Search Count: 29
![]() |
Solution Nmr Structure Of The Pacs1 Furin Binding Region (Fbr)
Organism: Homo sapiens
Method: SOLUTION NMR Release Date: 2026-04-08 Classification: PROTEIN TRANSPORT |
Organism: Homo sapiens
Method: SOLUTION NMR
Release Date: 2026-04-08
![]() |
Structure Of The Complex Formed By Human Interleukin-2 And Scfv F10
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.71 Å Release Date: 2024-09-04 Classification: CYTOKINE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-09-04
![]() |
Structure Of The Complex Formed By Human Interleukin-2 And Scfv 602
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.64 Å Release Date: 2024-09-04 Classification: CYTOKINE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-09-04
![]() |
The Dbc1/Sirt1 Interaction Is Choreographed By Post-Translational Modification
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2024-03-27 Classification: GENE REGULATION |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-03-27
![]() |
1.4A Structure Of Drosophila Melanogaster Frataxin
Organism: Drosophila melanogaster
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2022-06-22 Classification: METAL TRANSPORT, Oxidoreductase Ligands: SO4 |
Organism: Drosophila melanogaster
Method: X-RAY DIFFRACTION
Release Date: 2022-06-22
Ligands: SO4
![]() |
Crystal Structure Of Beta-Site App-Cleaving Enzyme 1 Complexed With N-(3-((4As,7As)-2-Amino-4,4A,5,6-Tetrahydro-7Ah-Furo[2,3-D][1,3]Thiazin-7A-Yl)-4-Fluorophenyl)-5-Bromo-2-Pyridinecarboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.51 Å Release Date: 2016-11-23 Classification: HYDROLASE Ligands: 7H3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-23
Ligands: 7H3
![]() |
Compound 10
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2016-10-05 Classification: Hydrolase/Hydrolase Inhibitor Ligands: GOL, IOD, 5QU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-10-05
Ligands: GOL, IOD, 5QU
![]() |
(4~{S},6~{S})-4-[2,4-Bis(Fluoranyl)Phenyl]-4-Methyl-6-Pyrimidin-5-Yl-5,6-Dihydro-1,3-Thiazin-2-Amine (Compound 12) Bound To Bace1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2016-09-07 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 6WD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-07
Ligands: 6WD
![]() |
(4~{S},6~{S})-4-[2,4-Bis(Fluoranyl)Phenyl]-6-(3,5-Dimethyl-1,2-Oxazol-4-Yl)-4-Methyl-5,6-Dihydro-1,3-Thiazin-2-Amine (Compound 5) Bound To Bace1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.12 Å Release Date: 2016-09-07 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: IOD, 6WE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-07
Ligands: IOD, 6WE
![]() |
Compound 18
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.11 Å Release Date: 2016-07-06 Classification: Hydrolase/Hydrolase Inhibitor Ligands: GOL, IOD, 5QV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-07-06
Ligands: GOL, IOD, 5QV
![]() |
Human Tau Tubulin Kinase 1 (Ttbk1)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.12 Å Release Date: 2014-02-05 Classification: TRANSFERASE Ligands: GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-02-05
Ligands: GOL
![]() |
Human Tau Tubulin Kinase 1 (Ttbk1) Complexed With 3-({5-[(4-Amino-4-Methylpiperidin-1-Yl)Methyl]Pyrrolo[2,1-F][1,2,4]Triazin-4-Yl}Amino)-5-Bromophenol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.42 Å Release Date: 2014-02-05 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 2KC, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-02-05
Ligands: 2KC, SO4
![]() |
Crystal Structure Of Beta-Site App-Cleaving Enzyme 1 (Bace-Wt) Complex With N-(N-(4-Amino-3,5- Dichlorobenzyl)Carbamimidoyl)-3-(4-Methoxyphenyl)-5- Methyl-4-Isothiazolecarboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2012-10-10 Classification: HYDROLASE/INHIBITOR Ligands: 0VA, IOD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-10-10
Ligands: 0VA, IOD
![]() |
Crystal Structure Of Beta-Site App-Cleaving Enzyme 1 (Bace-Db-Mut) Complex With N-(N-(4- Acetamido-3-Chloro-5-Methylbenzyl)Carbamimidoyl)-3-(4- Methoxyphenyl)-5-Methyl-4-Isothiazolecarboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2012-10-10 Classification: HYDROLASE/INHIBITOR Ligands: 0VB, IOD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-10-10
Ligands: 0VB, IOD
![]() |
Crystal Structure Of Beta-Site App-Cleaving Enzyme 1 (Bace-Wt) Complex With (2S)-2-((3R)-3-Acetamido-3-Isobutyl-2-Oxo-1-Pyrrolidinyl)-N-((1S,2R)-1-(3,5-Difluorobenzyl)-2-Hydroxy-2-(1,2,3,4-Tetrahydro-3-Isoquinolinyl)Ethyl)-4-Phenylbutanamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.88 Å Release Date: 2011-09-07 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: PB8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-09-07
Ligands: PB8
![]() |
Crystal Structure Of Beta-Site App-Cleaving Enzyme 1 (Bace-Wt) Complex With Bms-693391 Aka (2S)-2-((3R)-3-Acetamido-3-Isobutyl-2-Oxo-1-Pyrrolidinyl)-N-((1S,2R)-1-(3,5-Difluorobenzyl)-2-Hydroxy-2-((2R,4R)-4-Propoxy-2-Pyrrolidinyl)Ethyl)-4-Phenylbutanamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.53 Å Release Date: 2011-08-31 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: PB0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-08-31
Ligands: PB0
![]() |
Crystal Structure Of Beta-Site App-Cleaving Enzyme 1 (Bace-Wt) Complex With (2S)-2-((3S)-3-(Acetylamino)-3-(Butan-2-Yl)-2-Oxopyrrolidin-1-Yl)-N-((2S,3R)-3-Hydroxy-4-((3-Methoxybenzyl)Amino)-1-Phenylbutan-2-Yl)-4-Phenylbutanamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2011-08-31 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: PB7, IOD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-08-31
Ligands: PB7, IOD
![]() |
Crystal Structure Of Plasminogen Activator Inhibitor-1 In A Metastable Active Conformation.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2011-06-22 Classification: HYDROLASE INHIBITOR Ligands: CL, ZN, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-06-22
Ligands: CL, ZN, EDO
![]() |
Crystal Structure Of Plasminogen Activator Inhibitor-1 In A Metastable Active Conformation.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.64 Å Release Date: 2011-06-22 Classification: HYDROLASE INHIBITOR Ligands: ZN, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-06-22
Ligands: ZN, CL
![]() |
Crystal Structure Of Beta-Site App-Cleaving Enzyme 1 (Bace-Wt) Complex With Bms-655295 Aka N~3~-((1S,2R)-1- Benzyl-2-Hydroxy-3-((3-Methoxybenzyl)Amino)Propyl)-N~1~, N~1~-Dibutyl-1H-Indole-1,3-Dicarboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2011-04-06 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 3HF, IOD, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-04-06
Ligands: 3HF, IOD, GOL
