Search Count: 29
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Cryoem Structure Of Nlrp3 Nacht Domain In Complex With G2394
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2022-11-02 Classification: HYDROLASE Ligands: MG, ADP, WTN |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2022-11-02
Ligands: MG, ADP, WTN
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Crystal Structure Of Lysine Specific Demethylase 1 (Lsd1) With Cc-90011
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.93 Å Release Date: 2020-10-21 Classification: FLAVOPROTEIN Ligands: V0Y, FAD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-10-21
Ligands: V0Y, FAD
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Crystal Structure Of Brd4 With Qc4956
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.62 Å Release Date: 2018-05-02 Classification: GENE REGULATION/INHIBITOR Ligands: F5V |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-02
Ligands: F5V
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Crystal Structure Of Brd4 With Qc4956
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2018-05-02 Classification: GENE REGULATION/INHIBITOR Ligands: F5Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-02
Ligands: F5Y
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Crystal Structure Of Kdm4A With Compound 14
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.16 Å Release Date: 2018-04-18 Classification: OXIDOREDUCTASE/INHIBITOR Ligands: NI, ZN, QC1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-04-18
Ligands: NI, ZN, QC1
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Crystal Structure Of Kdm4A With Compound 8
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.34 Å Release Date: 2018-04-18 Classification: OXIDOREDUCTASE/INHIBITOR Ligands: NI, ZN, QC2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-04-18
Ligands: NI, ZN, QC2
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Crystal Structure Of Kdm4 With The Small Molecule Inhibitor Qc6352
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.07 Å Release Date: 2017-09-27 Classification: OXIDOREDUCTASE/INHIBITOR Ligands: NI, ZN, 9DJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-09-27
Ligands: NI, ZN, 9DJ
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Crystal Structure Of Human Kdm4 With Small Molecule Inhibitor Qc5714
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.48 Å Release Date: 2017-09-27 Classification: OXIDOREDUCTASE/INHIBITOR Ligands: NI, ZN, 9FJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-09-27
Ligands: NI, ZN, 9FJ
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Crystal Structure Of Benzamide Snx-1321 Bound To Hsp90
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2010-08-11 Classification: CHAPERONE Ligands: SD1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-08-11
Ligands: SD1
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Cdk2/Cyclina Complexed With A Pyrazolopyridazine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.15 Å Release Date: 2008-10-21 Classification: Transferase/Cell Cycle Ligands: PO5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-10-21
Ligands: PO5
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Cdk2/Cyclina Complexed With A Pyrazolopyridazine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.22 Å Release Date: 2008-10-21 Classification: Transferase/Cell cycle Ligands: 5BP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-10-21
Ligands: 5BP
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Crystal Structure Of Vegfr2 In Complex With A 3,4,5-Trimethoxy Aniline Containing Pyrimidine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2008-10-07 Classification: TRANSFERASE Ligands: SO4, SAV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-10-07
Ligands: SO4, SAV
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Crystal Structure Of Vegfr2 In Complex With A 3,4,5-Trimethoxy Aniline Containing Pyrimidine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2008-10-07 Classification: TRANSFERASE Ligands: SO4, KIM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-10-07
Ligands: SO4, KIM
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Crystal Structure Of Benzamide Tetrahydro-4H-Carbazol-4-One Bound To Hsp90
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.74 Å Release Date: 2008-06-17 Classification: CHAPERONE Ligands: SNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-06-17
Ligands: SNX
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Crystal Structure Of Vegfr2 With A Benzimidazole-Urea Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2007-09-18 Classification: TRANSFERASE Ligands: SO4, GIG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-09-18
Ligands: SO4, GIG
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Crystal Structure Of Vegfr2 In Complex With A 2-Anilino-5-Aryl-Oxazole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2005-06-07 Classification: TRANSFERASE Ligands: AAZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-06-07
Ligands: AAZ
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Crystal Structure Of Vegfr2 In Complex With A 2-Anilino-5-Aryl-Oxazole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2005-06-07 Classification: TRANSFERASE Ligands: AAX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-06-07
Ligands: AAX
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Cdk2 Complexed With N-Methyl-4-{[(2-Oxo-1,2-Dihydro-3H-Indol-3-Ylidene)Methyl]Amino}Benzenesulfonamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2002-05-14 Classification: TRANSFERASE Ligands: LS1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2002-05-14
Ligands: LS1
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Cyclin-Dependent Kinase 2 (Cdk2) Complexed With N-Methyl-{4-[2-(7-Oxo-6,7-Dihydro-8H-[1,3]Thiazolo[5,4-E]Indol-8-Ylidene)Hydrazino]Phenyl}Methanesulfonamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2002-05-14 Classification: TRANSFERASE Ligands: LS2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2002-05-14
Ligands: LS2
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Cyclin-Dependent Kinase 2 (Cdk2) Complexed With 3-{[(2,2-Dioxido-1,3-Dihydro-2-Benzothien-5-Yl)Amino]Methylene}-5-(1,3-Oxazol-5-Yl)-1,3-Dihydro-2H-Indol-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2002-05-14 Classification: TRANSFERASE Ligands: LS3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2002-05-14
Ligands: LS3
