Search Count: 30
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Structure Of Pou2F3 Pou Domains Bound To Coactivator Oca-T2 And Dna (2.8 Angstrom Resolution)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.79 Å Release Date: 2025-10-01 Classification: TRANSCRIPTION |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-10-01
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Structure Of Pou2F3 Pou Domains Bound To Coactivator Oca-T2 And Dna (2.1 Angstrom Resolution)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2025-10-01 Classification: TRANSCRIPTION |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-10-01
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Structure Of Pou2F3 Pou Domains Bound To Coactivator Oca-T1 And Dna
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2025-10-01 Classification: TRANSCRIPTION Ligands: BO3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-10-01
Ligands: BO3
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X-Ray Structure Of Nsd3-Pwwp1 In Complex With Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2019-06-26 Classification: ONCOPROTEIN Ligands: EH2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-26
Ligands: EH2
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X-Ray Structure Of Nsd3-Pwwp1 In Complex With Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.43 Å Release Date: 2019-06-26 Classification: ONCOPROTEIN Ligands: EHQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-26
Ligands: EHQ
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X-Ray Structure Of Nsd3-Pwwp1 In Complex With Compound 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2019-06-26 Classification: ONCOPROTEIN Ligands: EHE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-26
Ligands: EHE
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X-Ray Structure Of Nsd3-Pwwp1 In Complex With Compound 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2019-06-26 Classification: ONCOPROTEIN Ligands: EHK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-26
Ligands: EHK
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X-Ray Structure Of Nsd3-Pwwp1 In Complex With Compound 8
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.61 Å Release Date: 2019-06-26 Classification: ONCOPROTEIN Ligands: EH8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-26
Ligands: EH8
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X-Ray Structure Of Nsd3-Pwwp1 In Complex With Compound 9
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.76 Å Release Date: 2019-06-26 Classification: ONCOPROTEIN Ligands: EHT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-26
Ligands: EHT
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X-Ray Structure Of Nsd3-Pwwp1 In Complex With Compound 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2019-06-26 Classification: ONCOPROTEIN Ligands: EHH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-26
Ligands: EHH
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X-Ray Structure Of Nsd3-Pwwp1 In Complex With Compound 16
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.74 Å Release Date: 2019-06-26 Classification: ONCOPROTEIN Ligands: EHW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-26
Ligands: EHW
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X-Ray Structure Of Nsd3-Pwwp1 In Complex With Compound Bi-9321
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.81 Å Release Date: 2019-06-26 Classification: ONCOPROTEIN Ligands: EJE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-26
Ligands: EJE
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X-Ray Structure Of Seleno-Methionine Labelled Nsd3-Pwwp1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2019-06-26 Classification: ONCOPROTEIN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-26
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X-Ray Structure Of Nsd3-Pwwp1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.53 Å Release Date: 2019-06-26 Classification: ONCOPROTEIN Ligands: EPE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-26
Ligands: EPE
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Wdr5 In Complex With A Win Site Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2019-03-13 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: HH7, DMS, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-03-13
Ligands: HH7, DMS, SO4
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Wdr5 In Complex With A Win Site Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.56 Å Release Date: 2019-03-13 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: HHM, SO4, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-03-13
Ligands: HHM, SO4, DMS
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Discovery Of Potent 2-Aryl-6,7-Dihydro-5Hpyrrolo[ 1,2-A]Imidazoles As Wdr5 Win-Site Inhibitors Using Fragment-Based Methods And Structure-Based Design
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.22 Å Release Date: 2019-03-13 Classification: gene regulation/inhibitor Ligands: HLM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-03-13
Ligands: HLM
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Displacement Of Wdr5 From Chromatin By A Pharmacological Win Site Inhibitor With Picomolar Affinity
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.10 Å Release Date: 2019-03-13 Classification: gene regulation/inhibitor Ligands: HLP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-03-13
Ligands: HLP
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Displacement Of Wdr5 From Chromatin By A Pharmacological Win Site Inhibitor With Picomolar Affinity
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2019-03-13 Classification: gene regulation/inhibitor Ligands: HLS, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-03-13
Ligands: HLS, SO4
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Displacement Of Wdr5 From Chromatin By A Pharmacological Win Site Inhibitor With Picomolar Affinity
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.66 Å Release Date: 2019-03-13 Classification: gene regulation/inhibitor Ligands: HLJ, EPE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-03-13
Ligands: HLJ, EPE
