Search Count: 8
![]() |
Jak3 Kinase Domain In Complex With 1-[(3S)-1-Isobutylsulfonyl-3-Piperidyl]-3-(5H-Pyrrolo[2,3-B]Pyrazin-2-Yl)Urea
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2015-05-27 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3C9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-05-27
Ligands: 3C9
![]() |
Crystal Structure Of Jak3 Kinase Domain In Complex With A Pyrrolopyrazine-2-Phenyl Ether Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2013-12-11 Classification: TRANSFERASE Ligands: 1NX, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-12-11
Ligands: 1NX, GOL
![]() |
Jak3 Kinase Domain In Complex With 2-Phenoxy-5H-Pyrrolo[2,3-B]Pyrazine-7-Carboxylic Acid ((S)-1-Cyclopropyl-Ethyl)-Amide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2013-10-16 Classification: Transferase/Transferase Inhibitor Ligands: PHU, 1DT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-10-16
Ligands: PHU, 1DT
![]() |
Crystal Structure Of Jak3 Kinase Domain In Complex With An Indazole Substituted Pyrrolopyrazine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.42 Å Release Date: 2013-09-25 Classification: TRANSFERASE Ligands: VFC, PEG, CL, PG4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-09-25
Ligands: VFC, PEG, CL, PG4
![]() |
Jak3 Kinase Domain In Complex With 2-Cyclopropyl-5H-Pyrrolo[2,3-B]Pyrazine-7-Carboxylic Acid ((S)-1,2,2-Trimethyl-Propyl)-Amide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2013-01-16 Classification: Transferase/Transferase Inhibitor Ligands: PHU, 933 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-01-16
Ligands: PHU, 933
![]() |
Jak3 Kinase Domain In Complex With 2-Cyclopropyl-5H-Pyrrolo[2,3-B]Pyrazine-7-Carboxylic Acid ((S)-2-Hydroxy-1,2-Dimethyl-Propyl)-Amide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.75 Å Release Date: 2013-01-16 Classification: Transferase/Transferase Inhibitor Ligands: 19Q |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-01-16
Ligands: 19Q
![]() |
Jak3 Kinase Domain In Complex With 2-Cyclopropyl-5H-Pyrrolo[2,3-B]Pyrazine-7-Carboxylic Acid ((R)-2-Hydroxy-1,2-Dimethyl-Propyl
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2013-01-16 Classification: Transferase/Transferase Inhibitor Ligands: 19R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-01-16
Ligands: 19R
![]() |
Jak3 Kinase Domain In Complex With 2-Cyclopropyl-5H-Pyrrolo[2,3-B]Pyrazine-7-Carboxylic Acid ((R)-1-Methyl-2-Oxo-2-Piperidin-1-Yl-Ethyl)-Amide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2013-01-16 Classification: Transferase/Transferase Inhibitor Ligands: 19S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-01-16
Ligands: 19S
