Search Count: 10
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Crystal Structure Of 2-(3-Alkoxy-1-Azetidinyl) Quinolines As Pde10A Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.77 Å Release Date: 2014-12-17 Classification: Hydrolase/Hydrolase Inhibitor Ligands: SO4, GOL, 35E, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-17
Ligands: SO4, GOL, 35E, ZN
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2-(3-Alkoxy-1-Azetidinyl) Quinolines As Novel Pde10A Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2014-12-17 Classification: Hydrolase/Hydrolase Inhibitor Ligands: ZN, SO4, GOL, 35D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-17
Ligands: ZN, SO4, GOL, 35D
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Crystal Structure Of Pde10A With A Novel Imidazo[4,5-B]Pyridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.08 Å Release Date: 2014-10-01 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 1IS, 1IR, ZN, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-10-01
Ligands: 1IS, 1IR, ZN, SO4, GOL
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Crystal Structure Of Pde10A With 1H-Benzimidazol-2-Yl(4-((3-(Tetrahydro-2H-Pyran-4-Yl)-2-Pyridinyl)Oxy)Phenyl)Methanone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2014-08-06 Classification: Hydrolase/Hydrolase Inhibitor Ligands: ZN, SO4, 2W1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-08-06
Ligands: ZN, SO4, 2W1
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Crystal Structure Of Pde10A With Imidazo[4,5-B]Pyridines As Potent And Selective Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2014-07-23 Classification: HYDROLASE/HYDROLASE INBHITOR Ligands: ZN, SO4, GOL, 2KR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-23
Ligands: ZN, SO4, GOL, 2KR
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Crystal Structure Of Pde10A With Novel Keto-Benzimidazole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.64 Å Release Date: 2013-10-23 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, SO4, GOL, 2F4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-10-23
Ligands: ZN, SO4, GOL, 2F4
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Crystal Structure Of Pde10A With Novel Keto-Benzimidazole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2013-10-23 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, SO4, 2F5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-10-23
Ligands: ZN, SO4, 2F5
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Crystal Structure Of Pde10A With A Biaryl Ether Inhibitor ((1-(3-(4-((1H-Benzo[D]Imidazol-2-Yl)Amino)Phenoxy)Pyridin-2-Yl)Piperidin-4-Yl)Methanol)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2012-12-12 Classification: hydrolase/hydrolase inhibitor Ligands: ZN, SO4, 15J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-12-12
Ligands: ZN, SO4, 15J
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Crystal Structure Of Pde10A With A Biaryl Ether Inhibitor (1-(1-(3-(4-(Benzo[D]Thiazol-2-Ylamino)Phenoxy)Pyrazin-2-Yl)Piperidin-4-Yl)Ethanol)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2012-12-12 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, SO4, GOL, 15H |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-12-12
Ligands: ZN, SO4, GOL, 15H
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Pde10A Crystal Structure Complexed With Novel Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.07 Å Release Date: 2012-03-21 Classification: Hydrolase/Hydrolase Inhibitor Ligands: ZN, SO4, 0JQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-03-21
Ligands: ZN, SO4, 0JQ
