Search Count: 15
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Crystal Structure Of Pqsr Co-Inducer Binding Domain Of Pseudomonas Aeruginosa With Inhibitor 3Nh2-7Cl-C9Qzn
Organism: Pseudomonas aeruginosa
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2013-08-07 Classification: TRANSCRIPTION REGULATOR/INHIBITOR Ligands: QZN |
Organism: Pseudomonas aeruginosa
Method: X-RAY DIFFRACTION
Release Date: 2013-08-07
Ligands: QZN
 |
Brd4 First Bromodomain (Bd1) In Complex With Dual Pi3 Kinase Inhibitor Sf2523
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2017-02-08 Classification: TRANSCRIPTION REGULATOR/INHIBITOR Ligands: 82V, PEG, SCN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-08
Ligands: 82V, PEG, SCN
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Brd4 First Bromodomain (Bd1) In Complex With Dual Pi3 Kinase (Pi3K) Inhibitor Sf2558Ha
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.53 Å Release Date: 2017-02-08 Classification: TRANSCRIPTION REGULATOR/INHIBITOR Ligands: 82Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-08
Ligands: 82Y
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Brd4 First Bromodomain (Bd1) In Complex With Dual Pi3 Kinase (Pi3K) Inhibitor Sf2535
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2017-02-08 Classification: TRANSCRIPTION REGULATOR/INHIBITOR Ligands: 837 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-08
Ligands: 837
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Brd4 Second Bromodomain (Bd2) In Complex With Dual Pi3 Kinase (Pi3K) Inhibitor Sf2558Ha
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.30 Å Release Date: 2017-02-08 Classification: TRANSCRIPTION REGULATOR/INHIBITOR Ligands: 82Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-08
Ligands: 82Y
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Crystal Structure Of The First Bromodomain Of Human Brdt In Complex With The Inhibitor Jq1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.23 Å Release Date: 2012-07-11 Classification: TRANSCRIPTION REGULATOR/INHIBITOR Ligands: JQ1, K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-07-11
Ligands: JQ1, K
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Crebbp Bromodomain In Complex With Cpd3 ((S)-1-(3-(6-(1-Methyl-1H-Pyrazol-4-Yl)-3,4-Dihydroquinolin-1(2H)-Yl)-1-(Tetrahydrofuran-3-Yl)-1,4,6,7-Tetrahydro-5H-Pyrazolo[4,3-C]Pyridin-5-Yl)Ethan-1-One)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2018-03-07 Classification: TRANSCRIPTION REGULATOR/INHIBITOR Ligands: 9U7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-07
Ligands: 9U7
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Crebbp Bromodomain In Complex With Cpd17 (N,2,7-Trimethyl-2,3-Dihydro-4H-Benzo[B][1,4]Oxazine-4-Carboxamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2018-03-07 Classification: TRANSCRIPTION REGULATOR/INHIBITOR Ligands: SO4, 9UG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-07
Ligands: SO4, 9UG
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Crystal Structure Of Eed In Complex With Unc4859
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.74 Å Release Date: 2017-01-11 Classification: TRANSCRIPTION REGULATOR/INHIBITOR Ligands: SO4, UNX |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2017-01-11
Ligands: SO4, UNX
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Crebbp Bromodomain In Complex With Cpd19 (3-(7-(Difluoromethyl)-6-(1-Methyl-1H-Pyrazol-4-Yl)-3,4-Dihydroquinolin-1(2H)-Yl)-N-Methyl-1-(Tetrahydro-2H-Pyran-4-Yl)-1,4,6,7-Tetrahydro-5H-Pyrazolo[4,3-C]Pyridine-5-Carboxamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.41 Å Release Date: 2018-02-21 Classification: TRANSCRIPTION REGULATOR/INHIBITOR Ligands: 9U4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-02-21
Ligands: 9U4
 |
Structure Of Brd4 Bromodomain 1 With A 3-Methyl-4-Phenylisoxazol-5-Amine Fragment
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.29 Å Release Date: 2013-08-07 Classification: TRANSCRIPTION REGULATOR/INHIBITOR Ligands: FMT, 1XA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-08-07
Ligands: FMT, 1XA
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Structure Of Brd4 Bromodomain 1 With A Dimethyl Thiophene Isoxazole Azepine Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.21 Å Release Date: 2013-08-07 Classification: TRANSCRIPTION REGULATOR/INHIBITOR Ligands: 1XB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-08-07
Ligands: 1XB
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Brd4-Bd1 In Complex With Cpd19 (3-(7-(Difluoromethyl)-6-(1-Methyl-1H-Pyrazol-4-Yl)-3,4-Dihydroquinolin-1(2H)-Yl)-N-Methyl-1-(Tetrahydro-2H-Pyran-4-Yl)-1,4,6,7-Tetrahydro-5H-Pyrazolo[4,3-C]Pyridine-5-Carboxamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.71 Å Release Date: 2018-05-30 Classification: TRANSCRIPTION REGULATOR/INHIBITOR Ligands: EDO, 9U4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-30
Ligands: EDO, 9U4
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Crebbp Bromodomain In Complex With Cpd10 (1-(3-(7-(Difluoromethyl)-6-(1-Methyl-1H-Pyrazol-4-Yl)-3,4-Dihydroquinolin-1(2H)-Yl)-1-(Tetrahydro-2H-Pyran-4-Yl)-1,4,6,7-Tetrahydro-5H-Pyrazolo[4,3-C]Pyridin-5-Yl)Ethan-1-One)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2018-03-07 Classification: TRANSCRIPTION REGULATOR/INHIBITOR Ligands: 9UD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-07
Ligands: 9UD
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Bet Brd4-Bd1 In Complex With Peptide 9.2
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.47 Å Release Date: 2026-02-11 Classification: TRANSCRIPTION |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2026-02-11