Search Count: 25
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Kras-Wt(1-169) - Gdp In Complex With Compound (R)-1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.31 Å Release Date: 2025-07-23 Classification: HYDROLASE Ligands: MG, SO4, A1I89, GDP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-07-23
Ligands: MG, SO4, A1I89, GDP
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Kras-G12D(1-169) - Gdp In Covalent Complex With Compound (3R,4R)-3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2025-07-23 Classification: HYDROLASE Ligands: MG, SO4, A1I9E, GDP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-07-23
Ligands: MG, SO4, A1I9E, GDP
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Kras-G12D(1-169) - Gdp In Covalent Complex With Compound (3S,4R)-8
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.30 Å Release Date: 2025-07-23 Classification: HYDROLASE Ligands: MG, A1I9F, GDP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-07-23
Ligands: MG, A1I9F, GDP
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Kras G12C In Complex With Gdp And Compound 16
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2022-12-07 Classification: HYDROLASE Ligands: MG, NZ6, GDP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-12-07
Ligands: MG, NZ6, GDP
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Kras G12C In Complex With Gdp And Compound 9
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2022-12-07 Classification: HYDROLASE Ligands: MG, NZX, GDP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-12-07
Ligands: MG, NZX, GDP
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Crystal Structure Of Brd9 Bromodomain In Complex With Compound Ea-89
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.76 Å Release Date: 2022-08-10 Classification: TRANSCRIPTION Ligands: L8L |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-10
Ligands: L8L
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Krasg12C In Complex With Gdp And Jdq443
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.61 Å Release Date: 2022-04-27 Classification: HYDROLASE Ligands: MG, H2T, GDP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-04-27
Ligands: MG, H2T, GDP
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Krasg12C In Complex With Gdp And Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.20 Å Release Date: 2022-04-27 Classification: HYDROLASE Ligands: MG, H40, GDP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-04-27
Ligands: MG, H40, GDP
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Krasg12C In Complex With Gdp And Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2022-04-27 Classification: HYDROLASE Ligands: MG, H0O, GDP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-04-27
Ligands: MG, H0O, GDP
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Crystal Structure Of Brd4-Bd1 In Complex With Nvs-Bet-1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2020-12-23 Classification: TRANSCRIPTION Ligands: QFN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-23
Ligands: QFN
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Hdm2 (17-111, Wild Type) Complexed With Compound 12 At 1.8A; Structural States Of Hdm2 And Hdmx: X-Ray Elucidation Of Adaptations And Binding Interactions For Different Chemical Compound Classes
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2019-05-15 Classification: LIGASE Ligands: HRE, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-15
Ligands: HRE, SO4
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Hdm2 (17-111, Wild Type) Complexed With Compound 11 At 2.0A; Structural States Of Hdm2 And Hdmx: X-Ray Elucidation Of Adaptations And Binding Interactions For Different Chemical Compound Classes
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2019-05-15 Classification: LIGASE Ligands: HRH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-15
Ligands: HRH
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Hdm2 (17-111, Wildtype) Complexed With Compound 9 At 1.13A; Structural States Of Hdm2 And Hdmx: X-Ray Elucidation Of Adaptations And Binding Interactions For Different Chemical Compound Classes
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.13 Å Release Date: 2019-05-15 Classification: LIGASE Ligands: HTZ, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-15
Ligands: HTZ, CL
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Hdm2 (17-111, Wildtype) Complexed With Compound 10 At 1.21A; Structural States Of Hdm2 And Hdmx: X-Ray Elucidation Of Adaptations And Binding Interactions For Different Chemical Compound Classes
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.21 Å Release Date: 2019-05-15 Classification: LIGASE Ligands: HU8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-15
Ligands: HU8
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Hdmx (14-111; C17S) Complexed With Compound 13 At 2.1A; Structural States Of Hdm2 And Hdmx: X-Ray Elucidation Of Adaptations And Binding Interactions For Different Chemical Compound Classes
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2019-05-15 Classification: APOPTOSIS Ligands: HUE, O4B, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-15
Ligands: HUE, O4B, SO4, GOL
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Hdmx (14-111; C17S) Complexed With Compound 14 At 2.4A: Structural States Of Hdm2 And Hdmx: X-Ray Elucidation Of Adaptations And Binding Interactions For Different Chemical Compound Classes
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2019-05-15 Classification: APOPTOSIS Ligands: HRN, O4B, SO4, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-15
Ligands: HRN, O4B, SO4, NA
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Hdmx (14-111; C17S) Complexed With Compound 12 At 2.4A; Structural States Of Hdm2 And Hdmx: X-Ray Elucidation Of Adaptations And Binding Interactions For Different Chemical Compound Classes
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2019-05-15 Classification: APOPTOSIS Ligands: HRE, O4B, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-15
Ligands: HRE, O4B, CL
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X-Ray Structure Of Compound 15 Bound To Hdmx: Structural States Of Hdm2 And Hdmx: X-Ray Elucidation Of Adaptations And Binding Interactions For Different Chemical Compound Classes
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2019-05-15 Classification: APOPTOSIS Ligands: HRT, SO4, O4B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-15
Ligands: HRT, SO4, O4B
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Hdmx (14-111; C17S) Complexed With Compound 16 At 1.20A; Structural States Of Hdm2 And Hdmx: X-Ray Elucidation Of Adaptations And Binding Interactions For Different Chemical Compound Classes
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.20 Å Release Date: 2019-05-15 Classification: APOPTOSIS Ligands: HRQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-15
Ligands: HRQ
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In Vitro And In Vivo Characterization Of A Novel, Highly Potent P53-Mdm2 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2018-09-26 Classification: CELL CYCLE Ligands: EYH, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-09-26
Ligands: EYH, CL
