Search Count: 20
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Qr2 Inhibitor From A Novel Sulfanamide Series To Tackle Age Related Oxidative Stress And Cognitive Decline
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2022-08-17 Classification: OXIDOREDUCTASE Ligands: ZN, FAD, SO4, V1Z |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-17
Ligands: ZN, FAD, SO4, V1Z
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Crystal Structure Of Human Naa50 In Complex With A Cofactor Derived Inhibitor (Compound 1)
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.29 Å Release Date: 2020-07-01 Classification: TRANSFERASE/INHIBITOR Ligands: COA |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2020-07-01
Ligands: COA
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Crystal Structure Of Human Naa50 In Complex With A Truncated Cofactor Derived Inhibitor (Compound 2)
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2020-07-01 Classification: TRANSFERASE/INHIBITOR Ligands: U44 |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2020-07-01
Ligands: U44
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Crystal Structure Of Human Naa50 In Complex With An Inhibitor (Compound 3) Identified Using Dna Encoded Library Technology
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.16 Å Release Date: 2020-07-01 Classification: TRANSFERASE/INHIBITOR Ligands: COA, U3V |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-01
Ligands: COA, U3V
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Crystal Structure Of Human Naa50 In Complex With Coa And An Inhibitor (Compound 4A) Identified Using Dna Encoded Library Technology
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.87 Å Release Date: 2020-07-01 Classification: TRANSFERASE Ligands: COA, U2J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-01
Ligands: COA, U2J
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Crystal Structure Of Human Naa50 In Complex With Accoa And An Inhibitor (Compound 4A) Identified Using Dna Encoded Library Technology
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.07 Å Release Date: 2020-07-01 Classification: TRANSFERASE/INHIBITOR Ligands: ACO, U2J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-01
Ligands: ACO, U2J
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Crystal Structure Of Human Naa50 In Complex With Accoa And An Inhibitor (Compound 4B) Identified Using Dna Encoded Library Technology
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2020-07-01 Classification: TRANSFERASE/INHIBITOR Ligands: ACO, U3Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-01
Ligands: ACO, U3Y
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Map2K7 C276S Mutant-Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.28 Å Release Date: 2019-01-02 Classification: TRANSFERASE Ligands: 95U, EPE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-01-02
Ligands: 95U, EPE
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Map2K7 C218S Mutant-Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2019-01-02 Classification: TRANSFERASE Ligands: 95U |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-01-02
Ligands: 95U
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Identification And Profiling Of A Selective And Brain Penetrant Radioligand For In Vivo Target Occupancy Measurement Of Casein Kinase 1 (Ck1) Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2017-06-28 Classification: TRANSFERASE/INHIBITOR Ligands: 9WG, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-28
Ligands: 9WG, SO4
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Crystal Structure Of Tubulin-Stathmin-Ttl-Compound 11 Complex
Organism: Rattus norvegicus, Gallus gallus, Ovis aries
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2016-12-28 Classification: STRUCTURAL PROTEIN/INHIBITOR Ligands: GTP, MG, CA, GDP, 6YK, ADP |
Organism: Rattus norvegicus, Gallus gallus, Ovis aries
Method: X-RAY DIFFRACTION
Release Date: 2016-12-28
Ligands: GTP, MG, CA, GDP, 6YK, ADP
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Discovery Of Cytotoxic Dolastatin 10 Analogs With N-Terminal Modifications
Organism: Rattus norvegicus, Ovis aries
Method: X-RAY DIFFRACTION Resolution:3.11 Å Release Date: 2015-03-25 Classification: STRUCTURAL PROTEIN/INHIBITOR Ligands: GTP, MG, GDP, LOC, 3WD |
Organism: Rattus norvegicus, Ovis aries
Method: X-RAY DIFFRACTION
Release Date: 2015-03-25
Ligands: GTP, MG, GDP, LOC, 3WD
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Discovery Of Cytotoxic Dolastatin 10 Analogs With N-Terminal Modifications
Organism: Rattus norvegicus, Ovis aries
Method: X-RAY DIFFRACTION Resolution:3.50 Å Release Date: 2015-03-25 Classification: Structural Protein/Inhibitor Ligands: GTP, MG, GDP, LOC, 3WZ |
Organism: Rattus norvegicus, Ovis aries
Method: X-RAY DIFFRACTION
Release Date: 2015-03-25
Ligands: GTP, MG, GDP, LOC, 3WZ
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Discovery Of Cytotoxic Dolastatin 10 Analogs With N-Terminal Modifications
Organism: Rattus norvegicus, Ovis aries
Method: X-RAY DIFFRACTION Resolution:3.19 Å Release Date: 2015-03-25 Classification: Structural Protein/Inhibitor Ligands: GTP, MG, GDP, LOC, 3WV |
Organism: Rattus norvegicus, Ovis aries
Method: X-RAY DIFFRACTION
Release Date: 2015-03-25
Ligands: GTP, MG, GDP, LOC, 3WV
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Discovery Of Cytotoxic Dolastatin 10 Analogs With N-Terminal Modifications
Organism: Rattus norvegicus, Ovis aries
Method: X-RAY DIFFRACTION Resolution:3.50 Å Release Date: 2015-03-25 Classification: Structural Protein/Inhibitor Ligands: GTP, MG, GDP, LOC, 3WY |
Organism: Rattus norvegicus, Ovis aries
Method: X-RAY DIFFRACTION
Release Date: 2015-03-25
Ligands: GTP, MG, GDP, LOC, 3WY
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Crystal Structure Of Akt-1-Inhibitor Complexes
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.47 Å Release Date: 2010-06-02 Classification: TRANSFERASE Ligands: MN, XFE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-06-02
Ligands: MN, XFE
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Crystal Structure Of Akt-1-Inhibitor Complexes
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.01 Å Release Date: 2010-06-02 Classification: TRANSFERASE Ligands: MN, WFE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-06-02
Ligands: MN, WFE
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Human Cyclic Amp-Dependent Protein Kinase Pka Inhibitor Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2010-06-02 Classification: TRANSFERASE Ligands: XFE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-06-02
Ligands: XFE
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Staphylococcus Aureus S1:Dhfr
Organism: Staphylococcus aureus
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2009-03-24 Classification: OXIDOREDUCTASE |
Organism: Staphylococcus aureus
Method: X-RAY DIFFRACTION
Release Date: 2009-03-24
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Crystal Structure Of The Catalytic Domain Of Mmp-13 Complexed With A Potent Pyrimidinetrione Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2005-03-15 Classification: HYDROLASE Ligands: ZN, CA, SO4, PFD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-03-15
Ligands: ZN, CA, SO4, PFD