Search Count: 45
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Crystal Structure Of Mammalian Ric-8A:Galpha(I):Nanobody Complex
Organism: Rattus norvegicus, Lama glama
Method: X-RAY DIFFRACTION Resolution:3.30 Å Release Date: 2020-03-11 Classification: SIGNALING PROTEIN |
Organism: Rattus norvegicus, Lama glama
Method: X-RAY DIFFRACTION
Release Date: 2020-03-11
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Cryo-Em Structure Of Mammalian Ric-8A:Galpha(I):Nanobody Complex
Organism: Rattus norvegicus, Lama glama
Method: ELECTRON MICROSCOPY Release Date: 2020-03-11 Classification: SIGNALING PROTEIN |
Organism: Rattus norvegicus, Lama glama
Method: ELECTRON MICROSCOPY
Release Date: 2020-03-11
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Crystal Structure Of Human Interleukin-1 Receptor Associated Kinase 4 (Irak 4, Cid 100300) In Complex With Compound Ncc00371481 (Bsi 107591)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2019-10-16 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: JX4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-10-16
Ligands: JX4, EDO
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Fumarate Hydratase Of Mycobacterium Tuberculosis In Complex With Formate And Allosteric Modulator N-(5-(Azocan-1-Ylsulfonyl)-2-Methoxyphenyl)-2-(4-Oxo-3,4-Dihydrophthalazin-1-Yl)Acetamide
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:1.42 Å Release Date: 2019-09-25 Classification: LYASE Ligands: KUE, FMT, MG |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2019-09-25
Ligands: KUE, FMT, MG
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Fumarate Hydratase Of Mycobacterium Tuberculosis In Complex With Formate And Allosteric Modulator N-(2-Methoxy-5-(N-Methylsulfamoyl)Phenyl)-2-(4-Oxo-3,4-Dihydrophthalazin-1-Yl)Acetamide
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2019-09-25 Classification: LYASE Ligands: KYZ, FMT, MG |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2019-09-25
Ligands: KYZ, FMT, MG
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Fumarate Hydratase Of Mycobacterium Tuberculosis In Complex With Formate And Allosteric Modulator N-(2-Methoxy-5-(N-Phenylsulfamoyl)Phenyl)-2-(4-Oxo-3,4-Dihydrophthalazin-1-Yl)Acetamide
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2019-09-25 Classification: LYASE Ligands: KZ8, FMT |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2019-09-25
Ligands: KZ8, FMT
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Fumarate Hydratase Of Mycobacterium Tuberculosis In Complex With Formate And Allosteric Modulator N-(5-(Azepan-1-Ylsulfonyl)-2-Methoxyphenyl)-2-(1H-Indol-3-Yl)Acetamide
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:1.48 Å Release Date: 2019-09-25 Classification: LYASE Ligands: KZK, FMT, MG |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2019-09-25
Ligands: KZK, FMT, MG
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Fumarate Hydratase Of Mycobacterium Tuberculosis In Complex With Formate And Allosteric Modulator N-(5-(Azepan-1-Ylsulfonyl)-2-Methoxyphenyl)-2-(Quinolin-4-Yl)Acetamide
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:1.44 Å Release Date: 2019-09-25 Classification: LYASE Ligands: KZT, FMT, MG |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2019-09-25
Ligands: KZT, FMT, MG
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Fumarate Hydratase Of Mycobacterium Tuberculosis In Complex With Formate And Allosteric Modulator N-(5-((3,4-Dihydroisoquinolin-2(1H)-Yl)Sulfonyl)-2-Methoxyphenyl)-2-(4-Oxo-3,4-Dihydrophthalazin-1-Yl)Acetamide
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2019-09-25 Classification: LYASE Ligands: KZN, MG, FMT |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2019-09-25
Ligands: KZN, MG, FMT
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Fumarate Hydratase Of Mycobacterium Tuberculosis In Complex With Formate And Allosteric Modulator N-(2-Methoxy-5-((1,2,4,5-Tetrahydro-3H-Benzo[D]Azepin-3-Yl)Sulfonyl)Phenyl)-2-(4-Oxo-3,4-Dihydrophthalazin-1-Yl)Acetamide
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2019-09-25 Classification: LYASE Ligands: L0K, FMT, MG |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2019-09-25
