Search Count: 135
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Crystal Structure Of Apoform Human Usp18
Organism: Homo sapiens, Myxococcus xanthus (strain dk1622)
Method: X-RAY DIFFRACTION Resolution:1.92 Å Release Date: 2026-04-29 Classification: HYDROLASE Ligands: ZN |
Organism: Homo sapiens, Myxococcus xanthus (strain dk1622)
Method: X-RAY DIFFRACTION
Release Date: 2026-04-29
Ligands: ZN
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Crystal Structure Of Apoform Human Eif4A1 C-Terminal Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.73 Å Release Date: 2026-02-18 Classification: TRANSLATION |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-02-18
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Crystal Structure Of Human Eif4A1 C-Terminal Domain In Complex With Hippuristanol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2026-02-18 Classification: TRANSLATION Ligands: A1I1L |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-02-18
Ligands: A1I1L
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Crystal Structure Of Dhps In Complex With An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2024-11-20 Classification: TRANSFERASE Ligands: XTQ, EDO, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-11-20
Ligands: XTQ, EDO, DMS
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Crystal Structure Of Mnk2-D228G In Complex With Tinodasertib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.59 Å Release Date: 2024-06-12 Classification: TRANSFERASE Ligands: ZN, X8K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-06-12
Ligands: ZN, X8K
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Crystal Structure Of Ternary Complex Of Pol Theta Polymerase Domain
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.26 Å Release Date: 2022-10-12 Classification: TRANSFERASE Ligands: MG, DG3 |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2022-10-12
Ligands: MG, DG3
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Crystal Structure Of Pol Theta Polymerase Domain In Complex With Compound 5
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.99 Å Release Date: 2022-10-12 Classification: TRANSFERASE Ligands: MG, DG3, K7X |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2022-10-12
Ligands: MG, DG3, K7X
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Crystal Structure Of Pol Theta Polymerase Domain In Complex With Compound 22
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.83 Å Release Date: 2022-10-12 Classification: TRANSFERASE Ligands: MG, DG3, K8I |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2022-10-12
Ligands: MG, DG3, K8I
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Pgk1 In Complex With Crt0063465 (3-[2-(4-Bromophenyl)-5,7-Dimethyl-Pyrazolo[1,5-A]Pyrimidin-6-Yl]Propanoic Acid)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2018-05-16 Classification: TRANSFERASE Ligands: 93T, EDO, 3PG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-16
Ligands: 93T, EDO, 3PG
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Crystal Structure Of Usp7 In Complex With The Non-Covalent Inhibitor, Ft671
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2017-10-18 Classification: HYDROLASE Ligands: 8WK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-10-18
Ligands: 8WK
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Crystal Structure Of Usp7 In Complex With The Covalent Inhibitor, Ft827
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.33 Å Release Date: 2017-10-18 Classification: HYDROLASE Ligands: 8WN, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-10-18
Ligands: 8WN, EDO
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Crystal Structure Of Murine Autotaxin In Complex With A Small Molecule Inhibitor
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.92 Å Release Date: 2016-11-09 Classification: HYDROLASE Ligands: NAG, 6XN, ZN, SO4, CA, NA, K, EDO |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2016-11-09
Ligands: NAG, 6XN, ZN, SO4, CA, NA, K, EDO
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Human Pfkfb3 In Complex With An Indole Inhibitor 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.01 Å Release Date: 2015-04-22 Classification: TRANSFERASE Ligands: PO4, 8R2, FDP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: PO4, 8R2, FDP
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Human Pfkfb3 In Complex With An Indole Inhibitor 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2015-04-22 Classification: TRANSFERASE Ligands: PHS, PO4, F6P, S6L |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: PHS, PO4, F6P, S6L
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Human Pfkfb3 In Complex With An Indole Inhibitor 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.58 Å Release Date: 2015-04-22 Classification: TRANSFERASE Ligands: PHS, PO4, F6P, FD9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: PHS, PO4, F6P, FD9
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Human Pfkfb3 In Complex With An Indole Inhibitor 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.37 Å Release Date: 2015-04-22 Classification: TRANSFERASE Ligands: PHS, PO4, F6P, 87T |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: PHS, PO4, F6P, 87T
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Human Pfkfb3 In Complex With An Indole Inhibitor 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2015-04-22 Classification: TRANSFERASE Ligands: PHS, F6P, PO4, MJP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: PHS, F6P, PO4, MJP
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Human Pfkfb3 In Complex With An Indole Inhibitor 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.03 Å Release Date: 2015-04-22 Classification: TRANSFERASE Ligands: PHS, PO4, F6P, 8V1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: PHS, PO4, F6P, 8V1
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Identification Of Novel Hsp90/Isoform Selective Inhibitors Using Structure-Based Drug Design. Demonstration Of Potential Utility In Treating Cns Disorders Such As Huntington'S Disease
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2014-12-24 Classification: CHAPERONE/CHAPERONE INHIBITOR Ligands: 2Q8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-24
Ligands: 2Q8
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11B-Hydroxysteroid Dehydrogenase Type I In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.16 Å Release Date: 2014-09-03 Classification: OXIDOREDUCTASE Ligands: NAP, 4YQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-09-03
Ligands: NAP, 4YQ
