Search Count: 15
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Crystal Structure Of Human Pyruvate Dehydrogenase Kinase Isoform 1 In Complex With Atp Competitive Inhibitor 29
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.14 Å Release Date: 2025-06-25 Classification: TRANSFERASE Ligands: SO4, TF3, EDO, GOL, A1EQH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-06-25
Ligands: SO4, TF3, EDO, GOL, A1EQH
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Crystal Structure Of Human Pyruvate Dehydrogenase Kinase Isoform 2 In Complex With Atp Competitive Inhibitor 24
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.92 Å Release Date: 2025-06-25 Classification: TRANSFERASE Ligands: EDO, TF3, GOL, A1EQJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-06-25
Ligands: EDO, TF3, GOL, A1EQJ
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Crystal Structure Of Human Pyruvate Dehydrogenase Kinase Isoform 2 In Complex With Atp Competitive Inhibitor 22
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.08 Å Release Date: 2025-06-11 Classification: TRANSFERASE Ligands: TF3, A1EQI, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-06-11
Ligands: TF3, A1EQI, DMS
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Rapid Optimisation Of Fragments And Hits To Lead Compounds From Screening Of Crude Reaction Mixtures
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.08 Å Release Date: 2020-10-14 Classification: TRANSFERASE Ligands: MG, NN8, TF3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-10-14
Ligands: MG, NN8, TF3
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Rapid Optimisation Of Fragments And Hits To Lead Compounds From Screening Of Crude Reaction Mixtures
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.11 Å Release Date: 2020-10-14 Classification: TRANSFERASE Ligands: TF3, NMW, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-10-14
Ligands: TF3, NMW, DMS
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Rapid Optimisation Of Fragments And Hits To Lead Compounds From Screening Of Crude Reaction Mixtures
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.71 Å Release Date: 2020-10-14 Classification: TRANSFERASE Ligands: TF3, MG, NN8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-10-14
Ligands: TF3, MG, NN8
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Rapid Optimisation Of Fragments And Hits To Lead Compounds From Screening Of Crude Reaction Mixtures
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.91 Å Release Date: 2020-10-14 Classification: TRANSFERASE Ligands: TF3, NLZ, DMS, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-10-14
Ligands: TF3, NLZ, DMS, CL
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Rapid Optimisation Of Fragments And Hits To Lead Compounds From Screening Of Crude Reaction Mixtures
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2020-10-14 Classification: TRANSFERASE Ligands: TF3, NL8, DMS, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-10-14
Ligands: TF3, NL8, DMS, CL
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Application Of Off-Rate Screening In The Identification Of Novel Pan-Isoform Inhibitors Of Pyruvate Dehydrogenase Kinase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2017-02-22 Classification: TRANSFERASE Ligands: TF3, 7F9, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: TF3, 7F9, MG
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Application Of Off-Rate Screening In The Identification Of Novel Pan-Isoform Inhibitors Of Pyruvate Dehydrogenase Kinase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2017-02-22 Classification: TRANSFERASE Ligands: 7FW, TF3, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: 7FW, TF3, CL
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Application Of Off-Rate Screening In The Identification Of Novel Pan-Isoform Inhibitors Of Pyruvate Dehydrogenase Kinase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2017-02-22 Classification: TRANSFERASE Ligands: 7FV, TF3, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: 7FV, TF3, CL
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Application Of Off-Rate Screening In The Identification Of Novel Pan-Isoform Inhibitors Of Pyruvate Dehydrogenase Kinase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2017-02-22 Classification: TRANSFERASE Ligands: 7FE, TF3, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: 7FE, TF3, CL
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Ver-246608, A Novel Pan-Isoform Atp Competitive Inhibitor Of Pyruvate Dehydrogenase Kinase, Disrupts Warburg Metabolism And Induces Context- Dependent Cytostasis In Cancer Cells
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2014-12-03 Classification: TRANSFERASE Ligands: TF3, MG, SZ6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-03
Ligands: TF3, MG, SZ6
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Ver-246608, A Novel Pan-Isoform Atp Competitive Inhibitor Of Pyruvate Dehydrogenase Kinase, Disrupts Warburg Metabolism And Induces Context- Dependent Cytostasis In Cancer Cells
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2014-12-03 Classification: TRANSFERASE Ligands: TF3, MG, 7TJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-03
Ligands: TF3, MG, 7TJ
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Crystal Structures Of Human Pyruvate Dehydrogenase Kinase 2 Containing Physiological And Synthetic Ligands
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2006-02-02 Classification: TRANSFERASE Ligands: TF3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-02-02
Ligands: TF3