Search Count: 26
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Adam-8 Metalloproteinase Domain With Bound Batimastat
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2012-06-06 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: BAT, CA, ZN, NA, CL, K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-06-06
Ligands: BAT, CA, ZN, NA, CL, K
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Crystal Structure Of Human Mmp-13 Complexed With An Amino-2-Indanol Compound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2011-02-02 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: CA, ZN, SO4, LA3, EPE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-02-02
Ligands: CA, ZN, SO4, LA3, EPE
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Caspase 3 Bound To A Covalent Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2010-08-11 Classification: HYDROLASE Ligands: B92 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-08-11
Ligands: B92
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Caspase 8 Bound To A Covalent Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2010-08-11 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: DTT, B93 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-08-11
Ligands: DTT, B93
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Caspase 8 With Covalent Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2010-08-11 Classification: HYDROLASE Ligands: B94 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-08-11
Ligands: B94
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Structural And Thermodynamic Characterization Of The Tyk2 And Jak3 Kinase Domains In Complex With Cp-690550 And Cmp-6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2010-06-02 Classification: TRANSFERASE Ligands: MI1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-06-02
Ligands: MI1
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Structural And Thermodynamic Characterization Of The Tyk2 And Jak3 Kinase Domains In Complex With Cp-690550 And Cmp-6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.74 Å Release Date: 2010-06-02 Classification: TRANSFERASE Ligands: IZA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-06-02
Ligands: IZA
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Structural And Thermodynamic Characterization Of The Tyk2 And Jak3 Kinase Domains In Complex With Cp-690550 And Cmp-6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2010-06-02 Classification: TRANSFERASE Ligands: MI1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-06-02
Ligands: MI1
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Structural And Thermodynamic Characterization Of The Tyk2 And Jak3 Kinase Domains In Complex With Cp-690550 And Cmp-6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2010-06-02 Classification: TRANSFERASE Ligands: IZA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-06-02
Ligands: IZA
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Crystal Structure Of The Catalytic Domain Of Adamts-5 In Complex With An Amino-2-Indanol Compound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2010-03-31 Classification: HYDROLASE Ligands: LA3, EDO, ZN, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-03-31
Ligands: LA3, EDO, ZN, CA
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Crystal Structure Of The Catalytic Domain Of Adamts-5 In Complex With Marimastat
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2009-07-07 Classification: HYDROLASE Ligands: 097, ZN, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-07-07
Ligands: 097, ZN, CA
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Crystal Structure Of The Catalytic Domain Of Adamts-5 In Complex With An Amino-2-Indanol Compound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.02 Å Release Date: 2009-07-07 Classification: HYDROLASE Ligands: ZN, CA, 098 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-07-07
Ligands: ZN, CA, 098
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Crystal Structure Of The Catalytic Domain Of Adamts-5 In Complex With An Amino-2-Indanol Compound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2009-07-07 Classification: HYDROLASE Ligands: ZN, CA, 099 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-07-07
Ligands: ZN, CA, 099
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Potent And Selective Isophthalamide S2 Hydroxyethylamine Inhibitor Of Bace1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2007-06-19 Classification: HYDROLASE Ligands: PO4, MR0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-06-19
Ligands: PO4, MR0
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Crystal Structure Of Hydroxyethyl Secondary Amine-Based Peptidomimetic Inhibitor Of Human Beta-Secretase (Bace)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2007-02-27 Classification: HYDROLASE Ligands: F2I |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-02-27
Ligands: F2I
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Crystal Structure Of Human Beta-Secretase (Bace) In The Presence Of An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2007-01-23 Classification: HYDROLASE Ligands: PO4, LIJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-01-23
Ligands: PO4, LIJ
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Crystal Structure Of Human Beta-Secretase (Bace) In The Presence Of An Inhibitor (2)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2007-01-23 Classification: HYDROLASE Ligands: LIQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-01-23
Ligands: LIQ
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Crystal Structure Of The Complex Of Caspase-8 With The Tetrapeptide Inhibitor Ace-Ietd-Aldehyde
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.20 Å Release Date: 2000-09-20 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: DTD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2000-09-20
Ligands: DTD
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Hiv-1 Protease Complex With U095438 [3-[1-(4-Bromophenyl) Isobutyl]-4-Hydroxycoumarin
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:2.22 Å Release Date: 1996-10-14 Classification: HYDROLASE (ACID PROTEASE) Ligands: U01 |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 1996-10-14
Ligands: U01
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Hiv-1 Protease Complex With U100313 ([3-[[3-[Cyclopropyl [4-Hydroxy-2Oxo-6-[1-(Phenylmethyl)Propyl]-2H-Pyran-3-Yl] Methyl]Phenyl]Amino]-3-Oxo-Propyl]Carbamic Acid Tert-Butyl Ester)
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 1996-10-14 Classification: HYDROLASE (ACID PROTEASE) Ligands: U02 |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 1996-10-14
Ligands: U02
