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Search Count: 24

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8Q6F image
Human Pi4Kiiib In Complex With Covalently Bound Inhibitor (Compound 4)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.51 Å Release Date: 2023-12-13
Classification: TRANSFERASE
Ligands: KHR, MG, EDO, GOL

8Q6G image
Human Pi4Kiiib In Complex With Covalently Bound Inhibitor (Compound 8)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.54 Å Release Date: 2023-12-13
Classification: TRANSFERASE
Ligands: KIH, MG, EDO

8Q6H image
Human Pi4Kiiib In Complex With Covalently Bound Inhibitor (Compound 11)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.94 Å Release Date: 2023-12-13
Classification: TRANSFERASE
Ligands: MG, KI7, EDO

7QDL image
N-Terminal Bromodomain Of Human Brd4 With I-Bet567

7QDT image
Crystal Structure Of A Mutant (P393Gx) Thyroid Receptor Alpha Ligand Binding Domain Designed To Model Dominant Negative Human Mutations.

7P4S image
Bromodomain Of Human Taf1 (2) With Naphthyridinone Compound

7P6V image
N-Terminal Bromodomain Of Human Brd4 With Compound 3Ag

7P6W image
N-Terminal Bromodomain Of Human Brd4 With Compound 3Bg

7P6Y image
N-Terminal Bromodomain Of Human Brd4 With Compound 5Ef

7OE8 image
C-Terminal Bromodomain Of Human Brd2 With N5-((1R,5S,6R)-3-Oxabicyclo[3.1.0]Hexan-6-Yl)-3-(1H-Indol-4-Yl)-N7-Methyl-2,3-Dihydrobenzofuran-5,7-Dicarboxamide

7OE9 image
C-Terminal Bromodomain Of Human Brd2 With Rac-N5-((1R,5S)-3-Oxabicyclo[3.1.0]Hexan-6-Yl)-N7,3-Dimethyl-3-Phenyl-2,3-Dihydrobenzofuran-5,7-Dicarboxamide

6YQW image
Brd9 With 4-Chloro-2-Methyl-Methylamino-Pyridazinone

6YQR image
Brd9 With Biphenyl-Methylamino-Dimethylpyridazinone

6YQS image
Brd9 With Methylpiperazinyl-Benzyl-Amino-Dimethylpyridazinone

6YQZ image
N-Terminal Domain Of Brd4 With Biphenyl-Methyamino-Dimethylpyridazinone

7A9U image
N-Terminal Bromodomain Of Human Brd4 With 3-(3-(But-3-Yn-1-Yl)-3H-Diazirin-3-Yl)-N-(3-Methyl-[1,2,4]Triazolo[4,3-A]Pyridin-8-Yl)Propanamide

6YB4 image
Crystal Structure Of Human Atad2 Bromodomain In Complex With N-(4-Bromo-3-(3-Methylpyrrolidin-1-Yl)Sulfonyl)Phenyl)-2-(-4-Cyclopropyl-4-Methyl-2,5-Dioxoimidazolidin-1-Yl)Acetamide

4UIT image
Bromodomain Of Human Brd9 With 7-(3,4-Dimethoxyphenyl)-2-(4- Methanesulfonylpiperazine-1-Carbonyl)-5-Methyl-4H,5H-Thieno-3,2-C- Pyridin-4-One

4UIU image
Bromodomain Of Human Brd9 With 7-(3,4-Dimethoxyphenyl)-N-(1,1-Dioxo-1- Thian-4-Yl)-5-Methyl-4-Oxo-4H,5H-Thieno-3,2-C-Pyridine-2-Carboxamide

4UIV image
Bromodomain Of Human Brd9 With N-(1,1-Dioxo-1-Thian-4-Yl)-5-Methyl-4- Oxo-7-3-(Trifluoromethyl)Phenyl-4H,5H-Thieno-3,2-C-Pyridine-2- Carboximidamide
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