Ligands: L0K, FMT, MG
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Crystal Structure Of The Flt3 Kinase Bound To A Small Molecule Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2018-12-12 Classification: TRANSFERASE Ligands: A9R, PO4, CXS, GOL, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-12-12
Ligands: A9R, PO4, CXS, GOL, CL
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Crystal Structure Of Human O-Glcnac Transferase Bound To A Peptide From Hcf-1 Pro-Repeat 2 (11-26) And Inhibitor 4A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.75 Å Release Date: 2018-10-17 Classification: transferase/transferase inhibitor Ligands: JA4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-17
Ligands: JA4
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Crystal Structure Of Human O-Glcnac Transferase Bound To A Peptide From Hcf-1 Pro-Repeat 2 (11-26) And Inhibitor Ent-1A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2018-10-17 Classification: transferase/transferase inhibitor Ligands: J9S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-17
Ligands: J9S
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Crystal Structure Of Human O-Glcnac Transferase Bound To A Peptide From Hcf-1 Pro-Repeat 2 (11-26) And Inhibitor 2A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2018-10-17 Classification: transferase/transferase inhibitor Ligands: JAJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-17
Ligands: JAJ
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Crystal Structure Of Human O-Glcnac Transferase Bound To A Peptide From Hcf-1 Pro-Repeat 2 (11-26) And Inhibitor 3A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2018-10-17 Classification: transferase/transferase inhibitor Ligands: JA7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-17
Ligands: JA7
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Crystal Structure Of Human O-Glcnac Transferase Bound To A Peptide From Hcf-1 Pro-Repeat 2 (11-26) And Inhibitor 1A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2018-10-17 Classification: transferase/transferase inhibitor Ligands: J9V |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-17
Ligands: J9V
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Fumarate Hydratase Of Mycobacterium Tuberculosis In Complex With Formate And Allosteric Modulator (N-(5-(Azepan-1-Ylsulfonyl)-2-Methoxyphenyl)-2-(4-Oxo-3,4-Dihydrophthalazin-1-Yl)Acetamide)
Organism: Mycobacterium tuberculosis (strain cdc 1551 / oshkosh)
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2016-06-22 Classification: LYASE/LYASE INHIBITOR Ligands: 5WJ, CL, FMT |
Organism: Mycobacterium tuberculosis (strain cdc 1551 / oshkosh)
Method: X-RAY DIFFRACTION
Release Date: 2016-06-22
Ligands: 5WJ, CL, FMT
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Fumarate Hydratase Of Mycobacterium Tuberculosis In Complex With Formate
Organism: Mycobacterium tuberculosis (strain cdc 1551 / oshkosh)
Method: X-RAY DIFFRACTION Resolution:1.86 Å Release Date: 2016-06-22 Classification: LYASE Ligands: FMT, CL, PG4 |
Organism: Mycobacterium tuberculosis (strain cdc 1551 / oshkosh)
Method: X-RAY DIFFRACTION
Release Date: 2016-06-22
Ligands: FMT, CL, PG4
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Crystal Structure Of Hiv-1 Reverse Transcriptase In Complex With Rilpivirine (Tmc278) Based Analogue
Organism: Human immunodeficiency virus type 1 bh10
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2013-01-16 Classification: HYDROLASE, TRANSFERASE/INHIBITOR Ligands: G73 |
Organism: Human immunodeficiency virus type 1 bh10
Method: X-RAY DIFFRACTION
Release Date: 2013-01-16
Ligands: G73
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Crystal Structure Of K103N/Y181C Mutant Of Hiv-1 Reverse Transcriptase In Complex With Rilpivirine (Tmc278) Analogue
Organism: Human immunodeficiency virus type 1 bh10
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2013-01-16 Classification: HYDROLASE, TRANSFERASE/INHIBITOR Ligands: 1BT, EDO |
Organism: Human immunodeficiency virus type 1 bh10
Method: X-RAY DIFFRACTION
Release Date: 2013-01-16
Ligands: 1BT, EDO
