Search Count: 17
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Crystal Structure Of Wild Type Egfr In Complex With Tak-788
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.61 Å Release Date: 2022-12-07 Classification: HYDROLASE Ligands: R28 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-12-07
Ligands: R28
 |
Crystal Structure Of Egfr_D770_N771Insnpg/V948R In Complex With Tak-788
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2022-12-07 Classification: HYDROLASE/HYDROLASE Inhibitor Ligands: R28, EDO, CIT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-12-07
Ligands: R28, EDO, CIT
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Crystal Structure Of Wnk1 In Complex With 1-Cyclohexyl-N-({6-Fluoro-1-[2-(3-Methoxyphenyl)Pyridin-4-Yl]-1H-Indol-3-Yl}Methyl)Methanamine (Compound 6)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.46 Å Release Date: 2017-08-16 Classification: TRANSFERASE Ligands: ANP, A6S, MN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-08-16
Ligands: ANP, A6S, MN
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Crystal Structure Of Wnk1 In Complex With N-{(3R)-1-[(4-Chlorophenyl)Methyl]Pyrrolidin-3-Yl}-2-(3-Methoxyphenyl)-N-Methylquinoline-4-Carboxamide (Compound 8)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.01 Å Release Date: 2017-08-16 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: MN, ANP, A7Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-08-16
Ligands: MN, ANP, A7Y
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Rock 1 Bound To Thiazole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.20 Å Release Date: 2015-06-10 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 4KH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-10
Ligands: 4KH
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Rock 1 Bound To Methoxyphenyl Thiazole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.40 Å Release Date: 2015-06-10 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 4KK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-10
Ligands: 4KK
 |
Rock 1 Bound To A Pyridine Thiazole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.95 Å Release Date: 2015-06-10 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 4TW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-10
Ligands: 4TW
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Crystal Structure Of Human Glucokinase In Complex With A Synthetic Activator
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2009-10-06 Classification: TRANSFERASE Ligands: GLC, B84, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-10-06
Ligands: GLC, B84, NA
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Jnk3 Bound To (Z)-1-((6-Fluoro-4H-Benzo[D][1,3]Dioxin-8-Yl)Methyl)-3-(Hydroxyimino)-4-Styrylindolin-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2009-04-28 Classification: TRANSFERASE Ligands: J67 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-04-28
Ligands: J67
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Jnk-3 Bound To (Z)-5-Fluoro-1-((6-Fluoro-4H-Benzo[D][1,3]Dioxin-8-Yl)Methyl)-3-(Hydroxyimino)Indolin-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2009-02-24 Classification: TRANSFERASE Ligands: J72 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-02-24
Ligands: J72
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Jnk3 Bound To (Z)-1-((6-Fluoro-4H-Benzo[D][1,3]Dioxin-8-Yl)Methyl)-3-(Hydroxyimino)-4-Phenylindolin-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2009-02-24 Classification: TRANSFERASE Ligands: J88 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-02-24
Ligands: J88
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Discovery And Sar Of Novel 4-Thiazolyl-2-Phenylaminopyrimidines As Potent Inhibitors Of Spleen Tyrosine Kinase (Syk)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2008-12-02 Classification: TRANSFERASE Ligands: 685 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-12-02
Ligands: 685
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Crystal Structure Of Rock I Bound To H-1152P A Di-Methylated Variant Of Fasudil
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.30 Å Release Date: 2008-06-10 Classification: TRANSFERASE Ligands: H52 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-06-10
Ligands: H52
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Crystal Structure Of C-Amp Dependent Kinase (Pka) Bound To Hydroxyfasudil
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2005-11-08 Classification: TRANSFERASE Ligands: HFS |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2005-11-08
Ligands: HFS
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Crystal Structure Of Rock 1 Bound To Fasudil
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.20 Å Release Date: 2005-11-08 Classification: TRANSFERASE Ligands: M77 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-11-08
Ligands: M77
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Crystal Structure Of Rock 1 Bound To Hydroxyfasudil
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.96 Å Release Date: 2005-11-08 Classification: TRANSFERASE Ligands: HFS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-11-08
Ligands: HFS
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Crystal Structure Of Rock I Bound To Y-27632
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2005-11-08 Classification: TRANSFERASE Ligands: Y27 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-11-08
Ligands: Y27