Search Count: 13
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Stx-478, A Mutant-Selective, Allosteric Inhibitor Bound To Pi3Kalpha
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.11 Å Release Date: 2023-09-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: X3N, ZWE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-09-06
Ligands: X3N, ZWE
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Stx-478, A Mutant-Selective, Allosteric Inhibitor Bound To H1047R Pi3Kalpha
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.93 Å Release Date: 2023-09-06 Classification: TRANSFERASE/TRANSFERSE INHIBITOR Ligands: EDO, X3N, ZWE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-09-06
Ligands: EDO, X3N, ZWE
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Crystal Structure Of Mth1 In Complex With Compound 31
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.13 Å Release Date: 2021-11-03 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: ZRP, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-11-03
Ligands: ZRP, SO4
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Crystal Structure Of Mth1 In Complex With Compound 32
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2021-11-03 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: ZRV, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-11-03
Ligands: ZRV, SO4
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Crystal Structure Of 6-Phosphogluconate Dehydrogenase With ((4R,5R)-5-(Hydroxycarbamoyl)-2,2-Dimethyl-1,3-Dioxolan-4-Yl)Methyl Dihydrogen Phosphate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2018-08-22 Classification: OXIDOREDUCTASE Ligands: 8HS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-22
Ligands: 8HS
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Crystal Structure Of Trim24 Phd-Bromodomain Complexed With 1-Methyl-5-(2-Methyl-1 3-Thiazol-4-Yl)-2 3-Dihydro-1H-Indol-2-One (1)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2015-06-24 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: ZN, 4CN, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-24
Ligands: ZN, 4CN, SO4
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Crystal Structure Of Trim24 Phd-Bromodomain Complexed With 2,4-Dimethoxy-N-(1-Methyl-2-Oxo-1,2,3,4-Tetrahydroquinolin-6-Yl)Benzene-1-Sulfonamide (3B)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.73 Å Release Date: 2015-06-24 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: ZN, 4A7, GOL, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-24
Ligands: ZN, 4A7, GOL, CL
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Crystal Structure Of Trim24 Phd-Bromodomain Complexed With N-(1,3-Dimethyl-2-Oxo-2,3-Dihydro-1H-1,3-Benzodiazol-5-Yl)-4-Methoxybenzene-1-Sulfonamide (5B)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.18 Å Release Date: 2015-06-24 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: ZN, 4A8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-24
Ligands: ZN, 4A8
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Crystal Structure Of Trim24 Phd-Bromodomain Complexed With N-[6-(4-Methoxyphenoxy)-1,3-Dimethyl-2-Oxo-2,3-Dihydro-1H-1,3-Benzodiazol-5-Yl]Benzenesulfonamide (5G)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2015-06-24 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: 4AE, ZN, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-24
Ligands: 4AE, ZN, GOL, SO4
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Crystal Structure Of Trim24 Phd-Bromodomain Complexed With N-{6-[3-(Benzyloxy)Phenoxy]-1,3-Dimethyl-2-Oxo-2,3-Dihydro-1H-1,3-Benzodiazol-5-Yl}-3,4-Dimethoxybenzene-1-Sulfonamide (7B)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.46 Å Release Date: 2015-06-24 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: ZN, GOL, 4BJ, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-24
Ligands: ZN, GOL, 4BJ, SO4
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Crystal Structure Of Trim24 Phd-Bromodomain Complexed With N-{1,3-Dimethyl-6-[3-(2-Methylpropoxy)Phenoxy]-2-Oxo-2,3-Dihydro-1H-1,3-Benzodiazol-5-Yl}-1,2-Dimethyl-1H-Imidazole-4-Sulfonamide (7G)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2015-06-24 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: ZN, 4BK, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-24
Ligands: ZN, 4BK, DMS
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Crystal Structure Of Trim24 Phd-Bromodomain Complexed With N-{1,3-Dimethyl-2-Oxo-6-[3-(Oxolan-3-Ylmethoxy)Phenoxy]-2,3-Dihydro-1H-1,3-Benzodiazol-5-Yl}-1-Methyl-1H-Imidazole-4-Sulfonamide (7L)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2015-06-24 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: ZN, DMS, 4BV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-24
Ligands: ZN, DMS, 4BV
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Crystal Structure Of Trim24 Phd-Bromodomain Complexed With N-(6-{3-[4-(Dimethylamino)Butoxy]-5-Propoxyphenoxy}-1,3-Dimethyl-2-Oxo-2,3-Dihydro-1H-1,3-Benzodiazol-5-Yl)-3,4-Dimethoxybenzene-1-Sulfonamide (8I)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2015-06-24 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: ZN, GOL, 4C1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-24
Ligands: ZN, GOL, 4C1