Search Count: 29
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Bruton'S Tyrosine Kinase In Complex With 5-(Piperidin-1-Yl)-3-{[4-(Piperidin-4-Yl)Phenyl]Amino}Pyrazine-2-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2024-01-31 Classification: SIGNALING PROTEIN Ligands: YXJ, EDO, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-01-31
Ligands: YXJ, EDO, CL
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Bruton'S Tyrosine Kinase L528W Mutant In Complex With 5-(Piperidin-1-Yl)-3-{[4-(Piperidin-4-Yl)Phenyl]Amino}Pyrazine-2-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2024-01-31 Classification: SIGNALING PROTEIN Ligands: YXJ, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-01-31
Ligands: YXJ, EDO
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P110Delta/P85Alpha With Taselisib (Gdc-0032)
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION Resolution:2.91 Å Release Date: 2017-01-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 799 |
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2017-01-11
Ligands: 799
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Crystal Structure Of Murine Nf-Kappab Inducing Kinase (Nik) Bound To Imidazobenzoxepin Compound 3
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 2017-01-11 Classification: TRANSFERASE Ligands: SO4, 76Z |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2017-01-11
Ligands: SO4, 76Z
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Crystal Structure Of Murine Nf-Kappab Inducing Kinase (Nik) Bound To Benzoxepin Compound 2
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.32 Å Release Date: 2017-01-11 Classification: TRANSFERASE Ligands: 774, SO4 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2017-01-11
Ligands: 774, SO4
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Crystal Structure Of Murine Nf-Kappab Inducing Kinase (Nik) Bound To Aryl Pyrrole Fragment 17
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.63 Å Release Date: 2017-01-11 Classification: TRANSFERASE Ligands: SO4, 76Y |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2017-01-11
Ligands: SO4, 76Y
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Map4K4 In Complex With Inhibitor (Compound 6)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.18 Å Release Date: 2014-09-03 Classification: Transferase/Transferase inhibitor Ligands: 3D8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-09-03
Ligands: 3D8
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Map4K4 In Complex With Inhibitor (Compound 16)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.43 Å Release Date: 2014-09-03 Classification: Transferase/Transferase inhibitor Ligands: MES, NA, 3D9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-09-03
Ligands: MES, NA, 3D9
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Map4K4 In Complex With Inhibitor (Compound 25)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.58 Å Release Date: 2014-09-03 Classification: Transferase/Transferase inhibitor Ligands: MG, 3DC, MES |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-09-03
Ligands: MG, 3DC, MES
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Crystal Structure Of The Braf:Mek1 Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.85 Å Release Date: 2014-06-18 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ACP, MG, 573, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-06-18
Ligands: ACP, MG, 573, CL
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Crystal Structure Of Braf-V600E Bound To Gdc0879
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2014-06-18 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 29L, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-06-18
Ligands: 29L, CL
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Map4K4 In Complex With Inhibitor (Compound 22), 6-(3-Chlorophenyl)Quinazolin-4-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2014-04-23 Classification: transferase/transferase inhibitor Ligands: MES, NA, 2QV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-23
Ligands: MES, NA, 2QV
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Map4K4 In Complex With Inhibitor (Compound 29), 6-(2-Fluoropyridin-4-Yl)Pyrido[3,2-D]Pyrimidin-4-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.27 Å Release Date: 2014-04-23 Classification: transferase/transferase inhibitor Ligands: MG, MES, 2QU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-23
Ligands: MG, MES, 2QU
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Map4K4 In Complex With Inhibitor (Compound 31), N-[3-(4-Aminoquinazolin-6-Yl)-5-Fluorophenyl]-2-(Pyrrolidin-1-Yl)Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.19 Å Release Date: 2014-04-23 Classification: transferase/transferase inhibitor Ligands: MES, MG, 2QT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-23
Ligands: MES, MG, 2QT
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Fragment-Based Design Of 3-Aminopyridine-Derived Amides As Potent Inhibitors Of Human Nicotinamide Phosphoribosyltransferase (Nampt)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.86 Å Release Date: 2014-02-19 Classification: transferase/transferase inhibitor Ligands: PO4, 2HH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-02-19
Ligands: PO4, 2HH
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Fragment-Based Design Of 3-Aminopyridine-Derived Amides As Potent Inhibitors Of Human Nicotinamide Phosphoribosyltransferase (Nampt)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2014-02-19 Classification: transferase/transferase inhibitor Ligands: 2ZM, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-02-19
Ligands: 2ZM, PO4
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Fragment-Based Design Of 3-Aminopyridine-Derived Amides As Potent Inhibitors Of Human Nicotinamide Phosphoribosyltransferase (Nampt)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2014-02-19 Classification: transferase/transferase inhibitor Ligands: 2HJ, PO4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-02-19
Ligands: 2HJ, PO4, EDO
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Fragment-Based Design Of 3-Aminopyridine-Derived Amides As Potent Inhibitors Of Human Nicotinamide Phosphoribosyltransferase (Nampt)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2014-02-19 Classification: transferase/transferase inhibitor Ligands: 2HL, PO4, EDO, DTT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-02-19
Ligands: 2HL, PO4, EDO, DTT
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Tailoring Small Molecules For An Allosteric Site On Procaspase-6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.14 Å Release Date: 2014-01-01 Classification: hydrolase/hydrolase inhibitor Ligands: PO4, 2GQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-01-01
Ligands: PO4, 2GQ
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Tailoring Small Molecules For An Allosteric Site On Procaspase-6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2014-01-01 Classification: hydrolase/hydrolase inhibitor Ligands: 2J5, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-01-01
Ligands: 2J5, PO4