Structural Entry Filters:

Search Count: 26

Download
7MGJ image
Tnni3K Complexed With N-Methyl-4-(4-(3-(3-(Trifluoromethyl) Phenyl) Ureido) Phenoxy)Picolinamide

7MGK image
Tnni3K Complexed With 1-(3,5-Dichloro-4-((6-(Methylamino)Pyrimidin-4-Yl)Oxy)Phenyl)-3-(3-(Trifluoromethyl)Phenyl)Urea

6RLN image
Crystal Structure Of Rip1 Kinase In Complex With Gsk3145095
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.87 Å Release Date: 2019-07-03
Classification: TRANSFERASE
Ligands: K8K

6OCQ image
Crystal Structure Of Rip1 Kinase In Complex With A Pyrrolidine

6R5F image
Crystal Structure Of Rip1 Kinase In Complex With Dhp77
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:3.25 Å Release Date: 2019-05-01
Classification: TRANSFERASE
Ligands: JSW

6HMX image
Rip2 Kinase Catalytic Domain Complex With N(4,5Dimethyl1Hpyrazol3Yl)7Methoxy6(2Methylpropane2Sulfonyl)Quinolin4Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.53 Å Release Date: 2018-11-07
Classification: TRANSFERASE
Ligands: GEZ

5TX5 image
Rip1 Kinase ( Flag 1-294, C34A, C127A, C233A, C240A) With Gsk772

5J79 image
The Identification And Pharmacological Characterization Of 6-(Tert-Butylsulfonyl)-N-(5-Fluoro-1H-Indazol-3-Yl)Quinolin-4-Amine (Gsk583), A Highly Potent And Selective Inhibitor Of Rip2 Kinase, Compound 3 Complex

5J7B image
The Identification And Pharmacological Characterization Of 6-(Tert-Butylsulfonyl)-N-(5-Fluoro-1H-Indazol-3-Yl)Quinolin-4-Amine (Gsk583), A Highly Potent And Selective Inhibitor Of Rip2 Kinase, Gsk583 Complex

5HX6 image
Crystal Structure Of Rip1 Kinase With A Benzo[B][1,4]Oxazepin-4-One

4YZ9 image
Crystal Structure Of Human Phosphorylated Ire1Alpha In Complex With A Type Iii Kinase Inhibitor (Gsk2850163A)

4YZC image
Crystal Structure Of Pire1Alpha In Complex With Staurosporine

4YZD image
Crystal Structure Of Human Phosphorylated Ire1Alpha In Complex With Adp-Mg
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:3.10 Å Release Date: 2015-11-11
Classification: TRANSFERASE
Ligands: MG, ADP

5AR2 image
Rip2 Kinase Catalytic Domain (1 - 310)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.44 Å Release Date: 2015-10-21
Classification: TRANSFERASE
Ligands: CA

5AR3 image
Rip2 Kinase Catalytic Domain (1 - 310) Complex With Amp-Pcp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:3.23 Å Release Date: 2015-10-21
Classification: TRANSFERASE
Ligands: ACP, MG

5AR4 image
Rip2 Kinase Catalytic Domain (1 - 310) Complex With Sb-203580
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.70 Å Release Date: 2015-10-21
Classification: TRANSFERASE
Ligands: SB2

5AR5 image
Rip2 Kinase Catalytic Domain (1 - 310) Complex With Benzimidazole
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.66 Å Release Date: 2015-10-21
Classification: TRANSFERASE
Ligands: CA, IQ7

5AR7 image
Rip2 Kinase Catalytic Domain (1 - 310) Complex With Biaryl Urea
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.71 Å Release Date: 2015-10-21
Classification: TRANSFERASE
Ligands: SR8

5AR8 image
Rip2 Kinase Catalytic Domain (1 - 310) Complex With Biphenylsulfonamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.79 Å Release Date: 2015-10-21
Classification: TRANSFERASE
Ligands: XYW

4YFF image
Tnni3K Complexed With Inhibitor 2
Protein Functional Filters:
Feedback Form
Name
Email
Institute
Feedback