Search Count: 16
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Crystal Structure Of Parp1 Catalytic Domain Bound To Azd5305 (Saruparib)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2024-12-04 Classification: TRANSFERASE Ligands: A1H63, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-04
Ligands: A1H63, SO4
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Crystal Structure Of Parp1 Catalytic Domain Bound To Azd9574
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2024-12-04 Classification: TRANSFERASE Ligands: A1H64, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-04
Ligands: A1H64, SO4
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Crystal Structure Of Cdk9-Cyclin T1 Bound By Compound 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.81 Å Release Date: 2021-10-27 Classification: TRANSFERASE Ligands: UT5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-10-27
Ligands: UT5
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Parp1 Catalytic Domain In Complex With 8-Chloroquinazolinone-Based Inhibitor (Compound 9)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2021-09-15 Classification: TRANSFERASE Ligands: VKW, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-15
Ligands: VKW, SO4
 |
Parp1 Catalytic Domain In Complex With Isoquinolone-Based Inhibitor (Compound 16)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2021-09-15 Classification: TRANSFERASE Ligands: VKT, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-15
Ligands: VKT, SO4
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Parp1 Catalytic Domain In Complex With A Selective Pyridine Carboxamide-Based Inhibitor (Compound 22)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2021-09-15 Classification: TRANSFERASE Ligands: VKQ, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-15
Ligands: VKQ, SO4
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Oestrogen Receptor Ligand Binding Domain In Complex With Compound 16
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2021-01-20 Classification: GENE REGULATION Ligands: QNE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-20
Ligands: QNE
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Oestrogen Receptor Ligand Binding Domain In Complex With Compound 28
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2021-01-20 Classification: GENE REGULATION Ligands: QNH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-20
Ligands: QNH
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Oestrogen Receptor Ligand Binding Domain In Complex With Compound 18
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2021-01-20 Classification: GENE REGULATION Ligands: QNK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-20
Ligands: QNK
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Cdk9-Cyclin-T1 Complex Bound By Compound 24
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.37 Å Release Date: 2020-12-23 Classification: TRANSFERASE Ligands: Q6E, TRS, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-23
Ligands: Q6E, TRS, PO4
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Era_L536S (L536S/C381S/C471S,C530S) In Complex With A Bridged Tetracyclic Indole (Compound 8)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2019-10-30 Classification: GENE REGULATION Ligands: LRQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-10-30
Ligands: LRQ
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Era_L536S (L536S/C381S/C471S,C530S) In Complex With A Tricyclic Indole (Compound 6)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.74 Å Release Date: 2019-10-30 Classification: GENE REGULATION Ligands: LVH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-10-30
Ligands: LVH
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Crystal Structure Of Human Cdk12/Cyclink In Complex With An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.06 Å Release Date: 2017-12-27 Classification: TRANSFERASE/INHIBITOR Ligands: MG, CJM, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-27
Ligands: MG, CJM, EDO
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Pak1 In Complex With Bis-Anilino Pyrimidine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.58 Å Release Date: 2016-09-28 Classification: TRANSFERASE Ligands: IPV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-28
Ligands: IPV
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Pak1 In Complex With 7-Azaindole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.36 Å Release Date: 2016-09-28 Classification: TRANSFERASE Ligands: IPW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-28
Ligands: IPW
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Crystal Structure Of The Kinase Domain Of Human Pak1 In Complex With Compound 15
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2014-09-10 Classification: Transferase/Transferase inhibitor Ligands: 2K0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-09-10
Ligands: 2K0