Search Count: 26
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Human P300 Complexed With A Proline-Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2022-11-09 Classification: TRANSFERASE/INHIBITOR Ligands: ZN, EDO, C0C |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-09
Ligands: ZN, EDO, C0C
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Human P300 Complexed With A Glycine-Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.36 Å Release Date: 2022-11-09 Classification: TRANSFERASE/INHIBITOR Ligands: ZN, EDO, C3I, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-09
Ligands: ZN, EDO, C3I, ACT
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Human P300 Complexed With An Azaindazole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2022-11-09 Classification: TRANSFERASE/INHIBITOR Ligands: ETL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-09
Ligands: ETL
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Pi3 Kinase Delta In Complex With 5-[3,6-Dihydro-2H-Pyran-4-Yl]-2-Methoxy-N-[2-Methylpyridin-4-Yl]Pyridine-3-Sulfonamide
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2021-09-29 Classification: SIGNALING PROTEIN Ligands: 7VT |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2021-09-29
Ligands: 7VT
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Pi3 Kinase Delta In Complex With N-[2-(2-Fluoro-4-{[4-(Propan-2-Yl)Piperazin-1-Yl]Methyl}Phenyl)Pyridin-4-Yl]-2-Methoxy-5-(Morpholin-4-Yl)Pyridine-3-Sulfonamide
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.26 Å Release Date: 2021-09-29 Classification: SIGNALING PROTEIN Ligands: 7XH |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2021-09-29
Ligands: 7XH
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Pi3 Kinase Delta In Complex With 5-(3,6-Dihydro-2H-Pyran-4-Yl)-2-Methoxy-N-(5-{3-[4-(Propan-2-Yl)Piperazin-1-Yl]Prop-1-Yn-1-Yl}Pyridin-3-Yl)Pyridine-3-Sulfonamide
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2021-09-29 Classification: SIGNALING PROTEIN Ligands: 7XN |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2021-09-29
Ligands: 7XN
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Pi3 Kinase Delta In Complex With N-[5-(3,6-Dihydro-2H-Pyran-4-Yl)-2-Methoxypyridin-3-Yl]Benzenesulfonamide
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.39 Å Release Date: 2021-09-29 Classification: SIGNALING PROTEIN Ligands: 7XW |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2021-09-29
Ligands: 7XW
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Cell Penetrant Inhibitors Of The Jmjd2 (Kdm4) And Jarid1 (Kdm5) Families Of Histone Lysine Demethylases
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2016-01-27 Classification: OXIDOREDUCTASE Ligands: YC8, ZN, MG, BCN, CO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-01-27
Ligands: YC8, ZN, MG, BCN, CO
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Crystal Structure Of Human Kdm4D In Complex With 3-(4- Phenylbutanamido)Pyridine-4-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2016-01-27 Classification: TRANSCRIPTION Ligands: ZN, FE2, GOL, YC8, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-01-27
Ligands: ZN, FE2, GOL, YC8, SO4
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Crystal Structure Of Human Kdm4D In Complex With 3-4-Methylthiophen-2- Ylmethylaminopyridine-4-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2016-01-27 Classification: OXIDOREDUCTASE Ligands: ZN, CO, AUY, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-01-27
Ligands: ZN, CO, AUY, SO4
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Crystal Structure Of Human Kdm4D In Complex With 3-Aminopyridine-4- Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2016-01-27 Classification: OXIDOREDUCTASE Ligands: ZN, CO, GOL, 4SV, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-01-27
Ligands: ZN, CO, GOL, 4SV, SO4
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Crystal Structure Of Human Kdm4D In Complex With 3H,4H-Pyrido-3,4-D- Pyrimidin-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.96 Å Release Date: 2016-01-27 Classification: OXIDOREDUCTASE Ligands: ZN, CO, N5J, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-01-27
Ligands: ZN, CO, N5J, SO4
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Crystal Structure Of Human Kdm4D In Complex With 2-1H-Pyrazol-4-Yloxy- 3H,4H-Pyrido-3,4-D-Pyrimidin-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.91 Å Release Date: 2016-01-27 Classification: OXIDOREDUCTASE Ligands: ZN, CO, HA6, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-01-27
Ligands: ZN, CO, HA6, SO4
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Structure Of Nek2 Bound To Aminipyrazine Compound 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2010-11-03 Classification: TRANSFERASE Ligands: WI2, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-11-03
Ligands: WI2, CL
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Structure Of Nek2 Bound To Aminopyrazine Compound 35
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2010-10-27 Classification: TRANSFERASE Ligands: XK3, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-10-27
Ligands: XK3, CL
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Structure Of Nek2 Bound To Aminopyrazine Compound 17
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2010-10-27 Classification: TRANSFERASE Ligands: OL2, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-10-27
Ligands: OL2, CL
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Structure Of Nek2 Bound To Aminopyrazine Compound 36
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2010-10-27 Classification: TRANSFERASE Ligands: EQH, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-10-27
Ligands: EQH, CL
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Structure Of Nek2 Bound To Aminopyrazine Compound 23
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2010-10-27 Classification: TRANSFERASE Ligands: 30E, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-10-27
Ligands: 30E, CL
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Structure Of Nek2 Bound To Aminopyrazine Compound 15
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2010-10-27 Classification: TRANSFERASE Ligands: 5R1, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-10-27
Ligands: 5R1, CL
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Structure Of Nek2 Bound To Aminopyrazine Compound 14
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2010-10-27 Classification: TRANSFERASE Ligands: 4VQ, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-10-27
Ligands: 4VQ, CL
