Search Count: 15
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Erap1 In Complex With (3S,4S)-1-(3-Cyano-6-Methylpyridin-2-Yl)-4-(Propan-2-Yl)Pyrrolidine-3-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.87 Å Release Date: 2026-07-08 Classification: PEPTIDE BINDING PROTEIN Ligands: ZN, PO4, EDO, A1JVC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-08
Ligands: ZN, PO4, EDO, A1JVC
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Erap1 In Complex With (3R,4R)-1-(3-Cyano-6-Methylpyridin-2-Yl)-4-(Propan-2-Yl)Pyrrolidine-3-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2026-07-08 Classification: PEPTIDE BINDING PROTEIN Ligands: ZN, PO4, EDO, A1JVB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-08
Ligands: ZN, PO4, EDO, A1JVB
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Erap1 In Complex With (3R,4R)-1-[3-Cyano-6-(Cyclopropylamino)Pyridin-2-Yl]-4-(Propan-2-Yl)Pyrrolidine-3-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.73 Å Release Date: 2026-07-08 Classification: PEPTIDE BINDING PROTEIN Ligands: ZN, PO4, EDO, A1JVL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-08
Ligands: ZN, PO4, EDO, A1JVL
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Erap1 In Complex With (3R,4R)-1-{3-Cyano-4-Methyl-6-[(4-Methyloxan-4-Yl)Amino]Pyridin-2-Yl}-4-(Propan-2-Yl)Pyrrolidine-3-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.74 Å Release Date: 2026-07-08 Classification: PEPTIDE BINDING PROTEIN Ligands: ZN, PO4, EDO, A1JV2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-08
Ligands: ZN, PO4, EDO, A1JV2
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N-Terminal Bromodomain Of Human Brd4 With Ibet-Bd1 (Gsk778)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.28 Å Release Date: 2020-04-01 Classification: TRANSCRIPTION Ligands: GLU, LWB, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-01
Ligands: GLU, LWB, EDO
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C-Terminal Bromodomain Of Human Brd2 With Ibet-Bd1 (Gsk778)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2020-04-01 Classification: TRANSCRIPTION Ligands: LWB, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-01
Ligands: LWB, EDO
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C-Terminal Bromodomain Of Human Brd2 With Ibet-Bd2 (Gsk046)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2020-04-01 Classification: TRANSCRIPTION Ligands: EDO, LW5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-01
Ligands: EDO, LW5
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N-Terminal Bromodomain Of Human Brd4 With Ibet-Bd2 (Gsk046)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2020-04-01 Classification: TRANSCRIPTION Ligands: EDO, LW5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-01
Ligands: EDO, LW5
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1.68A Structure Pcaf Bromodomain With 4-Chloro-2-Methyl-5-(Methylamino)Pyridazin-3(2H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.68 Å Release Date: 2017-12-20 Classification: TRANSCRIPTION Ligands: 82I, SO4, EPE, BU1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-20
Ligands: 82I, SO4, EPE, BU1
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Bromodomain Of Human Brd9 With 4-Chloro-2-Methyl-5-((2-Methyl-1,2,3,4-Tetrahydroisoquinolin-5-Yl)Amino)Pyridazin-3(2H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.67 Å Release Date: 2017-12-20 Classification: TRANSCRIPTION Ligands: I0D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-20
Ligands: I0D
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N-Terminal Bromodomain Of Human Brd4 With 4-Chloro-2-Methyl-5-(((3-Methylthiophen-2-Yl)Methyl)Amino)Pyridazin-3(2H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.62 Å Release Date: 2017-12-20 Classification: TRANSCRIPTION Ligands: RNK, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-20
Ligands: RNK, GOL
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Bromodomain Of Mouse Pcaf With (R)-4-Chloro-2-Methyl-5-((1-Methylpiperidin-3-Yl)Amino)Pyridazin-3(2H)-One
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.64 Å Release Date: 2017-12-20 Classification: TRANSCRIPTION Ligands: P2L, EDO |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2017-12-20
Ligands: P2L, EDO
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N-Terminal Bromodomain Of Human Brd4 With 4-Chloro-2-Methyl-5-(Methylamino)Pyridazin-3(2H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2017-12-20 Classification: TRANSCRIPTION Ligands: 82I |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-20
Ligands: 82I
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Bromodomain Of Human Gcn5 With 4-Bromo-2-Methyl-5-(((3R,5R)-1-Methyl-5-Phenylpiperidin-3-Yl)Amino)Pyridazin-3(2H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2017-12-20 Classification: TRANSCRIPTION Ligands: EDO, 9ST |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-20
Ligands: EDO, 9ST
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Bromodomain Of Trypanosoma Brucei Bdf2 With Ibet-151
Organism: Trypanosoma brucei brucei
Method: X-RAY DIFFRACTION Resolution:1.25 Å Release Date: 2015-11-18 Classification: SIGNALING PROTEIN/INHIBITOR Ligands: 1GH, PO4, K, CL, GOL |
Organism: Trypanosoma brucei brucei
Method: X-RAY DIFFRACTION
Release Date: 2015-11-18
Ligands: 1GH, PO4, K, CL, GOL
