Search Count: 23
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Crystal Structure Of An Allosteric Inhibitor Bound To Human Ripk1 Kinase Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.98 Å Release Date: 2025-12-24 Classification: IMMUNE SYSTEM Ligands: A1IX7, IOD, 1HX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-12-24
Ligands: A1IX7, IOD, 1HX
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Crystal Structure Of An Allosteric Inhibitor Bound To Human Ripk1 Kinase Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.29 Å Release Date: 2025-12-24 Classification: IMMUNE SYSTEM Ligands: A1IX9, IOD, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-12-24
Ligands: A1IX9, IOD, PEG
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Hiv Protease (Pr) Dimer In Closed Form With Pepstatin In Active Site And Fragment Ak-2097 In The Outside/Top Of Flap
Organism: Human immunodeficiency virus 1, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.18 Å Release Date: 2014-09-24 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: K97, GOL |
Organism: Human immunodeficiency virus 1, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2014-09-24
Ligands: K97, GOL
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Hiv Protease (Pr) Dimer In Closed Form With Tl-3 In Active Site And Fragment Ak-2097 In The Outside/Top Of Flap
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2014-09-17 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 3TL, BME, K97 |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2014-09-17
Ligands: 3TL, BME, K97
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5-(4-Fluorophenyl)-3-Hydroxy-6-[4-(1H-1,2,3,4-Tetrazol-5-Yl)Phenyl]-1,2-Dihydropyridin-2-One Bound To Influenza 2009 Ph1N1 Endonuclease
Organism: Influenza a virus (a/lima/wrair1695p/2009(h1n1))
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2013-09-25 Classification: RNA BINDING PROTEIN/INHIBITOR Ligands: MN, SO4, 20F |
Organism: Influenza a virus (a/lima/wrair1695p/2009(h1n1))
Method: X-RAY DIFFRACTION
Release Date: 2013-09-25
Ligands: MN, SO4, 20F
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5-Bromopyridine-2,3-Diol Bound To Influenza 2009 Ph1N1 Endonuclease
Organism: Influenza a virus (a/lima/wrair1695p/2009(h1n1))
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2013-09-25 Classification: RNA BINDING PROTEIN/INHIBITOR Ligands: MN, SO4, EDO, 27Y |
Organism: Influenza a virus (a/lima/wrair1695p/2009(h1n1))
Method: X-RAY DIFFRACTION
Release Date: 2013-09-25
Ligands: MN, SO4, EDO, 27Y
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3-(5-Hydroxy-6-Oxo-1,6-Dihydropyridin-3-Yl)Benzonitrile Bound To Influenza 2009 Ph1N1 Endonuclease
Organism: Influenza a virus (a/lima/wrair1695p/2009(h1n1))
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2013-09-25 Classification: RNA BINDING PROTEIN/INHIBITOR Ligands: MN, SO4, EDO, 28B |
Organism: Influenza a virus (a/lima/wrair1695p/2009(h1n1))
Method: X-RAY DIFFRACTION
Release Date: 2013-09-25
Ligands: MN, SO4, EDO, 28B
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6-(3-Methoxyphenyl)Pyridine-2,3-Diol Bound To Influenza 2009 Ph1N1 Endonuclease
Organism: Influenza a virus (a/lima/wrair1695p/2009(h1n1))
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2013-09-25 Classification: RNA BINDING PROTEIN/INHIBITOR Ligands: MN, SO4, EDO, 28A |
Organism: Influenza a virus (a/lima/wrair1695p/2009(h1n1))
Method: X-RAY DIFFRACTION
Release Date: 2013-09-25
Ligands: MN, SO4, EDO, 28A
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5,6-Bis(4-Fluorophenyl)-3-Hydroxy-2,5-Dihydropyridin-2-One Bound To Influenza 2009 Ph1N1 Endonuclease
Organism: Influenza a virus (a/lima/wrair1695p/2009(h1n1))
Method: X-RAY DIFFRACTION Resolution:1.73 Å Release Date: 2013-09-18 Classification: RNA BINDING PROTEIN/INHIBITOR Ligands: MN, EDO, SO4, 1ZQ, MG |
Organism: Influenza a virus (a/lima/wrair1695p/2009(h1n1))
Method: X-RAY DIFFRACTION
Release Date: 2013-09-18
Ligands: MN, EDO, SO4, 1ZQ, MG
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6-(4-Fluorophenyl)-3-Hydroxy-5-[4-(1H-1,2,3,4-Tetrazol-5-Yl)Phenyl] -1,2-Dihydropyridin-2-One Bound To Influenza 2009 H1N1 Endonuclease
Organism: Influenza a virus (a/lima/wrair1695p/2009(h1n1))
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2013-09-18 Classification: RNA BINDING PROTEIN/INHIBITOR Ligands: MN, SO4, 21A, MG |
