Search Count: 10
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Human Aurkc Incenp Complex Bound To Vx-680
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2019-05-15 Classification: TRANSFERASE Ligands: VX6, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-15
Ligands: VX6, SO4
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Ddr1 Bound To Vx-680
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.23 Å Release Date: 2018-12-05 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: VX6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-12-05
Ligands: VX6
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Crystal Structure Of Murine Receptor-Interacting Protein 4 (Ripk4) D143N Bound To Tozasertib (Vx-680)
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2018-05-09 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: CL, VX6 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2018-05-09
Ligands: CL, VX6
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Vx-680/Mk-0457 Binds To Human Abl1 Also In Inactive Dfg Conformations.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2016-09-14 Classification: TRANSFERASE Ligands: VX6, MXE, MES |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-14
Ligands: VX6, MXE, MES
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Aurora B Kinase In Complex With Vx-680
Organism: Xenopus laevis
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2013-07-10 Classification: CELL CYCLE Ligands: VX6 |
Organism: Xenopus laevis
Method: X-RAY DIFFRACTION
Release Date: 2013-07-10
Ligands: VX6
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Novel Aurora Kinase Inhibitors Reveal Mechanisms Of Hurp In Nucleation Of Centrosomal And Kinetochore Microtubules
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2013-06-05 Classification: TRANSFERASE Ligands: VX6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-06-05
Ligands: VX6
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Human Aurora B Kinase In Complex With Incenp And Vx-680
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.75 Å Release Date: 2012-04-11 Classification: TRANSFERASE/INHIBITOR Ligands: VX6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-04-11
Ligands: VX6
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Protein Kinase A Sixfold Mutant Model Of Aurora B With Inhibitor Vx-680
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2011-08-03 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: VX6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-08-03
Ligands: VX6
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Crystal Structure Of Aurora A In Complex With Vx-680 And Tpx2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2008-10-28 Classification: TRANSFERASE Ligands: VX6, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-10-28
Ligands: VX6, SO4
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Structure Of The Kinase Domain Of An Imatinib-Resistant Abl Mutant In Complex With The Aurora Kinase Inhibitor Vx-680
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.91 Å Release Date: 2006-01-24 Classification: TRANSFERASE Ligands: VX6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-01-24
Ligands: VX6
