terminal Bromodomain Of Brd4 In Complex With Plx5981
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2018-08-01 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: EDO, 6JC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-01
Ligands: EDO, 6JC
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N-Terminal Bromodomain Of Brd4 In Complex With Otx-015
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.27 Å Release Date: 2018-08-01 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: 6JE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-01
Ligands: 6JE
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N-Terminal Bromodomain Of Brd4 In Complex With Otx-015
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.19 Å Release Date: 2018-08-01 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: EDO, 6JF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-01
Ligands: EDO, 6JF
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B-Raf Kinase V600E Oncogenic Mutant In Complex With Plx7904
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.47 Å Release Date: 2015-10-28 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 904 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-28
Ligands: 904
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B-Raf Kinase V600E Oncogenic Mutant In Complex With Dabrafenib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2015-10-28 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: P06 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-28
Ligands: P06
 |
B-Raf Kinase V600E Oncogenic Mutant In Complex With Plx7922
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2015-10-28 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: P02 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-28
Ligands: P02
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B-Raf Kinase Domain In Complex With Plx5568
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2015-10-28 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1OO, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-28
Ligands: 1OO, SO4
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Allosteric Modulation Of Caspase-3 Through Mutagenesis
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2012-06-06 Classification: HYDROLASE/HYDROLASE INHIBITOR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-06-06
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Allosteric Modulation Of Caspase-3 Through Mutagenesis
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.58 Å Release Date: 2012-06-06 Classification: HYDROLASE/HYDROLASE INHIBITOR |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2012-06-06
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Allosteric Modulation Of Caspase-3 Through Mutagenesis
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.66 Å Release Date: 2012-06-06 Classification: HYDROLASE/HYDROLASE INHIBITOR |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2012-06-06
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Allosteric Modulation Of Caspase-3 Through Mutagenesis
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.78 Å Release Date: 2012-06-06 Classification: HYDROLASE/HYDROLASE INHIBITOR |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2012-06-06
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Allosteric Modulation Of Caspase-3 Through Mutagenesis
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.67 Å Release Date: 2012-06-06 Classification: HYDROLASE/HYDROLASE INHIBITOR |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2012-06-06
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Allosteric Modulation Of Caspase-3 Through Mutagenesis
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2012-06-06 Classification: HYDROLASE/HYDROLASE INHIBITOR |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2012-06-06
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Allosteric Modulation Of Caspase-3 Through Mutagenesis
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2012-06-06 Classification: HYDROLASE/HYDROLASE INHIBITOR |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2012-06-06
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Caspase-3 E246A, K242A Double Mutant
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2011-02-23 Classification: Hydrolase/Hydrolase Inhibitor |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-02-23
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Caspase-3 K242A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.62 Å Release Date: 2011-02-23 Classification: HYDROLASE/HYDROLASE INHIBITOR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-02-23
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Caspase-3 E246A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2011-02-16 Classification: Hydrolase/Hydrolase Inhibitor Ligands: CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-02-16
Ligands: CL
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Crystal Structure Of Pseudo-Activated Procaspase-3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2010-03-02 Classification: HYDROLASE/HYDROLASE INHIBITOR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-03-02
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Crystal Structure Of Human Factor Xa Complexed With 3-Chloro-4-(2-Methylamino-Imidazol-1-Ylmethyl)-Thiophene-2-Carboxylic Acid [4-Chloro-2-(5-Chloro-Pyridin-2-Ylcarbamoyl)-6-Methoxy-Phenyl]-Amide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.92 Å Release Date: 2008-01-22 Classification: BLOOD CLOTTING Ligands: CA, CL, 993 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-01-22
Ligands: CA, CL, 993