Search Count: 24
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Structure Of The Kdm1A/Corest Complex With The Inhibitor 2-[3-{4-Chloro-3-[(4-Chlorophenyl)Ethynyl]Phenyl}-1-(3-Morpholin-4-Ylpropyl)-1,4,6,7-Tetrahydro-5H-Pyrazolo[4,3-C]Pyridin-5-Yl]-2-Oxoethanol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.11 Å Release Date: 2020-06-03 Classification: OXIDOREDUCTASE Ligands: N4K, FAD, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-06-03
Ligands: N4K, FAD, GOL
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Thieno[3,2-B]Pyrrole-5-Carboxamides As Novel Reversible Inhibitors Of Histone Lysine Demethylase Kdm1A/Lsd1: Compound 19
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.20 Å Release Date: 2017-02-22 Classification: OXIDOREDUCTASE Ligands: FAD, 6W0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: FAD, 6W0
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Thieno[3,2-B]Pyrrole-5-Carboxamides As Novel Reversible Inhibitors Of Histone Lysine Demethylase Kdm1A/Lsd1: Compound 15
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2017-02-22 Classification: OXIDOREDUCTASE Ligands: FAD, 6W3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: FAD, 6W3
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Thieno[3,2-B]Pyrrole-5-Carboxamides As Novel Reversible Inhibitors Of Histone Lysine Demethylase Kdm1A/Lsd1: Compound 34
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.20 Å Release Date: 2017-02-22 Classification: OXIDOREDUCTASE Ligands: FAD, 6W1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: FAD, 6W1
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Structure Of The Kdm1A/Corest Complex With The Inhibitor 4-Methyl-N-[4-[[4-(1-Methylpiperidin-4-Yl)Oxyphenoxy]Methyl]Phenyl]Thieno[3,2-B]Pyrrole-5-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.34 Å Release Date: 2017-02-22 Classification: OXIDOREDUCTASE Ligands: FAD, GOL, 6X3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: FAD, GOL, 6X3
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Structure Of The Kdm1A/Corest Complex With The Inhibitor 4-Ethyl-N-[3-(Methoxymethyl)-2-[[4-[[(3R)-Pyrrolidin-3-Yl]Methoxy]Phenoxy]Methyl]Phenyl]Thieno[3,2-B]Pyrrole-5-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.05 Å Release Date: 2017-02-22 Classification: OXIDOREDUCTASE Ligands: FAD, GOL, 6X0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: FAD, GOL, 6X0
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Structure Of The Kdm1A/Corest Complex With The Inhibitor N-[3-(Ethoxymethyl)-2-[[4-[[(3R)-Pyrrolidin-3-Yl]Methoxy]Phenoxy]Methyl]Phenyl]-4-Methylthieno[3,2-B]Pyrrole-5-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.40 Å Release Date: 2017-02-22 Classification: OXIDOREDUCTASE Ligands: FAD, 6X5, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: FAD, 6X5, GOL
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Lsd1(Kdm1A)-Corest In Complex With Z-Pro Derivative Of Mc2580
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.85 Å Release Date: 2015-02-25 Classification: OXIDOREDUCTASE Ligands: FAD, M8A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-02-25
Ligands: FAD, M8A
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Lsd1(Kdm1A)-Corest In Complex With 1-Benzyl-Tranylcypromine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2014-09-10 Classification: TRANSCRIPTION Ligands: D69 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-09-10
Ligands: D69
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Lsd1(Kdm1A)-Corest In Complex With 1-Ethyl-Tranylcypromine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2014-09-10 Classification: TRANSCRIPTION Ligands: D70 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-09-10
Ligands: D70
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Lsd1(Kdm1A)-Corest In Complex With 1-Methyl-Tranylcypromine (1R,2S)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2014-09-10 Classification: TRANSCRIPTION Ligands: D73 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-09-10
Ligands: D73
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Lsd1(Kdm1A)-Corest In Complex With 1-Methyl-Tranylcypromine (1S,2R)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2014-09-10 Classification: TRANSCRIPTION Ligands: D51 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-09-10
Ligands: D51
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Lsd1(Kdm1A)-Corest In Complex With 1-Phenyl-Tranylcypromine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.10 Å Release Date: 2014-09-10 Classification: TRANSCRIPTION Ligands: D52 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-09-10
Ligands: D52
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Pyrrole-3-Carboxamides As Potent And Selective Jak2 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2014-07-23 Classification: TRANSFERASE Ligands: GOL, VVQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-23
Ligands: GOL, VVQ
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Pyrrole-3-Carboxamides As Potent And Selective Jak2 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2014-07-23 Classification: TRANSFERASE Ligands: 953, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-23
Ligands: 953, GOL
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Pyrrole-3-Carboxamides As Potent And Selective Jak2 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.66 Å Release Date: 2014-07-23 Classification: TRANSFERASE Ligands: BJG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-23
Ligands: BJG
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Human Bcl-2 With Phenylacylsulfonamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2012-06-06 Classification: APOPTOSIS Ligands: 398 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-06-06
Ligands: 398
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Aurora-A T288E Complexed With Pha-828300
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2010-09-29 Classification: TRANSFERASE Ligands: 400 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-09-29
Ligands: 400
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Structure Of Cdk2-Cyclin A With Pha-848125
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2009-07-28 Classification: TRANSFERASE Ligands: P48, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-07-28
Ligands: P48, SO4
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Structure Of Cdk2-Cyclin A Complexed With 8-Anilino-1-Methyl-4,5-Dihydro- 1H-Pyrazolo[4,3-H] Quinazoline-3-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2009-07-28 Classification: TRANSFERASE Ligands: P49, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-07-28
Ligands: P49, SO4