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Search Count: 26

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7NPK image
Alpha-1 Antitrypsin C232S Complexed With Cmpd3

7NPL image
Alpha-1 Antitrypsin (C232S) Complexed With Cmpd 11

7AEL image
Alpha 1-Antitrypsin (C232S) Complexed With Gsk716

6T6R image
Human Endoplasmic Reticulum Aminopeptidase 1 (Erap1) In Complex With (4Ar,5S,6R,8S,8Ar)-5-(2-(Furan-3-Yl)Ethyl)-8-Hydroxy-5,6,8A-Trimethyl-3,4,4A,5,6,7,8,8A-Octahydronaphthalene-1-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.67 Å Release Date: 2020-03-18
Classification: HYDROLASE
Ligands: ZN, MLT, EDO, MNZ

5NA5 image
Pseudomonas Fluorescens Kynurenine 3-Monooxygenase (Kmo) Apo Structure

5NAB image
Pseudomonas Fluorescens Kynurenine 3-Monooxygenase (Kmo) In Complex With 3-(5-Chloro-6-Methyl-2-Oxo-2,3-Dihydro-1,3-Benzoxazol-3-Yl)Propanoic Acid

5NAE image
Pseudomonas Fluorescens Kynurenine 3-Monooxygenase (Kmo) In Complex With 3-{5-Chloro-2-Oxo-6-[(1R)-1-(Pyridin-2-Yl)Ethoxy]-2,3-Dihydro-1,3-Benzoxazol-3-Yl}Propanoic Acid

5NAG image
Pseudomonas Fluorescens Kynurenine 3-Monooxygenase (Kmo) In Complex With 3-{5-Chloro-6-[(1R)-1-(Pyridin-2-Yl)Ethoxy]-1,2-Benzoxazol-3-Yl}Propanoic Acid

5NAH image
Pseudomonas Fluorescens Kynurenine 3-Monooxygenase (Kmo) In Complex With 3-{5-Chloro-6-[(1R)-1-(6-Methylpyridazin-3-Yl)Ethoxy]-1,2-Benzoxazol-3-Yl}Propanoic Acid

5NAK image
Pseudomonas Fluorescens Kynurenine 3-Monooxygenase (Kmo) In Complex With The Enzyme Substrate L-Kynurenine

5N7T image
Pseudomonas Fluorescens Kynurenine 3-Monooxygenase (Kmo) In Complex With 3-(5,6-Dichloro-2-Oxo-2,3-Dihydro-1,3-Benzoxazol-3-Yl)Propanoic Acid

5MZC image
Pseudomonas Fluorescens Kynurenine 3-Monooxygenase (Kmo) In Complex With 3-(5-Chloro-6-Ethoxy-2-Oxo-2,3-Dihydro-1,3-Benzoxazol-3-Yl)Propanoic Acid

5MZI image
Pseudomonas Fluorescens Kynurenine 3-Monooxygenase (Kmo) In Complex With 3-(5-Chloro-6-Cyclopropoxy-2-Oxo-2,3-Dihydro-1,3-Benzoxazol-3-Yl)Propanoic Acid

5MZK image
Pseudomonas Fluorescens Kynurenine 3-Monooxygenase (Kmo) In Complex With 3-[5-Chloro-6-(Cyclobutylmethoxy)-2-Oxo-2,3-Dihydro-1,3-Benzoxazol-3-Yl]Propanoic Acid

5FN0 image
Crystal Structure Of Pseudomonas Fluorescens Kynurenine-3- Monooxygenase (Kmo) In Complex With Gsk180

4C66 image
Discovery Of Epigenetic Regulator I-Bet762: Lead Optimization To Afford A Clinical Candidate Inhibitor Of The Bet Bromodomains
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.87 Å Release Date: 2013-10-02
Classification: CELL CYCLE
Ligands: H4C

4C67 image
Discovery Of Epigenetic Regulator I-Bet762: Lead Optimization To Afford A Clinical Candidate Inhibitor Of The Bet Bromodomains
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.55 Å Release Date: 2013-10-02
Classification: CELL CYCLE
Ligands: L5S, EDO

2YDW image
Crystal Structure Of The First Bromodomain Of Human Brd2 With The Inhibitor Gw841819X

2YEK image
Crystal Structure Of The First Bromodomain Of Human Brd2 With The Inhibitor Gsk525762 (Ibet)

2YEL image
Crystal Structure Of The First Bromodomain Of Human Brd4 With The Inhibitor Gw841819X
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