Search Count: 26
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Crystal Structure Of Mouse Sting Ctd Complex With Sr-717.
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2020-08-26 Classification: IMMUNE SYSTEM Ligands: V67 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2020-08-26
Ligands: V67
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Crystal Structure Of Human Sting Ctd Complex With Sr-717
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2020-08-26 Classification: IMMUNE SYSTEM Ligands: V67, GOL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-08-26
Ligands: V67, GOL, EDO
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Crystal Structure Of Human Phosphodiesterase 2A With N-(1-Adamantyl)-1-(2-Chlorophenyl)-4-Methyl-[1,2,4]Triazolo[4,3-A]Quinoxaline-8-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.79 Å Release Date: 2018-08-15 Classification: HYDROLASE Ligands: EOJ, ZN, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-15
Ligands: EOJ, ZN, MG
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Crystal Structure Of Human Phosphodiesterase 2A With 1-(2-Chlorophenyl)-N,4-Dimethyl-[1,2,4]Triazolo[4,3-A]Quinoxaline-8-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.43 Å Release Date: 2018-08-15 Classification: HYDROLASE Ligands: EOG, ZN, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-15
Ligands: EOG, ZN, MG
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Crystal Structure Of Human Phosphodiesterase 2A With 1-(2-Chloro-5-Isobutoxy-Phenyl)-N,4-Dimethyl-[1,2,4]Triazolo[4,3-A]Quinoxaline-8-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2018-08-15 Classification: HYDROLASE Ligands: EOS, ZN, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-15
Ligands: EOS, ZN, MG
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Crystal Structure Of Human Phosphodiesterase 2A With N-(1-Adamantyl)-1-(2-Chloro-5-Isobutoxy-Phenyl)-4-Methyl-[1,2,4]Triazolo[4,3-A]Quinoxaline-8-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.68 Å Release Date: 2018-08-15 Classification: HYDROLASE Ligands: EOY, ZN, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-15
Ligands: EOY, ZN, MG
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Crystal Structure Of Human Phosphodiesterase 2A With 1-(2-Chloro-5-Methoxy-Phenyl)-N-Isobutyl-4-Methyl-[1,2,4]Triazolo[4,3-A]Quinoxaline-8-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.71 Å Release Date: 2018-08-15 Classification: HYDROLASE Ligands: EP7, ZN, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-15
Ligands: EP7, ZN, MG
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Crystal Structure Of Human Phosphodiesterase 2A With 1-(5-Tert-Butoxy-2-Chloro-Phenyl)-N-Isobutyl-4-Methyl-[1,2,4]Triazolo[4,3-A]Quinoxaline-8-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2018-08-15 Classification: HYDROLASE Ligands: EPV, ZN, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-15
Ligands: EPV, ZN, MG
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Crystal Structure Of Human Phosphodiesterase 2A In Complex With [1,2,4]Triazolo[1,5-A]Pyrimidin-7-Yl}-N-(Naphthalene-2-Yl)Piperidine-3-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2017-02-22 Classification: Hydrolase/Hydrolase Inhibitor Ligands: 7OM, ZN, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: 7OM, ZN, MG
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Crystal Structure Of Human Phosphodiesterase 2A With 3-{5-Methyl-[1,2,4]Triazolo[1,5-A]Pyrimidin-7-Yl-1-[(Naphthalene-2-Yl)Carbonyl]Piperidine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2017-02-22 Classification: Hydrolase/Hydrolase Inhibitor Ligands: 7OG, ZN, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: 7OG, ZN, MG
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Crystal Structure Of Human Pde2A In Complex With (5S)-1-[(3-Bromo-4-Fluorophenyl)Carbonyl]-3,3-Difluoro-5-{5-Methyl-[1,2,4]Triazolo[1,5-A]Pyrimidin-7-Yl}Piperidine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.36 Å Release Date: 2017-02-22 Classification: Hydrolase/Hydrolase Inhibitor Ligands: 7OJ, ZN, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: 7OJ, ZN, MG
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Crystal Structure Of Human Phosphodiesterase 2A In Complex With 3,3-Difluoro-1-[(4-Fluorophenyl)Carbonyl]-5-{5-Methyl-[1,2,4]Triazolo[1,5-A]Pyrimidin-7-Yl}Piperidine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2017-02-22 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 7OP, ZN, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: 7OP, ZN, MG
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Crystal Structure Of Human Phosphodiesterase 2A In Complex With 1-[(3,4-Difluorophenyl)Carbonyl]-3,3-Difluoro-5-{5-Methyl-[1,2,4]Triazolo[1,5-A]Pyrimidin-7-Yl}Piperidine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2017-02-22 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 7P4, ZN, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: 7P4, ZN, MG
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Crystal Structure Of Human Phosphodiesterase 2A In Complex With 1-[(3-Chloro-4-Fluorophenyl)Carbonyl]-3,3-Difluoro-5-{5-Methyl-[1,2,4]Triazolo[1,5-A]Pyrimidin-7-Yl}Piperidine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2017-02-22 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 7OY, ZN, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: 7OY, ZN, MG
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Crystal Structure Of Human Phosphodiesterase 2A In Complex With 1-[(3-Bromo-4-Fluorophenyl)Carbonyl]-3,3-Difluoro-5-{5-Methyl-[1,2,4]Triazolo[1,5-A]Pyrimidin-7-Yl}Piperidine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2017-02-22 Classification: Hydrolase/Hydrolase Inhibitor Ligands: 7OJ, ZN, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: 7OJ, ZN, MG
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Crystal Structure Of Human Phosphodiesterase 2A In Complex With 3,3-Difluoro-1-[(4-Fluoro-3-Iodophenyl)Carbonyl]-5-{5-Methyl-[1,2,4]Triazolo[1,5-A]Pyrimidin-7-Yl}Piperidine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.41 Å Release Date: 2017-02-22 Classification: Hydrolase/Hydrolase Inhibitor Ligands: 7OV, ZN, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: 7OV, ZN, MG
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Egfr (L858R, T790M, V948R) In Complex With N-{3-[(2-{[4-(4-Methylpiperazin-1-Yl)Phenyl]Amino}-7H-Pyrrolo[2,3-D]Pyrimidin-4-Yl)Oxy]Phenyl}Prop-2-Enamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.52 Å Release Date: 2016-02-03 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 633, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-03
Ligands: 633, SO4, GOL
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Egfr (L858R, T790M, V948R) In Complex With N-[3-({2-[(1-Methyl-1H-Pyrazol-4-Yl)Amino]-7H-Pyrrolo[2,3-D]Pyrimidin-4-Yl}Oxy)Phenyl]Prop-2-Enamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.42 Å Release Date: 2016-02-03 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 634, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-03
Ligands: 634, SO4, GOL
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Egfr (L858R, T790M, V948R) In Complex With 1-[(3R,4R)-3-[({2-[(1-Methyl-1H-Pyrazol-4-Yl)Amino]-7H-Pyrrolo[2,3-D]Pyrimidin-4-Yl}Oxy)Methyl]-4-(Trifluoromethyl)Pyrrolidin-1-Yl]Prop-2-En-1-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2016-02-03 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 63A, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-03
Ligands: 63A, SO4, GOL
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Egfr (L858R, T790M, V948R) In Complex With 1-{(3R,4R)-3-[5-Chloro-2-(1-Methyl-1H-Pyrazol-4-Ylamino)-7H-Pyrrolo[2,3-D]Pyrimidin-4-Yloxymethyl]-4-Methoxy-Pyrrolidin-1-Yl}Propenone (Pf-06459988)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2016-01-27 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 630, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-01-27
Ligands: 630, SO4