Structural Entry Filters:

Search Count: 10

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6GR9 image
Human Aurkc Incenp Complex Bound To Vx-680
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.25 Å Release Date: 2019-05-15
Classification: TRANSFERASE
Ligands: VX6, SO4


5WNM image
Crystal Structure Of Murine Receptor-Interacting Protein 4 (Ripk4) D143N Bound To Tozasertib (Vx-680)

4ZOG image
Vx-680/Mk-0457 Binds To Human Abl1 Also In Inactive Dfg Conformations.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.30 Å Release Date: 2016-09-14
Classification: TRANSFERASE
Ligands: VX6, MXE, MES

4B8M image
Aurora B Kinase In Complex With Vx-680

4JBQ image
Novel Aurora Kinase Inhibitors Reveal Mechanisms Of Hurp In Nucleation Of Centrosomal And Kinetochore Microtubules
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.30 Å Release Date: 2013-06-05
Classification: TRANSFERASE
Ligands: VX6

4AF3 image
Human Aurora B Kinase In Complex With Incenp And Vx-680

3AMB image
Protein Kinase A Sixfold Mutant Model Of Aurora B With Inhibitor Vx-680

3E5A image
Crystal Structure Of Aurora A In Complex With Vx-680 And Tpx2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.30 Å Release Date: 2008-10-28
Classification: TRANSFERASE
Ligands: VX6, SO4

2F4J image
Structure Of The Kinase Domain Of An Imatinib-Resistant Abl Mutant In Complex With The Aurora Kinase Inhibitor Vx-680
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.91 Å Release Date: 2006-01-24
Classification: TRANSFERASE
Ligands: VX6
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