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5H1V image
Complex Structure Of Trim24 Phd-Bromodomain And Inhibitor 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.00 Å Release Date: 2017-02-22
Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR
Ligands: ZN, 7FU, DMS

5H1T image
Complex Structure Of Trim24 Phd-Bromodomain And Inhibitor 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.95 Å Release Date: 2017-02-22
Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR
Ligands: ZN, 7FF, DMS

5H1U image
Complex Structure Of Trim24 Phd-Bromodomain And Inhibitor 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.90 Å Release Date: 2017-02-22
Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR
Ligands: 6KT, ZN, DMS

6CDY image
Crystal Structure Of Tead Complexed With Its Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.32 Å Release Date: 2020-07-01
Classification: transcription/transcription inhibitor
Ligands: EY1

5X54 image
Crystal Structure Of The Keap1 Kelch Domain In Complex With A Tetrapeptide
Organism: Homo sapiens, Enterobacteria phage t7
Method: X-RAY DIFFRACTION
Resolution:2.30 Å Release Date: 2017-03-29
Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR
Ligands: ACT

6UYB image
Crystal Structure Of Tead2 Bound To Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.54 Å Release Date: 2020-06-24
Classification: Transcription/Transcription Inhibitor
Ligands: GOL, QSJ, TRS

5SUX image
Crystal Structure Of Toxt From Vibrio Cholerae O395 Bound To (E)-4-(8-Methylnaphthalen-1-Yl)But-3-Enoic Acid
Organism: Vibrio cholerae
Method: X-RAY DIFFRACTION
Resolution:2.00 Å Release Date: 2017-04-12
Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR
Ligands: 70H, MES

5EPJ image
Crystal Structure Of Chromodomain Of Cbx7 In Complex With Inhibitor Unc3866
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.60 Å Release Date: 2015-12-16
Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR
Ligands: UNX

6DMJ image
A Multiconformer Ligand Model Of Inhibitor 53W Bound To Creb Binding Protein Bromodomain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.15 Å Release Date: 2018-12-19
Classification: transcription/transcription inhibitor
Ligands: 53W

4NUE image
Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With Ms267 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.30 Å Release Date: 2014-04-02
Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR
Ligands: NUE, EDO

4NUD image
Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With Ms436 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.20 Å Release Date: 2014-04-02
Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR
Ligands: NUD, EDO

5C4O image
Identification Of A Novel Allosteric Binding Site For Rorgt Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.24 Å Release Date: 2015-12-16
Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR
Ligands: 4F1, GOL, SO4

5C4U image
Identification Of A Novel Allosteric Binding Site For Rorgt Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.08 Å Release Date: 2015-12-16
Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR
Ligands: 4Y7, GOL

5C4T image
Identification Of A Novel Allosteric Binding Site For Rorgt Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.77 Å Release Date: 2015-12-16
Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR
Ligands: 4Y6, SO4, GOL

5C4S image
Identification Of A Novel Allosteric Binding Site For Rorgt Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.23 Å Release Date: 2015-12-16
Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR
Ligands: 4Y5, GOL

7LKY image
Crystal Structure Of Phf1 Tudor Domain In Complex With A Peptidomimetic Ligand Unc6641
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Resolution:1.85 Å Release Date: 2021-12-15
Classification: Transcription/Transcription Inhibitor
Ligands: ZN, DMS

6NUQ image
Stat3 Core In Complex With Compound Si109
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:3.15 Å Release Date: 2019-12-04
Classification: transcription/transcription inhibitor
Ligands: KQV

6NJS image
Stat3 Core In Complex With Compound Sd36
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.70 Å Release Date: 2019-12-04
Classification: transcription/transcription inhibitor
Ligands: KQV

6MO8 image
N-Terminal Bromodomain Of Human Brd2 In Complex With 4,4'-(Quinoline-5,7-Diyl)Bis(3,5-Dimethylisoxazole) Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.80 Å Release Date: 2019-01-23
Classification: transcription/transcription inhibitor
Ligands: JWD, SO4

6MO7 image
N-Terminal Bromodomain Of Human Brd2 With N-((4-(3-(N-Cyclopentylsulfamoyl)-4-Methylphenyl)-3-Methylisoxazol-5-Yl)Methyl)Acetamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.85 Å Release Date: 2019-01-23
Classification: transcription/transcription inhibitor
Ligands: JWA
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