Search Count: 10
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Tead1 In Complex With A Reversible Inhibitor N-[(1S)-2-Hydroxy-1-(1-Methyl-1H-Pyrazol-3-Yl)Ethyl]-2-Methyl-8-[4-(Trifluoromethyl)Phenyl]-2H,8H-Pyrazolo[3,4-B]Indole-5-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.93 Å Release Date: 2025-01-22 Classification: TRANSCRIPTION Ligands: GOL, A1IJL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-22
Ligands: GOL, A1IJL, SO4
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Tead1/Yap In Complex With A Reversible Inhibitor N-[(4-Phenoxyphenyl)Methyl]Imidazo[1,2-A]Pyridine-3-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.21 Å Release Date: 2024-10-16 Classification: TRANSCRIPTION Ligands: CL, A1IHH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-16
Ligands: CL, A1IHH
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Optimization Of Tead P-Site Binding Fragment Hit Into In Vivo Active Lead Msc-4106
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.19 Å Release Date: 2022-07-13 Classification: TRANSCRIPTION Ligands: JJU, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-07-13
Ligands: JJU, SO4
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Human Tead3 In Complex With 1-Cyclopentyl-1H-Pyrazolo[3,4-B]Pyridine-5-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2022-07-13 Classification: TRANSCRIPTION Ligands: JIK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-07-13
Ligands: JIK
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Crystal Structure Of Murine Autotaxin In Complex With A Small Molecule Inhibitor
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.92 Å Release Date: 2016-11-09 Classification: HYDROLASE Ligands: NAG, 6XN, ZN, SO4, CA, NA, K, EDO |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2016-11-09
Ligands: NAG, 6XN, ZN, SO4, CA, NA, K, EDO
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Crystal Structure Of Human 17Beta-Hydroxysteroid Dehydrogenase Type 5 In Complex With (4-(4-Chlorophenyl)Piperazin-1-Yl)(Morpholino)Methanone (24)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2013-11-13 Classification: Oxidoreductase/Oxidoreductase inhibitor Ligands: NAP, 16J, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-11-13
Ligands: NAP, 16J, EDO
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Crystal Structure Of Human 17Beta-Hydroxysteroid Dehydrogenase Type 5 In Complex With 1-{4-[(2-Methyl-1-Piperidinyl)Sulfonyl]Phenyl}-2-Pyrrolidinone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2013-03-20 Classification: oxidoreductase/oxidoreductase inhibitor Ligands: NAP, 10H |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-20
Ligands: NAP, 10H
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Crystal Structure Of Human 17Beta-Hydroxysteroid Dehydrogenase Type 5 In Complex With (R)-1-(Naphthalen-2-Ylsulfonyl)Piperidine-3-Carboxylic Acid (86)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2012-10-10 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE inhibitor Ligands: NAP, 0SL, EDO, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-10-10
Ligands: NAP, 0SL, EDO, ACT
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Crystal Structure Of Human 17Beta-Hydroxysteroid Dehydrogenase Type 5 In Complex With 3-((3,4-Dihydroisoquinolin-2(1H)-Yl)Sulfonyl)-N-Methylbenzamide (80)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2012-10-10 Classification: oxidoreductase/oxidoreductase inhibitor Ligands: NAP, 0T0, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-10-10
Ligands: NAP, 0T0, EDO
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Crystal Structure Of Human 17Beta-Hydroxysteroid Dehydrogenase Type 5 In Complex With 3-((3,4-Dihydroisoquinolin-2(1H)-Yl)Sulfonyl)Benzoic Acid (17)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2012-10-10 Classification: oxidoreductase/oxidoreductase inhibitor Ligands: NAP, 0SZ, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-10-10
Ligands: NAP, 0SZ, EDO