Search Count: 67
![]() |
Crystal Structure Of Casdatifan Bound To Hif2A-B*:Arnt-B* Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.56 Å Release Date: 2026-02-18 Classification: TRANSCRIPTION Ligands: A1I0H, FMT, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-02-18
Ligands: A1I0H, FMT, MG
![]() |
Pvrbp2B N-Terminal Domain Stabilised Mutant Wht2483
Organism: Plasmodium vivax
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2025-02-26 Classification: CELL ADHESION Ligands: MPD, GOL, EPE, PEG |
Organism: Plasmodium vivax
Method: X-RAY DIFFRACTION
Release Date: 2025-02-26
Ligands: MPD, GOL, EPE, PEG
![]() |
Pvrbp2B N-Terminal Domain Stabilised Mutant Wht2484
Organism: Plasmodium vivax
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2025-02-26 Classification: CELL ADHESION Ligands: GOL, PEG |
Organism: Plasmodium vivax
Method: X-RAY DIFFRACTION
Release Date: 2025-02-26
Ligands: GOL, PEG
![]() |
Crystal Structure Of Human Pi3K-Gamma In Complex With Compound 17
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.96 Å Release Date: 2021-11-03 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: V84 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-11-03
Ligands: V84
![]() |
Human Ecto-5'-Nucleotidase (Cd73) In Complex With The Ampcp Derivative A894 (Compound 2N In Publication) In The Closed Form (Crystal Form Iv)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.66 Å Release Date: 2021-01-20 Classification: HYDROLASE Ligands: ZN, OO2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-20
Ligands: ZN, OO2
![]() |
Human Ecto-5'-Nucleotidase (Cd73) In Complex With The Ampcp Derivative A1202 (Compound 4A In Publication) In The Closed Form (Crystal Form Iv)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.44 Å Release Date: 2021-01-20 Classification: HYDROLASE Ligands: ZN, OO5, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-20
Ligands: ZN, OO5, CA
![]() |
Crystal Structure Of Human Pi3K-Gamma In Complex With Inhibitor Ipi-549
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.99 Å Release Date: 2020-09-16 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: V7Y, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-09-16
Ligands: V7Y, SO4
![]() |
Crystal Structure Of Human Pi3K-Gamma In Complex With Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.88 Å Release Date: 2020-09-16 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: V81, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-09-16
Ligands: V81, SO4
![]() |
Human Ecto-5'-Nucleotidase (Cd73) In Complex With Aopcp Derivative Ab680 (Compound 55 In Publication) In The Closed Form (Crystal Form Iii)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2020-09-16 Classification: HYDROLASE Ligands: ZN, CA, QDH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-09-16
Ligands: ZN, CA, QDH
![]() |
Human Ecto-5'-Nucleotidase (Cd73) In Complex With Aopcp Derivative A830 (Compound 16 In Publication) In The Closed Form (Crystal Form Iii)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.17 Å Release Date: 2020-07-22 Classification: HYDROLASE Ligands: ZN, CA, QCQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-22
Ligands: ZN, CA, QCQ
![]() |
Human Ecto-5'-Nucleotidase (Cd73) In Complex With A2396 (Compound 74 In Publication) In The Closed Form In Crystal Form Iv
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2020-04-22 Classification: HYDROLASE Ligands: ZN, CA, PO4, O1H |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-22
Ligands: ZN, CA, PO4, O1H
![]() |
Human Ecto-5'-Nucleotidase (Cd73) In Complex With A2410 (Compound 53 In Publication) In The Closed Form In Crystal Form Iv
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.09 Å Release Date: 2020-04-22 Classification: HYDROLASE Ligands: ZN, CA, PO4, O1Q |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-22
Ligands: ZN, CA, PO4, O1Q
![]() |
Human Ecto-5'-Nucleotidase (Cd73) In Complex With A1618 (Compound 1B In Publication) In The Closed State In Crystal Form Iii
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2020-04-22 Classification: HYDROLASE Ligands: ZN, CA, O1T |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-22
Ligands: ZN, CA, O1T
![]() |
Crystal Structure Of Irak-4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2016-01-13 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: T20 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-01-13
Ligands: T20
![]() |
Crystal Structure Of Human Lcat (L4F, N5D) In Complex With Fab Of An Agonistic Antibody
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2015-12-16 Classification: HYDROLASE/IMMUNE SYSTEM Ligands: NAG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-12-16
Ligands: NAG
![]() |
Crystal Structure Of Kinase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2015-09-16 Classification: TRANSFERASE Ligands: UNL, EDO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-16
Ligands: UNL, EDO, GOL
![]() |
Crystal Structure Of Kinase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2015-09-16 Classification: TRANSFERASE Ligands: AGS, MG, GOL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-16
Ligands: AGS, MG, GOL, EDO
![]() |
Crystal Structure Of Lcat (C31Y) In Complex With Fab1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2015-07-29 Classification: Hydrolase/Immune system Ligands: ZN, NAG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-07-29
Ligands: ZN, NAG
![]() |
Low Resolution Structure Of Lcat In Complex With Fab1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.60 Å Release Date: 2015-07-29 Classification: Hydrolase/Immune system Ligands: NAG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-07-29
Ligands: NAG
![]() |
Crystal Structure Of A Cdk6/Vcyclin Complex With Inhibitor Bound
Organism: Saimiriine herpesvirus 2, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2014-08-06 Classification: TRANSFERASE/CELL CYCLE/INHIBITOR Ligands: 24V |
Organism: Saimiriine herpesvirus 2, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-08-06
Ligands: 24V
