Search Count: 39
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Crystal Structure Of The Human Dcaf1 Wdr Domain In Complex With Oicr-41109
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2025-11-26 Classification: TRANSPORT PROTEIN Ligands: A1CY9, NA, UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-11-26
Ligands: A1CY9, NA, UNX
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Crystal Structure Of Setdb1 Tudor Domain In Complex With Unc100013
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.53 Å Release Date: 2024-10-02 Classification: TRANSFERASE Ligands: A1AZ6, EDO, UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-02
Ligands: A1AZ6, EDO, UNX
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Crystal Structure Of Setdb1 Tudor Domain In Complex With Unc100016
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.27 Å Release Date: 2024-10-02 Classification: TRANSFERASE Ligands: A1AZ5, SO4, EDO, UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-02
Ligands: A1AZ5, SO4, EDO, UNX
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Cryoem Structure Of Human Ddb1-Dcaf12 In Complex With Magea3
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Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2024-04-10
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Tead2 With A Covalent Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2023-12-13 Classification: SIGNALING PROTEIN Ligands: MYR, B3F |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-13
Ligands: MYR, B3F
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Tead2 With A Covalent Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2023-12-13 Classification: SIGNALING PROTEIN Ligands: F3Y, MYR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-13
Ligands: F3Y, MYR
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Structure Of Hdac6 Zinc-Finger Ubiquitin Binding Domain In Complex With 3-(3-(2-(Methylamino)-2-Oxoethyl)-4-Oxo-3,4-Dihydroquinazolin-2-Yl)Propanoic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2023-05-03 Classification: HYDROLASE/INHIBITOR Ligands: ZN, ZU6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-05-03
Ligands: ZN, ZU6
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Structure Of Hdac6 Zinc-Finger Ubiquitin Binding Domain In Complex With 3-(3-(2-(Benzylamino)-2-Oxoethyl)-4-Oxo-3,4-Dihydroquinazolin-2-Yl)Propanoic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2023-05-03 Classification: HYDROLASE/INHIBITOR Ligands: ZN, ZU9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-05-03
Ligands: ZN, ZU9
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Structure Of Hdac6 Zinc-Finger Ubiquitin Binding Domain In Complex With Sgc-Ubd253 Chemical Probe
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.62 Å Release Date: 2023-05-03 Classification: HYDROLASE/INHIBITOR Ligands: ZN, ZUE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-05-03
Ligands: ZN, ZUE
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Crystal Structure Of The Wdr Domain Of Human Dcaf1 In Complex With Oicr-6766
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2022-05-04 Classification: TRANSFERASE Ligands: N6O, UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-05-04
Ligands: N6O, UNX
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X-Ray Structure Of Smyd3 In Complex With Benzodiazepine-Type Inhibitor Compound 15
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.57 Å Release Date: 2021-07-07 Classification: TRANSFERASE Ligands: UZT, SAM, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: UZT, SAM, ZN
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X-Ray Structure Of Smyd3 In Complex With Benzodiazepine-Type Inhibitor 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.03 Å Release Date: 2021-07-07 Classification: TRANSFERASE Ligands: UZQ, ZN, SAM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: UZQ, ZN, SAM
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X-Ray Structure Of Smyd3 In Complex With The Benzodiazepine-Based Probe Bay-6035
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.52 Å Release Date: 2021-07-07 Classification: TRANSFERASE Ligands: UZK, SAM, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: UZK, SAM, ZN
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Histone-Lysine N-Methyltransferase Nsd2-Pwwp1 With Compound Mrt10241866A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.42 Å Release Date: 2021-05-05 Classification: TRANSFERASE Ligands: Y6V, UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-05
Ligands: Y6V, UNX
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Histone-Lysine N-Methyltransferase Nsd2-Pwwp1 With Compound Unc6934
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.64 Å Release Date: 2020-07-22 Classification: TRANSFERASE Ligands: V01, UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-22
Ligands: V01, UNX
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High Resolution Cryoem Structure Of Huntingtin In Complex With Hap40
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2020-06-17 Classification: PROTEIN BINDING |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2020-06-17
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Crystal Structure Of Human Protein Arginine N-Methyltransferase 6 (Prmt6) In Complex With Sgc6870 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.91 Å Release Date: 2020-04-29 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: SAH, T9A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-29
Ligands: SAH, T9A
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Pwwp1 Domain Of Nsd2 In Complex With Mr837
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2019-11-13 Classification: TRANSFERASE Ligands: Q5D, UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-13
Ligands: Q5D, UNX
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X-Ray Structure Of Nsd3-Pwwp1 In Complex With Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2019-06-26 Classification: ONCOPROTEIN Ligands: EH2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-26
Ligands: EH2
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X-Ray Structure Of Nsd3-Pwwp1 In Complex With Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.43 Å Release Date: 2019-06-26 Classification: ONCOPROTEIN Ligands: EHQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-26
Ligands: EHQ