Organism: Influenza a virus (a/lima/wrair1695p/2009(h1n1))
Method: X-RAY DIFFRACTION
Release Date: 2013-09-18
Ligands: MN, SO4, 21A, MG
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3-Hydroxy-6-Phenyl-1,2-Dihydropyridin-2-One Bound To Influenza 2009 H1N1 Endonuclease
Organism: Influenza a virus (a/lima/wrair1695p/2009(h1n1))
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2013-09-18 Classification: RNA BINDING PROTEIN/INHIBITOR Ligands: MN, SO4, EDO, X48 |
Organism: Influenza a virus (a/lima/wrair1695p/2009(h1n1))
Method: X-RAY DIFFRACTION
Release Date: 2013-09-18
Ligands: MN, SO4, EDO, X48
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High-Resolution Apo Influenza 2009 H1N1 Endonuclease Structure
Organism: Influenza a virus (a/lima/wrair1695p/2009(h1n1))
Method: X-RAY DIFFRACTION Resolution:1.53 Å Release Date: 2013-09-18 Classification: RNA BINDING PROTEIN Ligands: MN, EDO |
Organism: Influenza a virus (a/lima/wrair1695p/2009(h1n1))
Method: X-RAY DIFFRACTION
Release Date: 2013-09-18
Ligands: MN, EDO
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High-Resolution Influenza 2009 H1N1 Endonuclease Bound To 4-(1H-Imidazol-1-Yl)Phenol
Organism: Influenza a virus (a/lima/wrair1695p/2009(h1n1))
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2013-09-18 Classification: RNA BINDING PROTEIN/INHIBITOR Ligands: MN, MSR, SO4, EDO |
Organism: Influenza a virus (a/lima/wrair1695p/2009(h1n1))
Method: X-RAY DIFFRACTION
Release Date: 2013-09-18
Ligands: MN, MSR, SO4, EDO
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Influenza 2009 H1N1 Endonuclease With 100 Millimolar Calcium
Organism: Influenza a virus (a/lima/wrair1695p/2009(h1n1))
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2013-09-18 Classification: RNA BINDING PROTEIN Ligands: SO4, CA |
Organism: Influenza a virus (a/lima/wrair1695p/2009(h1n1))
Method: X-RAY DIFFRACTION
Release Date: 2013-09-18
Ligands: SO4, CA
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7-(4-Fluorophenyl)-3-Hydroxyquinolin-2(1H)-One Bound To Influenza 2009 H1N1 Endonuclease
Organism: Influenza a virus (a/lima/wrair1695p/2009(h1n1))
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2013-05-29 Classification: Rna binding protein/inhibitor Ligands: MN, SO4, EDO, 1R5 |
Organism: Influenza a virus (a/lima/wrair1695p/2009(h1n1))
Method: X-RAY DIFFRACTION
Release Date: 2013-05-29
Ligands: MN, SO4, EDO, 1R5
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Hiv-1 Reverse Transcriptase With Bound Fragment At Nnrti Adjacent Site
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2013-05-15 Classification: transferase/transferase inhibitor Ligands: 1QP, DMS, T27 |
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION
Release Date: 2013-05-15
Ligands: 1QP, DMS, T27
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Hiv-1 Reverse Transcriptase With Bound Fragment At The Incoming Dntp Binding Site
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2013-02-06 Classification: transferase/transferase inhibitor Ligands: T27, MG, DMS, 14N |
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION
Release Date: 2013-02-06
Ligands: T27, MG, DMS, 14N
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Hiv-1 Reverse Transcriptase With Bound Fragment At The Rnase H Primer Grip Site
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2013-02-06 Classification: transferase/transferase inhibitor Ligands: T27, DMS, 1FF, MG |
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION
Release Date: 2013-02-06
Ligands: T27, DMS, 1FF, MG
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Hiv-1 Reverse Transcriptase With Bound Fragment At The 428 Site
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2013-02-06 Classification: transferase/transferase inhibitor Ligands: T27, 1FE, MG, DMS |
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION
Release Date: 2013-02-06
Ligands: T27, 1FE, MG, DMS
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Detecting Allosteric Sites Of Hiv-1 Reverse Transcriptase By X-Ray Crystallographic Fragment Screening
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2013-02-06 Classification: transferase/transferase inhibitor Ligands: T27, FMQ, DMS, MG |
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION
Release Date: 2013-02-06
Ligands: T27, FMQ, DMS, MG
