Search Count: 38
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Discovery Of Vx-509 (Decernotinib): A Potent And Selective Janus Kinase (Jak) 3 Inhibitor For The Treatment Of Autoimmune Disease
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.16 Å Release Date: 2015-08-12 Classification: Transferase/Transferase Inhibitor Ligands: 4HW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-12
Ligands: 4HW
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Discovery Of Vx-509 (Decernotinib): A Potent And Selective Janus Kinase (Jak) 3 Inhibitor For The Treatment Of Autoimmune Diseases
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.78 Å Release Date: 2015-08-12 Classification: Transferase/Transferase Inhibitor Ligands: 4HZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-12
Ligands: 4HZ
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Discovery Of Vx-509 (Decernotinib): A Potent And Selective Janus Kinase (Jak) 3 Inhibitor For The Treatment Of Autoimmune Diseases
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2015-08-12 Classification: Transferase/Transferase Inhibitor Ligands: 467 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-12
Ligands: 467
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Discovery Of Vx-509 (Decernotinib): A Potent And Selective Janus Kinase (Jak) 3 Inhibitor For The Treatment Of Autoimmune Disease
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.52 Å Release Date: 2015-08-12 Classification: Transferase/Transferase Inhibitor Ligands: VJK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-12
Ligands: VJK
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Crystal Structure Of The Ectodomain Complex Of The Cgrp Receptor, A Class-B Gpcr, Reveals The Site Of Drug Antagonism
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2010-09-15 Classification: MEMBRANE PROTEIN Ligands: SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-09-15
Ligands: SO4
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Crystal Structure Of The Ectodomain Complex Of The Cgrp Receptor, A Class-B Gpcr, Reveals The Site Of Drug Antagonism
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2010-09-15 Classification: MEMBRANE PROTEIN Ligands: 3N6, N7R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-09-15
Ligands: 3N6, N7R
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Crystal Structure Of The Ectodomain Complex Of The Cgrp Receptor, A Class-B Gpcr, Reveals The Site Of Drug Antagonism
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2010-09-15 Classification: MEMBRANE PROTEIN Ligands: 3N6, 3N7, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-09-15
Ligands: 3N6, 3N7, SO4
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2-Aminopyrazolo[1,5-A]Pyrimidines As Potent And Selective Inhibitors Of Jak2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2009-11-10 Classification: TRANSFERASE Ligands: 1P5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-11-10
Ligands: 1P5
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2-Aminopyrazolo[1,5-A]Pyrimidines As Potent And Selective Inhibitors Of Jak2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2009-11-10 Classification: TRANSFERASE Ligands: 1P6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-11-10
Ligands: 1P6
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Crystal Structure Of Rock I Bound To H-1152P A Di-Methylated Variant Of Fasudil
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.30 Å Release Date: 2008-06-10 Classification: TRANSFERASE Ligands: H52 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-06-10
Ligands: H52
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Crystal Structure Of Hcv Ns3-4A R155K Mutant
Organism: Hepatitis c virus, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2007-06-05 Classification: HYDROLASE Ligands: ZN |
Organism: Hepatitis c virus, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2007-06-05
Ligands: ZN
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Crystal Structure Of C-Amp Dependent Kinase (Pka) Bound To Hydroxyfasudil
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2005-11-08 Classification: TRANSFERASE Ligands: HFS |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2005-11-08
Ligands: HFS
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Crystal Structure Of Rock 1 Bound To Fasudil
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.20 Å Release Date: 2005-11-08 Classification: TRANSFERASE Ligands: M77 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-11-08
Ligands: M77
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Crystal Structure Of Rock 1 Bound To Hydroxyfasudil
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.96 Å Release Date: 2005-11-08 Classification: TRANSFERASE Ligands: HFS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-11-08
Ligands: HFS
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Crystal Structure Of Rock I Bound To Y-27632
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2005-11-08 Classification: TRANSFERASE Ligands: Y27 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-11-08
Ligands: Y27
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Crystal Structure Of Pim-1 Bound To Staurosporine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2005-01-25 Classification: TRANSFERASE Ligands: STU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-01-25
Ligands: STU
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Crystal Structure Of Pim-1 Bound To Ly294002
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2005-01-25 Classification: TRANSFERASE Ligands: LY2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-01-25
Ligands: LY2
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Structure Of Pim-1 Bound To Adenosine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2005-01-25 Classification: TRANSFERASE Ligands: ADN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-01-25
Ligands: ADN
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Crystal Structure Of Escherichia Coli Topoisomerase Iv Pare 24Kda Subunit
Organism: Escherichia coli
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2004-05-04 Classification: ISOMERASE Ligands: NOV |
Organism: Escherichia coli
Method: X-RAY DIFFRACTION
Release Date: 2004-05-04
Ligands: NOV
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Crystal Structure Of E. Coli Topoisomerase Iv Pare 43Kda Subunit Complexed With Adpnp
Organism: Escherichia coli
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2004-05-04 Classification: ISOMERASE Ligands: MG, SO4, ANP |
Organism: Escherichia coli
Method: X-RAY DIFFRACTION
Release Date: 2004-05-04
Ligands: MG, SO4, ANP
