Search Count: 160
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Complex Structure Of Trim24 Phd-Bromodomain And Inhibitor 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2017-02-22 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: ZN, 7FU, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: ZN, 7FU, DMS
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Complex Structure Of Trim24 Phd-Bromodomain And Inhibitor 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2017-02-22 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: ZN, 7FF, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: ZN, 7FF, DMS
 |
Complex Structure Of Trim24 Phd-Bromodomain And Inhibitor 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2017-02-22 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: 6KT, ZN, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: 6KT, ZN, DMS
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Crystal Structure Of Tead Complexed With Its Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.32 Å Release Date: 2020-07-01 Classification: transcription/transcription inhibitor Ligands: EY1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-01
Ligands: EY1
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Crystal Structure Of The Keap1 Kelch Domain In Complex With A Tetrapeptide
Organism: Homo sapiens, Enterobacteria phage t7
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2017-03-29 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: ACT |
Organism: Homo sapiens, Enterobacteria phage t7
Method: X-RAY DIFFRACTION
Release Date: 2017-03-29
Ligands: ACT
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Crystal Structure Of Tead2 Bound To Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.54 Å Release Date: 2020-06-24 Classification: Transcription/Transcription Inhibitor Ligands: GOL, QSJ, TRS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-06-24
Ligands: GOL, QSJ, TRS
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Crystal Structure Of Toxt From Vibrio Cholerae O395 Bound To (E)-4-(8-Methylnaphthalen-1-Yl)But-3-Enoic Acid
Organism: Vibrio cholerae
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2017-04-12 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: 70H, MES |
Organism: Vibrio cholerae
Method: X-RAY DIFFRACTION
Release Date: 2017-04-12
Ligands: 70H, MES
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Crystal Structure Of Chromodomain Of Cbx7 In Complex With Inhibitor Unc3866
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2015-12-16 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-12-16
Ligands: UNX
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A Multiconformer Ligand Model Of Inhibitor 53W Bound To Creb Binding Protein Bromodomain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.15 Å Release Date: 2018-12-19 Classification: transcription/transcription inhibitor Ligands: 53W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-12-19
Ligands: 53W
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Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With Ms436 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.20 Å Release Date: 2014-04-02 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: NUD, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: NUD, EDO
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Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With Ms267 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.30 Å Release Date: 2014-04-02 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: NUE, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: NUE, EDO
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Identification Of A Novel Allosteric Binding Site For Rorgt Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.08 Å Release Date: 2015-12-16 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: 4Y7, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-12-16
Ligands: 4Y7, GOL
 |
Identification Of A Novel Allosteric Binding Site For Rorgt Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2015-12-16 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: 4F1, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-12-16
Ligands: 4F1, GOL, SO4
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Identification Of A Novel Allosteric Binding Site For Rorgt Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2015-12-16 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: 4Y6, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-12-16
Ligands: 4Y6, SO4, GOL
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Identification Of A Novel Allosteric Binding Site For Rorgt Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.23 Å Release Date: 2015-12-16 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: 4Y5, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-12-16
Ligands: 4Y5, GOL
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Crystal Structure Of Phf1 Tudor Domain In Complex With A Peptidomimetic Ligand Unc6641
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2021-12-15 Classification: Transcription/Transcription Inhibitor Ligands: ZN, DMS |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2021-12-15
Ligands: ZN, DMS
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Stat3 Core In Complex With Compound Sd36
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2019-12-04 Classification: transcription/transcription inhibitor Ligands: KQV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-04
Ligands: KQV
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Stat3 Core In Complex With Compound Si109
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.15 Å Release Date: 2019-12-04 Classification: transcription/transcription inhibitor Ligands: KQV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-04
Ligands: KQV
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N-Terminal Bromodomain Of Human Brd2 In Complex With 4,4'-(Quinoline-5,7-Diyl)Bis(3,5-Dimethylisoxazole) Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2019-01-23 Classification: transcription/transcription inhibitor Ligands: JWD, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-01-23
Ligands: JWD, SO4
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N-Terminal Bromodomain Of Human Brd2 With N-((4-(3-(N-Cyclopentylsulfamoyl)-4-Methylphenyl)-3-Methylisoxazol-5-Yl)Methyl)Acetamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2019-01-23 Classification: transcription/transcription inhibitor Ligands: JWA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-01-23
Ligands: JWA