Search Count: 28
 |
Krasg12C Ligand Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.18 Å Release Date: 2022-04-20 Classification: SIGNALING PROTEIN Ligands: V4T, MG, GDP, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-04-20
Ligands: V4T, MG, GDP, CA
 |
Krasg12C Ligand Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.38 Å Release Date: 2022-04-20 Classification: SIGNALING PROTEIN Ligands: MG, GDP, V52, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-04-20
Ligands: MG, GDP, V52, CA
 |
Krasg12C Ligand Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.48 Å Release Date: 2022-04-20 Classification: SIGNALING PROTEIN Ligands: MG, GDP, VLE, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-04-20
Ligands: MG, GDP, VLE, CA
 |
Krasg12C Ligand Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.37 Å Release Date: 2020-02-26 Classification: SIGNALING PROTEIN Ligands: MG, GDP, O7K, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-02-26
Ligands: MG, GDP, O7K, SO4
 |
Krasg12C Ligand Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2020-02-19 Classification: SIGNALING PROTEIN Ligands: MG, GDP, MKW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-02-19
Ligands: MG, GDP, MKW
 |
Krasg12C Ligand Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.31 Å Release Date: 2020-02-19 Classification: SIGNALING PROTEIN Ligands: MG, GDP, MKZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-02-19
Ligands: MG, GDP, MKZ
 |
Human Erk2 With Erk1/2 Inhibitor, Azd0364.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.33 Å Release Date: 2019-11-20 Classification: TRANSFERASE Ligands: LHZ, SO4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-20
Ligands: LHZ, SO4, EDO
 |
Human Erk2 With An Erk1/2 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.74 Å Release Date: 2017-04-19 Classification: TRANSFERASE Ligands: SO4, 8X2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-04-19
Ligands: SO4, 8X2
 |
Human Erk2 With An Erk1/2 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.14 Å Release Date: 2017-04-19 Classification: TRANSFERASE Ligands: SO4, 8X5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-04-19
Ligands: SO4, 8X5
 |
Human Erk2 With An Erk1/2 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2017-04-19 Classification: TRANSFERASE Ligands: SO4, 8XH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-04-19
Ligands: SO4, 8XH
 |
Human Erk2 With An Erk1/2 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.12 Å Release Date: 2017-04-19 Classification: TRANSFERASE Ligands: SO4, 8XE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-04-19
Ligands: SO4, 8XE
 |
Human Erk2 With An Erk1/2 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.07 Å Release Date: 2017-04-19 Classification: TRANSFERASE Ligands: SO4, 8XB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-04-19
Ligands: SO4, 8XB
 |
Human Erk2 With An Erk1/2 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2017-04-19 Classification: TRANSFERASE Ligands: SO4, 8XN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-04-19
Ligands: SO4, 8XN
 |
Human Erk2 With An Erk1/2 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2017-04-19 Classification: TRANSFERASE Ligands: SO4, 8XK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-04-19
Ligands: SO4, 8XK
 |
Human Erk2 With An Erk1/2 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2017-04-19 Classification: TRANSFERASE Ligands: SO4, 8QB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-04-19
Ligands: SO4, 8QB
 |
Crystal Structure Of Iso-Citrate Dehydrogenase R132H In Complex With A Novel Inhibitor (Compound 13A)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2016-12-14 Classification: OXIDOREDUCTASE Ligands: NDP, 6N3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-12-14
Ligands: NDP, 6N3
 |
Crystal Structure Of Iso-Citrate Dehydrogenase 1 [Idh1 (R132H)] In Complex With A Novel Inhibitor (Compound 2)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.04 Å Release Date: 2016-12-14 Classification: OXIDOREDUCTASE Ligands: NDP, 6MX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-12-14
Ligands: NDP, 6MX
 |
A Novel Oral Selective Estrogen Receptor Down-Regulator, Azd9496, Drives Tumour Growth Inhibition In Estrogen Receptor Positive And Esr1 Mutant Models
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2015-12-16 Classification: SIGNALING PROTEIN Ligands: KE9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-12-16
Ligands: KE9
 |
Optimization Of A Novel Binding Motif To To (E)-3-(3,5-Difluoro-4-((1R,3R)-2-(2-Fluoro-2-Methylpropyl)-3-Methyl-2,3,4,9-Tetrahydro-1H- Pyrido(3,4-B)Indol-1-Yl)Phenyl)Acrylic Acid (Azd9496), A Potent And Orally Bioavailable Selective Estrogen Receptor Downregulator And Antagonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2015-10-14 Classification: SIGNALING PROTEIN Ligands: XBR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-14
Ligands: XBR
 |
Optimization Of A Novel Binding Motif To To (E)-3-(3,5-Difluoro-4-((1R,3R)-2-(2-Fluoro-2-Methylpropyl)-3-Methyl-2,3,4,9-Tetrahydro-1H- Pyrido(3,4-B)Indol-1-Yl)Phenyl)Acrylic Acid (Azd9496), A Potent And Orally Bioavailable Selective Estrogen Receptor Downregulator And Antagonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2015-10-14 Classification: SIGNALING PROTEIN Ligands: GW5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-14
Ligands: GW5