Structural Entry Filters:

Search Count: 36

Download
9TF9 image
Pdgfra-G680R Mutant Kinase Domain In Complex With Avapritinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.20 Å Release Date: 2026-07-15
Classification: TRANSFERASE
Ligands: 9JI

9TFA image
Pdgfra-G680R Mutant Kinase Domain In Complex With A 6,7-Dimethoxyquinazoline-Based Compound (43)

9TFB image
Pdgfra-G680R Mutant Kinase Domain In Complex With A 6,7-Bis(2-Methoxyethoxy)Quinazoline-Based Compound (44)

9TFC image
Pdgfra-G680R Mutant Kinase Domain In Complex With A 7-Methoxyquinazolin-6-Ol-Based Compound (45)

9TFD image
Kit Kinase Domain In Complex With A Pyrrolotriazine-Based Compound (11)

9TFE image
Kit Kinase Domain In Complex With An Aminopyrimidine-Based Compound (15)

9TFF image
Kit Kinase Domain In Complex With A Pyrrolopyrimidine-Based Compound (17)

9TFG image
Kit Kinase Domain In Complex With A 6-,7-Dimethoxyquinoline-Based Compound (19)

9TFH image
Kit Kinase Domain In Complex With A 7-Methylquinazoline-Based Compound (25)

9TFI image
Kit Kinase Domain In Complex With A 6,7-Bis(2-Methoxyethoxy)Quinazoline-Based Compound (33)

9TFJ image
Kit Kinase Domain In Complex With A 6,7-Dimethoxyquinazoline-Based Compound (34)

9TFK image
Kit Kinase Domain In Complex With A Quinoline-3-Carbonitrile-Based Compound (38)

9TFL image
Kit Kinase Domain In Complex With A Methyl Quinazoline-7-Carboxylate-Based Compound (41)

9TFM image
Kit Kinase Domain In Complex With A 7-Methoxyquinazolin-6-Ol-Based Compound (45)

8S13 image
Apo C-Kit-Wt Kinase Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.00 Å Release Date: 2025-09-03
Classification: TRANSFERASE
Ligands: EDO

8S14 image
C-Kit Kinase Domain In Complex With Sunitinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.50 Å Release Date: 2025-09-03
Classification: TRANSFERASE
Ligands: B49, EDO, CL

8S15 image
C-Kit Kinase Domain In Complex With Nintedanib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.40 Å Release Date: 2025-09-03
Classification: TRANSFERASE
Ligands: XIN

8S16 image
C-Kit Kinase Domain In Complex With Imatinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.85 Å Release Date: 2025-09-03
Classification: TRANSFERASE
Ligands: STI, CL

8S17 image
C-Kit Kinase Domain In Complex With Ponatinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.20 Å Release Date: 2025-09-03
Classification: TRANSFERASE
Ligands: 0LI, CL

8S18 image
C-Kit Kinase Domain In Complex With S116836
Protein Functional Filters:
Feedback Form
Name
Email
Institute
Feedback