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2YIY image
Crystal Structure Of Compound 8 Bound To Tak1-Tab
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.49 Å Release Date: 2012-05-23
Classification: TRANSFERASE/TRANSFERASE ACTIVATOR
Ligands: YIY

3O0G image
Crystal Structure Of Cdk5:P25 In Complex With An Atp Analogue
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.95 Å Release Date: 2011-01-26
Classification: TRANSFERASE/TRANSFERASE ACTIVATOR
Ligands: 3O0

2EVA image
Structural Basis For The Interaction Of Tak1 Kinase With Its Activating Protein Tab1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.00 Å Release Date: 2006-05-02
Classification: TRANSFERASE/TRANSFERASE ACTIVATOR
Ligands: ADN

4ISG image
Human Glucokinase In Complex With Novel Activator (2S)-3-Cyclohexyl-2-[4-(Methylsulfonyl)-2-Oxopiperazin-1-Yl]-N-(1,3-Thiazol-2-Yl)Propanamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.65 Å Release Date: 2013-03-20
Classification: TRANSFERASE/TRANSFERASE ACTIVATOR
Ligands: GLC, 1FY, IOD

4ISE image
Human Glucokinase In Complex With Novel Activator (2S)-3-Cyclohexyl-2-(6-Fluoro-4-Oxoquinazolin-3(4H)-Yl)-N-(1,3-Thiazol-2-Yl)Propanamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.78 Å Release Date: 2013-03-20
Classification: TRANSFERASE/TRANSFERASE ACTIVATOR
Ligands: GLC, 1FW, IOD

4ISF image
Human Glucokinase In Complex With Novel Activator (2S)-3-Cyclohexyl-2-(6-Fluoro-2,4-Dioxo-1,4-Dihydroquinazolin-3(2H)-Yl)-N-(1,3-Thiazol-2-Yl)Propanamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.09 Å Release Date: 2013-03-20
Classification: TRANSFERASE/TRANSFERASE ACTIVATOR
Ligands: GLC, 1FX, IOD

3OTU image
Pdk1 Mutant Bound To Allosteric Disulfide Fragment Activator Js30
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.10 Å Release Date: 2011-03-23
Classification: TRANSFERASE/TRANSFERASE ACTIVATOR
Ligands: J30, BI4, SO4, CL

5V4X image
Human Glucokinase In Complex With Novel Pyrazole Activator.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.08 Å Release Date: 2017-05-31
Classification: transferase/transferase activator
Ligands: GLC, 8WJ, IOD

5V4W image
Human Glucokinase In Complex With Novel Indazole Activator.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.39 Å Release Date: 2017-05-31
Classification: transferase/transferase activator
Ligands: GLC, 8WM, IOD

3VEV image
Glucokinase In Complex With An Activator And Glucose
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.80 Å Release Date: 2012-02-08
Classification: TRANSFERASE/TRANSFERASE ACTIVATOR
Ligands: GLC, 0H4, NA

3VF6 image
Glucokinase In Complex With Glucose And Activator
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.86 Å Release Date: 2012-02-08
Classification: TRANSFERASE/TRANSFERASE ACTIVATOR
Ligands: GLC, 0H6, NA

3ORZ image
Pdk1 Mutant Bound To Allosteric Disulfide Fragment Activator 2A2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.00 Å Release Date: 2011-03-23
Classification: TRANSFERASE/TRANSFERASE ACTIVATOR
Ligands: 2A2, BI4

4MLE image
Human Glucokinase In Complex With Novel Amino Thiazole Activator
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.60 Å Release Date: 2013-09-25
Classification: TRANSFERASE/TRANSFERASE ACTIVATOR
Ligands: GLC, VO1

4MLH image
Human Glucokinase In Complex With A Novel Amino Thiazole Allosteric Activator
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.90 Å Release Date: 2013-09-25
Classification: TRANSFERASE/TRANSFERASE ACTIVATOR
Ligands: GLC, VO2

4DHY image
Crystal Structure Of Human Glucokinase In Complex With Glucose And Activator
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.38 Å Release Date: 2012-02-08
Classification: TRANSFERASE/TRANSFERASE ACTIVATOR
Ligands: GLC, S41, NA

4LQP image
Crystal Structure Of The Cbk1(T743E)-Mob2 Kinase-Coactivator Complex, In Crystal Form A
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION
Resolution:4.50 Å Release Date: 2014-07-30
Classification: TRANSFERASE/TRANSFERASE activator
Ligands: ANP

4LQQ image
Crystal Structure Of The Cbk1(T743E)-Mob2 Kinase-Coactivator Complex In Crystal Form B
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION
Resolution:3.60 Å Release Date: 2014-07-30
Classification: TRANSFERASE/TRANSFERASE activator
Ligands: ANP

4LQS image
Crystal Structure Of The Cbk1-Mob2 Kinase-Coactivator Complex
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION
Resolution:3.30 Å Release Date: 2014-07-30
Classification: TRANSFERASE/TRANSFERASE activator
Ligands: ANP

3U2Z image
Activator-Bound Structure Of Human Pyruvate Kinase M2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.10 Å Release Date: 2012-09-12
Classification: transferase/transferase activator
Ligands: FBP, UNX, 07T

4NO7 image
Human Glucokinase In Complex With A Nanomolar Activator.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.70 Å Release Date: 2014-10-29
Classification: TRANSFERASE/TRANSFERASE ACTIVATOR
Ligands: GLC, 2N8
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