Search Count: 5
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Discovery Of Imidazo[1,2-A]-Pyridine Inhibitors Of Pan-Pi3 Kinases That Are Efficacious In A Mouse Xenograft Model
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2016-02-03 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GOL, 5XV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-03
Ligands: GOL, 5XV
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Structure Of Pi3K Gamma With Imidazopyridine Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.87 Å Release Date: 2013-07-17 Classification: Transferase/Transferase Inhibitor Ligands: 1UJ, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-07-17
Ligands: 1UJ, SO4
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Structure Of Pi3K Gamma With Imidazopyridine Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.25 Å Release Date: 2013-07-17 Classification: Transferase/Transferase Inhibitor Ligands: 1UK, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-07-17
Ligands: 1UK, SO4
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Crystal Structure Of Pi3K Gamma With 5-(2,4-Dimorpholinopyrimidin-6-Yl)-4-(Trifluoromethyl)Pyridin-2-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.20 Å Release Date: 2012-01-04 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SD5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-01-04
Ligands: SD5
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Crystal Structure Of Pi3K Gamma With 3-(2-Morpholino-6-(Pyridin-3-Ylamino)Pyrimidin-4-Yl)Phenol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.20 Å Release Date: 2011-08-17 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: P2B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-08-17
Ligands: P2B
