Search Count: 21
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The Discovery Of A Novel Anticoagulant Mechanism: Factor Xi Activation Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.22 Å Release Date: 2026-07-29 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: A1CJA, NAG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-29
Ligands: A1CJA, NAG
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Ndm1-Inhibitor Co-Structure
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION Resolution:0.99 Å Release Date: 2023-03-08 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ACT, CA, ZN, CD, O0L |
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION
Release Date: 2023-03-08
Ligands: ACT, CA, ZN, CD, O0L
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Ndm1-Inhibitor Co-Structure
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION Resolution:1.47 Å Release Date: 2023-03-08 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, CD, O0F |
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION
Release Date: 2023-03-08
Ligands: ZN, CD, O0F
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Ndm1-Inhibitor Co-Structure
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION Resolution:1.11 Å Release Date: 2023-03-08 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, CD, NZR |
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION
Release Date: 2023-03-08
Ligands: ZN, CD, NZR
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Ndm1-Inhibitor Co-Structure
Organism: Pseudomonas aeruginosa
Method: X-RAY DIFFRACTION Resolution:1.13 Å Release Date: 2023-03-08 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, NZR |
Organism: Pseudomonas aeruginosa
Method: X-RAY DIFFRACTION
Release Date: 2023-03-08
Ligands: ZN, NZR
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Ndm1-Inhibitor Co-Structure
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2023-03-08 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: CD, ZN, NZ0, EPE |
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION
Release Date: 2023-03-08
Ligands: CD, ZN, NZ0, EPE
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Pcsk9 In Complex With Compound 16
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.53 Å Release Date: 2019-11-06 Classification: HYDROLASE/HYDROLASE Inhibitor Ligands: 063 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-06
Ligands: 063
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Pcsk9 In Complex With Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2019-11-06 Classification: HYDROLASE Ligands: PV7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-06
Ligands: PV7
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Pcsk9 In Complex With Compound 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2019-11-06 Classification: HYDROLASE Ligands: EDO, PUV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-06
Ligands: EDO, PUV
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Pcsk9 In Complex With A Fab And Compound 14
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2019-11-06 Classification: HYDROLASE/Immune System Ligands: PVM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-06
Ligands: PVM
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Pcsk9 In Complex With A Fab And Compound 8
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.73 Å Release Date: 2019-11-06 Classification: HYDROLASE/Immune System Ligands: PVJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-06
Ligands: PVJ
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Pcsk9 In Complex With Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.64 Å Release Date: 2019-11-06 Classification: HYDROLASE Ligands: PVV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-06
Ligands: PVV
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Irak4-Inhibitor Co-Structure
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2016-08-17 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: 6YD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-08-17
Ligands: 6YD
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Irak4-Inhibitor Co-Structure
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.67 Å Release Date: 2016-08-17 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6YE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-08-17
Ligands: 6YE
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Irak4-Inhibitor Co-Structure
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.39 Å Release Date: 2015-09-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 4S1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-02
Ligands: 4S1
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Irak4-Inhibitor Co-Structure
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.66 Å Release Date: 2015-09-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 4S2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-02
Ligands: 4S2
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Irak4-Inhibitor Co-Structure
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.23 Å Release Date: 2015-09-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 4S3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-02
Ligands: 4S3
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Irak4-Inhibitor Co-Structure
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.32 Å Release Date: 2015-05-20 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 4GD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-05-20
Ligands: 4GD
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Irak4-Inhibitor Co-Structure
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.64 Å Release Date: 2015-05-20 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 4GF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-05-20
Ligands: 4GF
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Structure Of E. Coli Fabf(C163Q) In Complex With Dihydroplatensimycin
Organism: Escherichia coli
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2009-03-17 Classification: TRANSFERASE Ligands: P9A |
Organism: Escherichia coli
Method: X-RAY DIFFRACTION
Release Date: 2009-03-17
Ligands: P9A
