Search Count: 23
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Human Fgfr4 Kinase Domain (447-753) In Complex With Roblitinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.13 Å Release Date: 2020-09-30 Classification: TRANSFERASE Ligands: FGF, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-09-30
Ligands: FGF, SO4
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Fibroblast Growth Factor Receptor 4 Kinase Domain (449-753) In Complex With Irreversible Ligand Cga159527
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2018-04-04 Classification: HORMONE/GROWTH FACTOR Ligands: 99K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-04-04
Ligands: 99K
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Fibroblast Growth Factor Receptor 4 Kinase Domain (449-753) In Complex With Irreversible Ligand Cga159527
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.37 Å Release Date: 2018-04-04 Classification: HORMONE/GROWTH FACTOR Ligands: 9CT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-04-04
Ligands: 9CT
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Serine/Threonine-Protein Kinase Pak1 Complexed With A Dibenzodiazepine: Identification Of An Allosteric Site On Pak1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2015-08-05 Classification: Transferase/transferase inhibitor Ligands: 4PV, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-05
Ligands: 4PV, GOL
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Pak1 In Complex With 2-Chloro-5-Ethyl-8-Fluoro-11-(4-Methylpiperazin-1-Yl)-Dibenzodiazepine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2015-06-24 Classification: TRANSFERASE Ligands: 4OQ, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-24
Ligands: 4OQ, MG
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Pak1 In Complex With (S)-N-(Tert-Butyl)-3-((2-Chloro-5-Ethyl-8-Fluoro-Dibenzodiazepin-11-Yl)Amino)Pyrrolidine-1-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2015-06-24 Classification: TRANSFERASE Ligands: 4OR, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-24
Ligands: 4OR, MG
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Dpp4 Complexed With Syn-7Aa
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2014-02-12 Classification: HYDROLASE Ligands: NAG, SO4, 2KS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-02-12
Ligands: NAG, SO4, 2KS
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Dpp4 Complexed With Compound 12A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2014-02-12 Classification: HYDROLASE Ligands: NAG, SO4, 2KV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-02-12
Ligands: NAG, SO4, 2KV
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Crystal Structure Of Renin In Complex With Pkf909-724 (Compound 3)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2013-02-13 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, 0LU, SO4, 0LW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-02-13
Ligands: NAG, 0LU, SO4, 0LW
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Crystal Structure Of Renin In Complex With Gp055321 (Compound 4)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2013-02-13 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, 0M2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-02-13
Ligands: NAG, 0M2
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Crystal Structure Of Renin In Complex With Nvp-Ayl747 (Compound 5)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2013-02-13 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, 0M3, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-02-13
Ligands: NAG, 0M3, SO4
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Crystal Structure Of Renin In Complex With Nvp-Bbv031 (Compound 6)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.75 Å Release Date: 2013-02-13 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, 0ME, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-02-13
Ligands: NAG, 0ME, SO4
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Crystal Structure Of Renin In Complex With Nvp-Bch965 (Compound 9)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2013-02-13 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, 0MJ, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-02-13
Ligands: NAG, 0MJ, SO4
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Crystal Structure Of Renin In Complex With Nvp-Bgq311 (Compound 12)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2013-02-13 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, 0N0, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-02-13
Ligands: NAG, 0N0, SO4
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Crystal Structure Of Human Dpp4 In Complex With A Noval Heterocyclic Dpp4 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.62 Å Release Date: 2012-02-08 Classification: HYDROLASE Ligands: N7F, NAG, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-02-08
Ligands: N7F, NAG, SO4
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Crystal Structure Of Jak2 Complexed With A Potent Quinoxaline Atp Site Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2010-07-21 Classification: TRANSFERASE Ligands: DQX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-07-21
Ligands: DQX
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Crystal Structure Of The Human Clk3 In Complex With Dki
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.92 Å Release Date: 2009-10-20 Classification: TRANSFERASE Ligands: DKI, SO4, DMS, EDO, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-10-20
Ligands: DKI, SO4, DMS, EDO, CL
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Crystal Structure Of The Human Clk3 In Complex With V25
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2009-10-20 Classification: TRANSFERASE Ligands: V25, SO4, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-10-20
Ligands: V25, SO4, CL
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Crystal Structure Of Human Proto-Oncogene Serine Threonine Kinase (Pim1) In Complex With A Consensus Peptide And A Beta Carboline Ligand I
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2008-07-15 Classification: TRANSFERASE Ligands: CL, 7CP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-07-15
Ligands: CL, 7CP
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Crystal Structure Of Human Proto-Oncogene Serine Threonine Kinase (Pim1) In Complex With A Consensus Peptide And A Beta Carboline Ligand Ii
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.01 Å Release Date: 2008-07-15 Classification: TRANSFERASE Ligands: CL, MB9, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-07-15
Ligands: CL, MB9, EDO
